FI51939C - Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi - Google Patents

Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi

Info

Publication number
FI51939C
FI51939C FI702170A FI217070A FI51939C FI 51939 C FI51939 C FI 51939C FI 702170 A FI702170 A FI 702170A FI 217070 A FI217070 A FI 217070A FI 51939 C FI51939 C FI 51939C
Authority
FI
Finland
Prior art keywords
aminoalkylamino
thieno
pyrimidines
preparation
platelet aggregation
Prior art date
Application number
FI702170A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI51939B (OSRAM
Inventor
Eberhard Woitun
Berthold Narr
Wolfgang Schroeter
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691940572 external-priority patent/DE1940572A1/de
Priority claimed from DE19702032687 external-priority patent/DE2032687A1/de
Priority claimed from DE19702032686 external-priority patent/DE2032686A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Application granted granted Critical
Publication of FI51939B publication Critical patent/FI51939B/fi
Publication of FI51939C publication Critical patent/FI51939C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Slide Fasteners (AREA)
FI702170A 1969-08-08 1970-08-06 Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi FI51939C (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702032687 DE2032687A1 (en) 1970-07-02 1970-07-02 Cardiovascular 2-aminoalkylamino-thienopyrimidines - and 4-morpholino derivatives from 4-diethanolamino-compounds by intramolecular cyclisa
DE19702032686 DE2032686A1 (de) 1970-07-02 1970-07-02 Verfahren zur Herstellung von neuen 2 Aminoalkylamino thieno eckige Klammer auf 3,2 d eckige Klammer zu Pynmidinen

Publications (2)

Publication Number Publication Date
FI51939B FI51939B (OSRAM) 1977-01-31
FI51939C true FI51939C (fi) 1977-05-10

Family

ID=27182086

Family Applications (1)

Application Number Title Priority Date Filing Date
FI702170A FI51939C (fi) 1969-08-08 1970-08-06 Menetelmä uusien verihiutaleiden kasautumista estävien 2-aminoalkyylia mino-tieno(3,2-d)pyrimidiinien valmistamiseksi

Country Status (14)

Country Link
US (1) US3838121A (OSRAM)
JP (1) JPS519759B1 (OSRAM)
BE (1) BE754606A (OSRAM)
BG (1) BG17591A3 (OSRAM)
CH (5) CH547301A (OSRAM)
ES (5) ES382551A1 (OSRAM)
FI (1) FI51939C (OSRAM)
FR (1) FR2068478B1 (OSRAM)
IE (1) IE34687B1 (OSRAM)
IL (1) IL35078A (OSRAM)
NL (1) NL7011592A (OSRAM)
NO (1) NO130538C (OSRAM)
PH (1) PH9574A (OSRAM)
SE (1) SE386449B (OSRAM)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
WO2004087707A1 (en) * 2003-03-31 2004-10-14 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
DE502006004066D1 (de) * 2006-04-19 2009-08-06 Boehringer Ingelheim Pharma Dihydrothienopyrimidine zur behandlung von entzündlichen erkrankungen
EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
CL2007001165A1 (es) * 2006-04-26 2008-01-25 Hoffmann La Roche 2-(1h-indazol-4-il)-6-(4-metanosulfonil-piperazin-1-ilmetil)-4-morfolin-4-il-tieno[3,2-d]pirimidina; procedimiento de preparacion; composicion farmaceutica; proceso de preparacion de dicha composicion; kit farmaceutico; y uso para tratar enfermedades tales como cancer, desordenes inmunes y enfermedades cardiovasculares.
PL2041139T3 (pl) * 2006-04-26 2012-05-31 Hoffmann La Roche Związki farmaceutyczne
CL2007001166A1 (es) 2006-04-26 2008-01-25 Piramed Ltd Compuestos derivados de pirimidina condensada, inhibidores de pi3-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicion farmaceutica
AR064155A1 (es) * 2006-12-07 2009-03-18 Piramed Ltd Compuestos de inhibidores de fosfoinositido-3 quinasa y metodos de uso
BRPI0717907A2 (pt) * 2006-12-07 2013-11-05 Genentech Inc "composto, composição farmacêutica, métodos para tratar um câncer, para inbir ou modular a atividade da lipídeo quinase, processo para a produçãoo de uma composição farmacêutica, uso de um composto e kit"
JP5341899B2 (ja) 2007-10-19 2013-11-13 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ヘテロ環置換ピペラジノ−ジヒドロチエノピリミジン
JP5563466B2 (ja) 2007-10-19 2014-07-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ピペラジノ−ジヒドロチエノピリミジン誘導体
ATE542825T1 (de) * 2007-10-19 2012-02-15 Boehringer Ingelheim Int Substituierte piperidino-dihydrothienopyrimidine
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
SG182247A1 (en) * 2009-05-27 2012-08-30 Hoffmann La Roche Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
SG175708A1 (en) * 2009-05-27 2011-12-29 Genentech Inc Bicyclic pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
MX345155B (es) * 2009-10-12 2017-01-18 F Hoffmann-La Roche Ag * Combinaciones de un inhibidor de pi3k y un inhibidor de mek.
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma

Also Published As

Publication number Publication date
CH546251A (de) 1974-02-28
JPS519759B1 (OSRAM) 1976-03-30
FI51939B (OSRAM) 1977-01-31
ES382552A1 (es) 1973-04-16
FR2068478A1 (OSRAM) 1971-08-27
ES382550A1 (es) 1973-04-16
US3838121A (en) 1974-09-24
NL7011592A (OSRAM) 1971-02-10
CH547304A (de) 1974-03-29
BE754606A (fr) 1971-02-08
SE386449B (sv) 1976-08-09
IL35078A0 (en) 1970-10-30
PH9574A (en) 1976-01-16
BG17591A3 (bg) 1973-11-10
NO130538C (OSRAM) 1975-01-08
FR2068478B1 (OSRAM) 1974-08-30
NO130538B (OSRAM) 1974-09-23
CH547301A (de) 1974-03-29
ES382549A1 (es) 1973-04-01
ES382548A1 (es) 1973-04-01
IL35078A (en) 1974-09-10
CH547300A (de) 1974-03-29
IE34687L (en) 1971-02-08
IE34687B1 (en) 1975-07-23
CH547299A (de) 1974-03-29
ES382551A1 (es) 1973-04-01

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