FI832960A7 - Menetelmä angiotensiiniä muuttavan entsyymin inhibiittorien valmistamiseksi. - Google Patents

Menetelmä angiotensiiniä muuttavan entsyymin inhibiittorien valmistamiseksi. Download PDF

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Publication number
FI832960A7
FI832960A7 FI832960A FI832960A FI832960A7 FI 832960 A7 FI832960 A7 FI 832960A7 FI 832960 A FI832960 A FI 832960A FI 832960 A FI832960 A FI 832960A FI 832960 A7 FI832960 A7 FI 832960A7
Authority
FI
Finland
Prior art keywords
converting enzyme
enzyme inhibitors
preparing angiotensin
angiotensin
preparing
Prior art date
Application number
FI832960A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI832960L (fi
FI832960A0 (fi
Inventor
Walter Mitsuo Nakatsukasa
Jon Stuart Mynderse
Sean Christopher O'connor
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US06/409,764 external-priority patent/US4404282A/en
Priority claimed from US06/409,763 external-priority patent/US4508901A/en
Priority claimed from US06/409,765 external-priority patent/US4404281A/en
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of FI832960A0 publication Critical patent/FI832960A0/fi
Publication of FI832960L publication Critical patent/FI832960L/fi
Publication of FI832960A7 publication Critical patent/FI832960A7/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/02Oxygen as only ring hetero atoms
    • C12P17/04Oxygen as only ring hetero atoms containing a five-membered hetero ring, e.g. griseofulvin, vitamin C
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/02Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing not further condensed quinolizine ring systems
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12NMICROORGANISMS OR ENZYMES; COMPOSITIONS THEREOF; PROPAGATING, PRESERVING, OR MAINTAINING MICROORGANISMS; MUTATION OR GENETIC ENGINEERING; CULTURE MEDIA
    • C12N1/00Microorganisms, e.g. protozoa; Compositions thereof; Processes of propagating, maintaining or preserving microorganisms or compositions thereof; Processes of preparing or isolating a composition containing a microorganism; Culture media therefor
    • C12N1/20Bacteria; Culture media therefor
    • C12N1/205Bacterial isolates
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/18Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms containing at least two hetero rings condensed among themselves or condensed with a common carbocyclic ring system, e.g. rifamycin
    • C12P17/182Heterocyclic compounds containing nitrogen atoms as the only ring heteroatoms in the condensed system
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12RINDEXING SCHEME ASSOCIATED WITH SUBCLASSES C12C - C12Q, RELATING TO MICROORGANISMS
    • C12R2001/00Microorganisms ; Processes using microorganisms
    • C12R2001/01Bacteria or Actinomycetales ; using bacteria or Actinomycetales
    • C12R2001/465Streptomyces

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Health & Medical Sciences (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Microbiology (AREA)
  • Biochemistry (AREA)
  • General Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Virology (AREA)
  • Biomedical Technology (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Micro-Organisms Or Cultivation Processes Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
FI832960A 1982-08-19 1983-08-18 Menetelmä angiotensiiniä muuttavan entsyymin inhibiittorien valmistamiseksi. FI832960A7 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/409,764 US4404282A (en) 1982-08-19 1982-08-19 Process for enzyme inhibitor
US06/409,763 US4508901A (en) 1982-08-19 1982-08-19 Quiuolizine and indolizine enzyme inhibitors
US06/409,765 US4404281A (en) 1982-08-19 1982-08-19 Process for enzyme inhibitors

Publications (3)

Publication Number Publication Date
FI832960A0 FI832960A0 (fi) 1983-08-18
FI832960L FI832960L (fi) 1984-02-20
FI832960A7 true FI832960A7 (fi) 1984-02-20

Family

ID=27410818

Family Applications (1)

Application Number Title Priority Date Filing Date
FI832960A FI832960A7 (fi) 1982-08-19 1983-08-18 Menetelmä angiotensiiniä muuttavan entsyymin inhibiittorien valmistamiseksi.

Country Status (15)

Country Link
EP (1) EP0103403B1 (Direct)
KR (1) KR860001215B1 (Direct)
AU (1) AU560417B2 (Direct)
DD (1) DD218389A5 (Direct)
DE (1) DE3381244D1 (Direct)
DK (1) DK377883A (Direct)
ES (1) ES8505721A1 (Direct)
FI (1) FI832960A7 (Direct)
GB (1) GB2126217B (Direct)
GR (1) GR78665B (Direct)
IL (1) IL69474A (Direct)
NZ (1) NZ205245A (Direct)
PL (1) PL243461A1 (Direct)
PT (1) PT77190B (Direct)
SU (1) SU1403991A3 (Direct)

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4316906A (en) * 1978-08-11 1982-02-23 E. R. Squibb & Sons, Inc. Mercaptoacyl derivatives of substituted prolines
US4316905A (en) * 1980-07-01 1982-02-23 E. R. Squibb & Sons, Inc. Mercaptoacyl derivatives of various 4-substituted prolines

Also Published As

Publication number Publication date
FI832960L (fi) 1984-02-20
FI832960A0 (fi) 1983-08-18
KR860001215B1 (ko) 1986-08-27
PL243461A1 (en) 1985-01-02
GB2126217A (en) 1984-03-21
DE3381244D1 (de) 1990-04-05
EP0103403B1 (en) 1990-02-28
EP0103403A3 (en) 1986-07-02
SU1403991A3 (ru) 1988-06-15
ES524874A0 (es) 1985-06-01
EP0103403A2 (en) 1984-03-21
DK377883A (da) 1984-02-20
AU560417B2 (en) 1987-04-09
IL69474A (en) 1986-11-30
AU1790483A (en) 1984-02-23
GR78665B (Direct) 1984-09-27
NZ205245A (en) 1987-01-23
DK377883D0 (da) 1983-08-18
ES8505721A1 (es) 1985-06-01
DD218389A5 (de) 1985-02-06
GB2126217B (en) 1986-04-03
IL69474A0 (en) 1983-11-30
PT77190B (en) 1986-03-20
PT77190A (en) 1983-09-01
KR840005743A (ko) 1984-11-15
GB8321679D0 (en) 1983-09-14

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Owner name: ELI LILLY AND COMPANY