BR6465569D0 - Processo para a producao de 1-glicosil-5-azacitozinas - Google Patents
Processo para a producao de 1-glicosil-5-azacitozinasInfo
- Publication number
- BR6465569D0 BR6465569D0 BR165569/64A BR16556964A BR6465569D0 BR 6465569 D0 BR6465569 D0 BR 6465569D0 BR 165569/64 A BR165569/64 A BR 165569/64A BR 16556964 A BR16556964 A BR 16556964A BR 6465569 D0 BR6465569 D0 BR 6465569D0
- Authority
- BR
- Brazil
- Prior art keywords
- azacitozins
- glycosyl
- production
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/12—Triazine radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Saccharide Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CS709363 | 1963-12-22 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR6465569D0 true BR6465569D0 (pt) | 1973-08-02 |
Family
ID=5419399
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR165569/64A BR6465569D0 (pt) | 1963-12-22 | 1964-12-22 | Processo para a producao de 1-glicosil-5-azacitozinas |
Country Status (13)
Country | Link |
---|---|
US (1) | US3350388A (pt) |
AT (1) | AT252458B (pt) |
BE (1) | BE657451A (pt) |
BR (1) | BR6465569D0 (pt) |
CH (1) | CH479595A (pt) |
DE (1) | DE1245384B (pt) |
DK (1) | DK108500C (pt) |
ES (1) | ES307376A1 (pt) |
FI (1) | FI46389C (pt) |
FR (1) | FR1450440A (pt) |
GB (1) | GB1050899A (pt) |
IT (1) | IT1043755B (pt) |
NL (1) | NL6414959A (pt) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB1030970A (en) * | 1964-05-15 | 1966-05-25 | Inst Mikrobiologii Im Akad D K | Method for the preparation of 2', 3', 5'-tri-o-acyl-6-azacytidines |
DE2012888C3 (de) * | 1970-03-14 | 1981-04-02 | Schering Ag, 1000 Berlin Und 4619 Bergkamen | Verfahren zur Herstellung von 5-Azapyrimidinnucleosiden |
US7038038B2 (en) * | 2003-03-17 | 2006-05-02 | Pharmion Corporation | Synthesis of 5-azacytidine |
US6887855B2 (en) * | 2003-03-17 | 2005-05-03 | Pharmion Corporation | Forms of 5-azacytidine |
US6943249B2 (en) * | 2003-03-17 | 2005-09-13 | Ash Stevens, Inc. | Methods for isolating crystalline Form I of 5-azacytidine |
US20060014949A1 (en) * | 2004-07-13 | 2006-01-19 | Supergen Inc. | Compositions and formulations of decitabine polymorphs and methods of use thereof |
WO2009042064A2 (en) | 2007-09-21 | 2009-04-02 | Nektar Therapeutics Al, Corporation | Oligomer-nucleoside phosphate conjugates |
BRPI0817269A2 (pt) * | 2007-09-26 | 2014-10-07 | Sinai School Medicine | Análogos de azacitidina e usos dos mesmos |
CN103479586B (zh) | 2008-05-15 | 2017-03-01 | 细胞基因公司 | 胞苷类似物的口服制剂和其使用方法 |
WO2010014883A2 (en) * | 2008-08-01 | 2010-02-04 | Dr. Reddy's Laboratories Ltd. | Azacitidine process and polymorphs |
JP5650643B2 (ja) * | 2008-08-08 | 2015-01-07 | サイノファーム タイワン リミテッド | 5−アザシトシンヌクレオシド及びその誘導体の製造方法 |
CA2755976C (en) * | 2009-03-23 | 2020-04-07 | Ambit Biosciences Corporation | Methods of treatment using combination therapy |
IT1399195B1 (it) | 2010-03-30 | 2013-04-11 | Chemi Spa | Processo per la sintesi di azacitidina e decitabina |
WO2012135405A1 (en) | 2011-03-31 | 2012-10-04 | Pharmion Llc | Systhesis of 5-azacytidine |
EA031986B1 (ru) | 2012-04-04 | 2019-03-29 | Галозим, Инк. | Способ и комбинация для лечения солидной раковой опухоли и набор, содержащий комбинацию |
CN108239128B (zh) | 2016-12-23 | 2019-03-29 | 江苏奥赛康药业股份有限公司 | β-核苷类化合物的制备方法 |
US20190351031A1 (en) | 2018-05-16 | 2019-11-21 | Halozyme, Inc. | Methods of selecting subjects for combination cancer therapy with a polymer-conjugated soluble ph20 |
-
0
- GB GB1050899D patent/GB1050899A/en active Active
-
1964
- 1964-12-08 DE DEC34587A patent/DE1245384B/de active Pending
- 1964-12-09 CH CH1590864A patent/CH479595A/de not_active IP Right Cessation
- 1964-12-10 AT AT1047164A patent/AT252458B/de active
- 1964-12-12 FI FI642632A patent/FI46389C/fi active
- 1964-12-14 US US418273A patent/US3350388A/en not_active Expired - Lifetime
- 1964-12-18 DK DK620664AA patent/DK108500C/da active
- 1964-12-19 IT IT27006/64A patent/IT1043755B/it active
- 1964-12-21 ES ES0307376A patent/ES307376A1/es not_active Expired
- 1964-12-22 NL NL6414959A patent/NL6414959A/xx unknown
- 1964-12-22 BR BR165569/64A patent/BR6465569D0/pt unknown
- 1964-12-22 FR FR999626A patent/FR1450440A/fr not_active Expired
- 1964-12-22 BE BE657451D patent/BE657451A/xx unknown
Also Published As
Publication number | Publication date |
---|---|
FR1450440A (fr) | 1966-06-24 |
ES307376A1 (es) | 1965-05-01 |
FI46389C (fi) | 1973-03-12 |
US3350388A (en) | 1967-10-31 |
IT1043755B (it) | 1980-02-29 |
FI46389B (pt) | 1972-11-30 |
GB1050899A (pt) | |
AT252458B (de) | 1967-02-27 |
CH479595A (de) | 1969-10-15 |
BE657451A (pt) | 1965-04-16 |
DK108500C (da) | 1967-12-27 |
DE1245384B (de) | 1967-07-27 |
NL6414959A (pt) | 1965-06-23 |
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