FI48082C - Menetelmä uusien verenpainetta alentavien 2-aryylihydratsino-imidatsol iinien-(2) valmistamiseksi - Google Patents

Menetelmä uusien verenpainetta alentavien 2-aryylihydratsino-imidatsol iinien-(2) valmistamiseksi

Info

Publication number
FI48082C
FI48082C FI672082A FI208267A FI48082C FI 48082 C FI48082 C FI 48082C FI 672082 A FI672082 A FI 672082A FI 208267 A FI208267 A FI 208267A FI 48082 C FI48082 C FI 48082C
Authority
FI
Finland
Prior art keywords
arylhydrazinoimidazoline
antihypertensive
preparation
Prior art date
Application number
FI672082A
Other languages
English (en)
Swedish (sv)
Other versions
FI48082B (fi
Inventor
Staehle
Kummer
Koeppe
Zeile
Hoefke
Samtleben
Original Assignee
Boehringer Sohn Ingelheim
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1966B0088361 external-priority patent/DE1670124B2/de
Application filed by Boehringer Sohn Ingelheim filed Critical Boehringer Sohn Ingelheim
Application granted granted Critical
Publication of FI48082B publication Critical patent/FI48082B/fi
Publication of FI48082C publication Critical patent/FI48082C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44Nitrogen atoms not forming part of a nitro radical
FI672082A 1966-08-05 1967-07-31 Menetelmä uusien verenpainetta alentavien 2-aryylihydratsino-imidatsol iinien-(2) valmistamiseksi FI48082C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE1966B0088361 DE1670124B2 (de) 1966-08-05 1966-08-05 2-phenylhydrazino-imidazoline-(2), verfahren zu deren herstellung sowie diese enthaltende blutdrucksenkende zubereitungen
DEB0090823 1967-01-20

Publications (2)

Publication Number Publication Date
FI48082B FI48082B (fi) 1974-02-28
FI48082C true FI48082C (fi) 1974-06-10

Family

ID=25968043

Family Applications (1)

Application Number Title Priority Date Filing Date
FI672082A FI48082C (fi) 1966-08-05 1967-07-31 Menetelmä uusien verenpainetta alentavien 2-aryylihydratsino-imidatsol iinien-(2) valmistamiseksi

Country Status (9)

Country Link
US (1) US3480630A (fi)
AT (1) AT284115B (fi)
CH (3) CH505111A (fi)
DK (1) DK118607B (fi)
FI (1) FI48082C (fi)
FR (2) FR1550151A (fi)
GB (1) GB1180794A (fi)
IL (1) IL28433A (fi)
YU (3) YU32176B (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3516995A (en) * 1969-02-27 1970-06-23 Sandoz Ag Benzalhydrazones
DE2041734A1 (de) * 1970-08-22 1972-02-24 Bayer Ag Carbamate der 2-Phenylhydrazino-2-imidazoline,Verfahren zu ihrer Herstellung und ihre Verwendung als Ektoparasitizide
US4028380A (en) * 1974-06-01 1977-06-07 Akzona Incorporated Hydrazino-imidazole derivatives
NL7407469A (nl) * 1974-06-01 1975-12-03 Akzo Nv Nieuwe amidinohydrazonverbindingen.
US4117146A (en) * 1977-06-27 1978-09-26 The Dow Chemical Company Method for treating depression and anxiety using phenyl hydrazo compounds
JP2864075B2 (ja) * 1991-12-04 1999-03-03 富士写真フイルム株式会社 イミダゾールアゾ色素およびそれを含有する熱転写色素供与材料
CN101687812A (zh) 2007-07-02 2010-03-31 弗·哈夫曼-拉罗切有限公司 对痕量胺相关受体(taar)具有良好亲和性的2-咪唑啉化合物
AU2008281918A1 (en) * 2007-07-27 2009-02-05 F. Hoffmann-La Roche Ag 2-azetidinemethaneamines and 2-pyrrolidinemethaneamines as TAAR-ligands
WO2009019149A1 (en) * 2007-08-03 2009-02-12 F. Hoffmann-La Roche Ag Pyridinecarboxamide and benzamide derivatives as taar1 ligands
US9452980B2 (en) * 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
MA53755A (fr) 2016-03-17 2021-08-04 Hoffmann La Roche Dérivé de 5-éthyl-4-méthyl-pyrazole-3-carboxamide ayant une activité comme agonist de taar

Also Published As

Publication number Publication date
GB1180794A (en) 1970-02-11
CH489502A (de) 1970-04-30
DK118607B (da) 1970-09-14
US3480630A (en) 1969-11-25
CH505111A (de) 1971-03-31
IL28433A (en) 1971-06-23
YU76573A (en) 1977-12-31
FR1550151A (fi) 1968-12-20
YU153867A (en) 1973-12-31
YU73377A (en) 1982-06-30
AT284115B (de) 1970-09-10
YU32176B (en) 1974-06-30
CH497432A (de) 1970-10-15
YU33864B (en) 1978-06-30
FR7322M (fi) 1969-10-06
FI48082B (fi) 1974-02-28

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