FI46389B - - Google Patents

Info

Publication number
FI46389B
FI46389B FI2632/64A FI263264A FI46389B FI 46389 B FI46389 B FI 46389B FI 2632/64 A FI2632/64 A FI 2632/64A FI 263264 A FI263264 A FI 263264A FI 46389 B FI46389 B FI 46389B
Authority
FI
Finland
Application number
FI2632/64A
Other languages
Finnish (fi)
Other versions
FI46389C (fi
Inventor
F Sorm
A Piskala
Original Assignee
Ceskoslovenska Akademie Ved
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ceskoslovenska Akademie Ved filed Critical Ceskoslovenska Akademie Ved
Publication of FI46389B publication Critical patent/FI46389B/fi
Application granted granted Critical
Publication of FI46389C publication Critical patent/FI46389C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12Triazine radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20Carbocyclic rings
    • C07H15/22Cyclohexane rings, substituted by nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Saccharide Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FI642632A 1963-12-22 1964-12-12 Menetelmä terapeuttisesti arvokkaiden 1-beetta-d-ribofuranosyyli- ja 1 -(2-desoksi-beetta-d-ribofuranosyyli)-5-atsasytosiinien valmistamiseks i. FI46389C (fi)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CS709363 1963-12-22

Publications (2)

Publication Number Publication Date
FI46389B true FI46389B (ru) 1972-11-30
FI46389C FI46389C (fi) 1973-03-12

Family

ID=5419399

Family Applications (1)

Application Number Title Priority Date Filing Date
FI642632A FI46389C (fi) 1963-12-22 1964-12-12 Menetelmä terapeuttisesti arvokkaiden 1-beetta-d-ribofuranosyyli- ja 1 -(2-desoksi-beetta-d-ribofuranosyyli)-5-atsasytosiinien valmistamiseks i.

Country Status (13)

Country Link
US (1) US3350388A (ru)
AT (1) AT252458B (ru)
BE (1) BE657451A (ru)
BR (1) BR6465569D0 (ru)
CH (1) CH479595A (ru)
DE (1) DE1245384B (ru)
DK (1) DK108500C (ru)
ES (1) ES307376A1 (ru)
FI (1) FI46389C (ru)
FR (1) FR1450440A (ru)
GB (1) GB1050899A (ru)
IT (1) IT1043755B (ru)
NL (1) NL6414959A (ru)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1030970A (en) * 1964-05-15 1966-05-25 Inst Mikrobiologii Im Akad D K Method for the preparation of 2', 3', 5'-tri-o-acyl-6-azacytidines
DE2012888C3 (de) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden
US6943249B2 (en) * 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US6887855B2 (en) * 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US7038038B2 (en) * 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
WO2009042064A2 (en) 2007-09-21 2009-04-02 Nektar Therapeutics Al, Corporation Oligomer-nucleoside phosphate conjugates
CN101815437A (zh) * 2007-09-26 2010-08-25 辛乃山医学院 氮杂胞苷类似物和其应用
DK3692983T3 (da) 2008-05-15 2021-09-20 Celgene Corp Orale formuleringer af cytidinanaloger og fremgangsmåder til anvendelse deraf
WO2010014883A2 (en) 2008-08-01 2010-02-04 Dr. Reddy's Laboratories Ltd. Azacitidine process and polymorphs
WO2010017547A1 (en) * 2008-08-08 2010-02-11 Scinopharm Taiwan Ldt. Process for making 5-azacytosine nucleosides and their derivatives
NZ595382A (en) * 2009-03-23 2014-02-28 Ambit Biosciences Corp Combination therapy involving n-(5-(tert-butyl-isoxazol-3-yl)-n’-{ 4-(7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl} urea
IT1399195B1 (it) 2010-03-30 2013-04-11 Chemi Spa Processo per la sintesi di azacitidina e decitabina
EP2691408B1 (en) 2011-03-31 2017-06-28 Celgene International SÁRL Synthesis of 5-azacytidine
EA031986B1 (ru) 2012-04-04 2019-03-29 Галозим, Инк. Способ и комбинация для лечения солидной раковой опухоли и набор, содержащий комбинацию
CN108239128B (zh) 2016-12-23 2019-03-29 江苏奥赛康药业股份有限公司 β-核苷类化合物的制备方法
US20190351031A1 (en) 2018-05-16 2019-11-21 Halozyme, Inc. Methods of selecting subjects for combination cancer therapy with a polymer-conjugated soluble ph20

Also Published As

Publication number Publication date
AT252458B (de) 1967-02-27
US3350388A (en) 1967-10-31
IT1043755B (it) 1980-02-29
DK108500C (da) 1967-12-27
GB1050899A (ru)
FR1450440A (fr) 1966-06-24
BE657451A (ru) 1965-04-16
NL6414959A (ru) 1965-06-23
FI46389C (fi) 1973-03-12
DE1245384B (de) 1967-07-27
ES307376A1 (es) 1965-05-01
BR6465569D0 (pt) 1973-08-02
CH479595A (de) 1969-10-15

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