BE754606A - Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication - Google Patents

Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication

Info

Publication number
BE754606A
BE754606A BE754606DA BE754606A BE 754606 A BE754606 A BE 754606A BE 754606D A BE754606D A BE 754606DA BE 754606 A BE754606 A BE 754606A
Authority
BE
Belgium
Prior art keywords
aminoalcoylamino
thieno
pyrimidines
new
manufacturing processes
Prior art date
Application number
Other languages
English (en)
French (fr)
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Publication date
Priority claimed from DE19691940572 external-priority patent/DE1940572A1/de
Priority claimed from DE19702032687 external-priority patent/DE2032687A1/de
Priority claimed from DE19702032686 external-priority patent/DE2032686A1/de
Publication of BE754606A publication Critical patent/BE754606A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Slide Fasteners (AREA)
BE754606D 1969-08-08 Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication BE754606A (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702032687 DE2032687A1 (en) 1970-07-02 1970-07-02 Cardiovascular 2-aminoalkylamino-thienopyrimidines - and 4-morpholino derivatives from 4-diethanolamino-compounds by intramolecular cyclisa
DE19702032686 DE2032686A1 (de) 1970-07-02 1970-07-02 Verfahren zur Herstellung von neuen 2 Aminoalkylamino thieno eckige Klammer auf 3,2 d eckige Klammer zu Pynmidinen

Publications (1)

Publication Number Publication Date
BE754606A true BE754606A (fr) 1971-02-08

Family

ID=27182086

Family Applications (1)

Application Number Title Priority Date Filing Date
BE754606D BE754606A (fr) 1969-08-08 Nouvelles 2-aminoalcoylamino-thieno(3,2-d)pyrimidines et leurs procedesde fabrication

Country Status (14)

Country Link
US (1) US3838121A (OSRAM)
JP (1) JPS519759B1 (OSRAM)
BE (1) BE754606A (OSRAM)
BG (1) BG17591A3 (OSRAM)
CH (5) CH547301A (OSRAM)
ES (5) ES382551A1 (OSRAM)
FI (1) FI51939C (OSRAM)
FR (1) FR2068478B1 (OSRAM)
IE (1) IE34687B1 (OSRAM)
IL (1) IL35078A (OSRAM)
NL (1) NL7011592A (OSRAM)
NO (1) NO130538C (OSRAM)
PH (1) PH9574A (OSRAM)
SE (1) SE386449B (OSRAM)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
WO2004087707A1 (en) * 2003-03-31 2004-10-14 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
DE502006004066D1 (de) * 2006-04-19 2009-08-06 Boehringer Ingelheim Pharma Dihydrothienopyrimidine zur behandlung von entzündlichen erkrankungen
EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
CL2007001165A1 (es) * 2006-04-26 2008-01-25 Hoffmann La Roche 2-(1h-indazol-4-il)-6-(4-metanosulfonil-piperazin-1-ilmetil)-4-morfolin-4-il-tieno[3,2-d]pirimidina; procedimiento de preparacion; composicion farmaceutica; proceso de preparacion de dicha composicion; kit farmaceutico; y uso para tratar enfermedades tales como cancer, desordenes inmunes y enfermedades cardiovasculares.
PL2041139T3 (pl) * 2006-04-26 2012-05-31 Hoffmann La Roche Związki farmaceutyczne
CL2007001166A1 (es) 2006-04-26 2008-01-25 Piramed Ltd Compuestos derivados de pirimidina condensada, inhibidores de pi3-quinasa; procesos para preparar los compuestos; composicion farmaceutica que los comprende; uso de los compuestos en la preparacion de medicamentos; proceso para preparar la composicion farmaceutica; y kit que incluye a la composicion farmaceutica
AR064155A1 (es) * 2006-12-07 2009-03-18 Piramed Ltd Compuestos de inhibidores de fosfoinositido-3 quinasa y metodos de uso
BRPI0717907A2 (pt) * 2006-12-07 2013-11-05 Genentech Inc "composto, composição farmacêutica, métodos para tratar um câncer, para inbir ou modular a atividade da lipídeo quinase, processo para a produçãoo de uma composição farmacêutica, uso de um composto e kit"
JP5341899B2 (ja) 2007-10-19 2013-11-13 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング ヘテロ環置換ピペラジノ−ジヒドロチエノピリミジン
JP5563466B2 (ja) 2007-10-19 2014-07-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ピペラジノ−ジヒドロチエノピリミジン誘導体
ATE542825T1 (de) * 2007-10-19 2012-02-15 Boehringer Ingelheim Int Substituierte piperidino-dihydrothienopyrimidine
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
SG182247A1 (en) * 2009-05-27 2012-08-30 Hoffmann La Roche Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
SG175708A1 (en) * 2009-05-27 2011-12-29 Genentech Inc Bicyclic pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
MX345155B (es) * 2009-10-12 2017-01-18 F Hoffmann-La Roche Ag * Combinaciones de un inhibidor de pi3k y un inhibidor de mek.
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma

Also Published As

Publication number Publication date
CH546251A (de) 1974-02-28
FI51939C (fi) 1977-05-10
JPS519759B1 (OSRAM) 1976-03-30
FI51939B (OSRAM) 1977-01-31
ES382552A1 (es) 1973-04-16
FR2068478A1 (OSRAM) 1971-08-27
ES382550A1 (es) 1973-04-16
US3838121A (en) 1974-09-24
NL7011592A (OSRAM) 1971-02-10
CH547304A (de) 1974-03-29
SE386449B (sv) 1976-08-09
IL35078A0 (en) 1970-10-30
PH9574A (en) 1976-01-16
BG17591A3 (bg) 1973-11-10
NO130538C (OSRAM) 1975-01-08
FR2068478B1 (OSRAM) 1974-08-30
NO130538B (OSRAM) 1974-09-23
CH547301A (de) 1974-03-29
ES382549A1 (es) 1973-04-01
ES382548A1 (es) 1973-04-01
IL35078A (en) 1974-09-10
CH547300A (de) 1974-03-29
IE34687L (en) 1971-02-08
IE34687B1 (en) 1975-07-23
CH547299A (de) 1974-03-29
ES382551A1 (es) 1973-04-01

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