FI783417A - Nya 9-(omega-heteroarylamino-alkylamino)-erytromyciner deras salter deras framstaellningsfoerfarande och dessa innehaollande laekemedel - Google Patents

Nya 9-(omega-heteroarylamino-alkylamino)-erytromyciner deras salter deras framstaellningsfoerfarande och dessa innehaollande laekemedel

Info

Publication number
FI783417A
FI783417A FI783417A FI783417A FI783417A FI 783417 A FI783417 A FI 783417A FI 783417 A FI783417 A FI 783417A FI 783417 A FI783417 A FI 783417A FI 783417 A FI783417 A FI 783417A
Authority
FI
Finland
Prior art keywords
deras
erytromyciner
nya
heteroarylamino
omega
Prior art date
Application number
FI783417A
Other languages
English (en)
Inventor
Eberhard Woitun
Bernd Wetzel
Roland Maier
Wolfgang Reuter
Uwe Lechner
Rolf G Werner
Hanns Goeth
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of FI783417A publication Critical patent/FI783417A/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
FI783417A 1977-11-10 1978-11-09 Nya 9-(omega-heteroarylamino-alkylamino)-erytromyciner deras salter deras framstaellningsfoerfarande och dessa innehaollande laekemedel FI783417A (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772750288 DE2750288A1 (de) 1977-11-10 1977-11-10 Neue 9-(omega-heteroarylamino- alkylamino)-erythromycine, ihre salze, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
FI783417A true FI783417A (fi) 1979-05-11

Family

ID=6023435

Family Applications (1)

Application Number Title Priority Date Filing Date
FI783417A FI783417A (fi) 1977-11-10 1978-11-09 Nya 9-(omega-heteroarylamino-alkylamino)-erytromyciner deras salter deras framstaellningsfoerfarande och dessa innehaollande laekemedel

Country Status (18)

Country Link
US (1) US4256738A (fi)
EP (1) EP0001981B1 (fi)
JP (1) JPS5476588A (fi)
AT (1) AT361623B (fi)
AU (1) AU4144878A (fi)
CA (1) CA1107726A (fi)
DE (2) DE2750288A1 (fi)
DK (1) DK499778A (fi)
ES (1) ES474693A1 (fi)
FI (1) FI783417A (fi)
GR (1) GR65281B (fi)
IL (1) IL55906A0 (fi)
IT (1) IT1109331B (fi)
NO (1) NO783767L (fi)
NZ (1) NZ188872A (fi)
PT (1) PT68771A (fi)
YU (1) YU261178A (fi)
ZA (1) ZA786313B (fi)

Families Citing this family (38)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2473525A1 (fr) * 1980-01-11 1981-07-17 Roussel Uclaf Nouvelles oximes derivees de l'erythromycine, leur procede de preparation et leur application comme medicaments
US5110800A (en) * 1986-02-18 1992-05-05 Eli Lilly And Company Derivatives of erythromycylamine
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
TW440563B (en) * 1996-05-23 2001-06-16 Hoffmann La Roche Aryl pyrimidine derivatives and a pharmaceutical composition thereof
US5958934A (en) * 1996-05-23 1999-09-28 Syntex (U.S.A.) Inc. Aryl pyrimidine derivatives and uses thereof
US5952331A (en) * 1996-05-23 1999-09-14 Syntex (Usa) Inc. Aryl pyrimidine derivatives
US5739127A (en) * 1996-11-08 1998-04-14 Bayer Aktiengesellschaft 2,4'-bridged bis-2,4-diaminoquinazolines
WO2003002064A2 (en) * 2001-06-28 2003-01-09 Essential Therapeutics, Inc. Fused pyrimidine dhfr inhibitors as antibacterials
AR059898A1 (es) 2006-03-15 2008-05-07 Janssen Pharmaceutica Nv Derivados de 3-ciano-piridona 1,4-disustituida y su uso como moduladores alostericos de los receptores mglur2
EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
BRPI0608387A2 (pt) * 2006-04-19 2009-12-29 Boehringer Ingelheim Int compostos para o tratamento de doenças inflamatórias
TW200845978A (en) * 2007-03-07 2008-12-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-tetrahydropyran-phenyl)-pyridin-2-one derivatives
TW200900065A (en) 2007-03-07 2009-01-01 Janssen Pharmaceutica Nv 3-cyano-4-(4-pyridinyloxy-phenyl)-pyridin-2-one derivatives
BRPI0816767B8 (pt) * 2007-09-14 2021-05-25 Addex Pharmaceuticals Sa composto 4-fenil-3,4,5,6-tetra-hidro-2h,1'h-[1,4']bipiridi¬nil-2'-onas 1',3'-dissubstituídas, composição farmacêutica e uso dos mesmos
AU2008297876B2 (en) 2007-09-14 2011-07-07 Addex Pharma S.A. 1,3-disubstituted 4-(aryl-x-phenyl)-1h-pyridin-2-ones
CN101801930B (zh) * 2007-09-14 2013-01-30 奥梅-杨森制药有限公司 1,3-二取代的-4-苯基-1h-吡啶-2-酮
ES2381452T3 (es) * 2007-10-19 2012-05-28 Boehringer Ingelheim International Gmbh PIPERIDINO-DIHIDROTIENOPIRIMIDINAS sustituidas
JP5563466B2 (ja) 2007-10-19 2014-07-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ピペラジノ−ジヒドロチエノピリミジン誘導体
BRPI0817781A2 (pt) * 2007-10-19 2019-09-24 Boehringer Ingelheim Int piperazino-diidroteinopirimidinas substituídas com heterociclo
ES2637794T3 (es) * 2007-11-14 2017-10-17 Janssen Pharmaceuticals, Inc. Derivados de imidazo[1,2-A]piridina y su uso como moduladores alostéricos positivos de receptores MGLUR2
AU2009289784B2 (en) 2008-09-02 2012-03-22 Addex Pharma S.A. 3-azabicyclo[3.1.0]hexyl derivatives as modulators of metabotropic glutamate receptors
WO2010043396A1 (en) 2008-10-16 2010-04-22 Ortho-Mcneil-Janssen Pharmaceuticals, Inc. Indole and benzomorpholine derivatives as modulators of metabotropic glutamate receptors
WO2010060589A1 (en) 2008-11-28 2010-06-03 Ortho-Mcneil-Janssen Pharmaceuticals, Inc. Indole and benzoxazine derivatives as modulators of metabotropic glutamate receptors
MY161325A (en) 2009-05-12 2017-04-14 Janssen Pharmaceuticals Inc 1, 2, 4-triazolo[4,3-a]pyridine derivatives and their use for the treatment or prevention of neurological and psychiatric disorders
US8946205B2 (en) 2009-05-12 2015-02-03 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
MY153913A (en) 2009-05-12 2015-04-15 Janssen Pharmaceuticals Inc 7-aryl-1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mglur2 receptors
PL2649069T3 (pl) 2010-11-08 2016-01-29 Janssen Pharmaceuticals Inc Pochodne 1,2,4-triazolo[4,3-a]pirydyny i ich zastosowanie jako dodatnich allosterycznych modulatorów receptorów mGluR2
CN103261195B (zh) 2010-11-08 2015-09-02 杨森制药公司 1,2,4-三唑并[4,3-a]吡啶衍生物及其作为MGLUR2受体的正变构调节剂的用途
AU2011328203B2 (en) 2010-11-08 2015-03-19 Janssen Pharmaceuticals, Inc. 1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive allosteric modulators of mGluR2 receptors
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
JO3368B1 (ar) 2013-06-04 2019-03-13 Janssen Pharmaceutica Nv مركبات 6، 7- ثاني هيدرو بيرازولو [5،1-a] بيرازين- 4 (5 يد)- اون واستخدامها بصفة منظمات تفارغية سلبية لمستقبلات ميجلور 2
JO3367B1 (ar) 2013-09-06 2019-03-13 Janssen Pharmaceutica Nv مركبات 2،1، 4- ثلاثي زولو [3،4-a] بيريدين واستخدامها بصفة منظمات تفارغية موجبة لمستقبلات ميجلور 2
CA2925211A1 (en) * 2013-09-27 2015-04-02 Nimbus Iris, Inc. Irak inhibitors and uses thereof
UA121965C2 (uk) 2014-01-21 2020-08-25 Янссен Фармацевтика Нв Комбінації, які містять позитивні алостеричні модулятори або ортостеричні агоністи метаботропного глутаматергічного рецептора 2 підтипу, та їх застосування
KR102461134B1 (ko) 2014-01-21 2022-10-28 얀센 파마슈티카 엔.브이. 대사 조절형 글루탐산 작동성 수용체 제2아형의 양성 알로스테릭 조절제 또는 오르토스테릭 작동제를 포함하는 조합 및 그 용도
CN106674132B (zh) * 2016-11-22 2019-04-26 上海书亚医药科技有限公司 一种嘧啶类除草剂的制备方法与应用
CN112569239B (zh) * 2020-12-18 2021-12-28 北京鑫开元医药科技有限公司 作为tlr8激动剂的药物组合物、其制备方法及其用途

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3650376A (en) * 1970-08-17 1972-03-21 Conveyor Systems Accumulating conveyor
GB1345524A (en) * 1970-09-30 1974-01-30 Lilly Industries Ltd N-heteroarylidene erythomycylamines
DE2515075C2 (de) * 1975-04-07 1985-10-24 Dr. Karl Thomae Gmbh, 7950 Biberach Erythromycinderivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel
DE2515077A1 (de) * 1975-04-07 1976-10-28 Thomae Gmbh Dr K Neue 9-alkylidenamino-erythromycine, ihre salze und verfahren zu ihrer herstellung
DK139522C (da) * 1975-04-07 1979-08-20 Thomae Gmbh Dr K Analogifremgangsmaade til fremstilling af 9-iminoalkylamino-erythromyciner eller syreadditionssalte deraf

Also Published As

Publication number Publication date
IT1109331B (it) 1985-12-16
IL55906A0 (en) 1979-01-31
NO783767L (no) 1979-05-11
YU261178A (en) 1982-08-31
DE2860585D1 (en) 1981-04-23
AU4144878A (en) 1979-05-17
ES474693A1 (es) 1979-04-01
ATA773178A (de) 1980-08-15
DE2750288A1 (de) 1979-05-17
ZA786313B (en) 1980-07-30
JPS5476588A (en) 1979-06-19
EP0001981B1 (de) 1981-04-01
US4256738A (en) 1981-03-17
NZ188872A (en) 1981-05-29
PT68771A (de) 1978-12-01
EP0001981A1 (de) 1979-05-30
CA1107726A (en) 1981-08-25
DK499778A (da) 1979-05-11
GR65281B (en) 1980-08-01
AT361623B (de) 1981-03-25
IT7851850A0 (it) 1978-11-09

Similar Documents

Publication Publication Date Title
FI783417A (fi) Nya 9-(omega-heteroarylamino-alkylamino)-erytromyciner deras salter deras framstaellningsfoerfarande och dessa innehaollande laekemedel
FI780365A (fi) Anordning foer dosering av laekemedel
FI780801A (fi) Nya cefem- och cefam-kompositioner och foerfarande foer deras framstaellning
AR214231A1 (es) Ferrocarril aereo suspendido
SE7806710L (sv) Nya karbostyrilderivat
SE7802867L (sv) Nya 4-acylamino-fenyl-etanolaminer
FI780757A (fi) Cefemderivat och foerfarande foer deras framstaellning
FI813862L (fi) Nya 8-arylalkyl-3-fenyl-3-nortropanoler deras syraadditionssalter dessa erhaollande laekemedel och foerfarande foer deras framstaellning
SE7807642L (sv) Nya 1-acyl-2-cyanaziridiner
FI790614A (fi) Nya penicilliner deras salter foerfarande foer deras framstaellning och dessa foereningar innehaollande laekemedel
FI783590A (fi) Nya prostacyklinderivat och foerfarande foer deras framstaellning
FI780565A (fi) Foerfarande foer framstaellning av d 1-5-metyltetrahydrofolsyra och salter daerav
IT1092308B (it) Sostegno per giocattolo piramidale
SE7811457L (sv) Nya kinolylguanidinderivat
FI781667A (fi) Nya i 11-staellning substituerade 5,11-dihydro-6h-pyrido (2,3-b) (1,4)-benzodiazepin-6-oner deras framstaellningsfoerfarande och dessa innehaollande laekemedel
SE7800739L (sv) Nya aminoalkoxifenylderivat
SE7810050L (sv) Nya 7-azabensimidazoler
FI781674A (fi) Nya fluoriderade aminosyror
FI781872A (fi) Nya bispidinderivat foerfarande foer deras framstaellning och laekemedel som innehaoller dessa foereningar
FI783991A (fi) Foerfarande foer behandling av hypertension och laekemedel foer detta
FI781218A (fi) Totalbestaemning av hormoner och laekemedel
FI782215A (fi) Nya nitrosoureafoereningar och deras framstaellningsfoerfarande
FI780083A (fi) Nya ditienylalkylaminer och foerfarande foer deras framstaellning
FI782173A (fi) Benzylpyrimidiner foerfarande foer framstaellning av dem och laekemedel innehaollande dessa
FI783769A (fi) Nya tetrapeptider och metoder