FI111951B - (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4]bensotiadiazin i form av sin S-enantiomer, förfarande för dess framställning och farmaceutiska kompositioner, som innehåller denna förening - Google Patents

(3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4]bensotiadiazin i form av sin S-enantiomer, förfarande för dess framställning och farmaceutiska kompositioner, som innehåller denna förening Download PDF

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Publication number
FI111951B
FI111951B FI953384A FI953384A FI111951B FI 111951 B FI111951 B FI 111951B FI 953384 A FI953384 A FI 953384A FI 953384 A FI953384 A FI 953384A FI 111951 B FI111951 B FI 111951B
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Finland
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formula
compound
medium
med
preparation
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FI953384A
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English (en)
Finnish (fi)
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FI953384A (sv
FI953384A0 (sv
Inventor
Alex Cordi
Michael Spedding
Bernard Serkiz
Jean Lepagnol
Patrice Desos
Philippe Morain
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Servier Lab
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Psychiatry (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
FI953384A 1994-07-12 1995-07-11 (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4]bensotiadiazin i form av sin S-enantiomer, förfarande för dess framställning och farmaceutiska kompositioner, som innehåller denna förening FI111951B (sv)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9408603A FR2722502B1 (fr) 1994-07-12 1994-07-12 Nouveau derive de benzothiadiazine, son procede depreparation et les compositions pharmaceutiques qui le contiennent
FR9408603 1994-07-12

Publications (3)

Publication Number Publication Date
FI953384A0 FI953384A0 (sv) 1995-07-11
FI953384A FI953384A (sv) 1996-01-13
FI111951B true FI111951B (sv) 2003-10-15

Family

ID=9465275

Family Applications (1)

Application Number Title Priority Date Filing Date
FI953384A FI111951B (sv) 1994-07-12 1995-07-11 (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4]bensotiadiazin i form av sin S-enantiomer, förfarande för dess framställning och farmaceutiska kompositioner, som innehåller denna förening

Country Status (17)

Country Link
US (1) US5536719A (sv)
EP (1) EP0692484B1 (sv)
JP (1) JP3159894B2 (sv)
CN (1) CN1043645C (sv)
AT (1) ATE178332T1 (sv)
AU (1) AU684367B2 (sv)
CA (1) CA2153549C (sv)
CY (1) CY2161B1 (sv)
DE (1) DE69508667T2 (sv)
DK (1) DK0692484T3 (sv)
ES (1) ES2132556T3 (sv)
FI (1) FI111951B (sv)
FR (1) FR2722502B1 (sv)
GR (1) GR3029847T3 (sv)
NO (1) NO306116B1 (sv)
NZ (1) NZ272543A (sv)
ZA (1) ZA955793B (sv)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE248598T1 (de) * 1995-11-15 2003-09-15 Yamanouchi Pharma Co Ltd Inhibitoren der kainsäure-neurotoxizität sowie pyridothiazinderivate
ZA991301B (en) * 1998-02-18 1999-09-13 Neurosearch As Glutamate receptor modulators.
US6943159B1 (en) 1998-02-18 2005-09-13 Neurosearch A/S Compounds and their use as positive AMPA receptor modulators
FR2812291B1 (fr) * 2000-07-28 2002-12-13 Adir Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2823753B1 (fr) * 2001-04-18 2004-07-16 Servier Lab Nouveau procede de synthese de la (3as)-5,5-dioxo-2,3,3a, 4-tetrahydro-1h-pyrrolo [2,1-c] [1,2,4] benzothiadiazine
ITBO20010271A1 (it) * 2001-05-08 2002-11-08 Giuseppe Cannazza Metodo per il trattamento e la prevenzione dei disturbi del sistema nervoso centrale associati ad una alterazione della neurotrasmissione gl
FR2833956B1 (fr) * 2001-12-21 2004-01-30 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2833955B1 (fr) * 2001-12-21 2004-01-30 Servier Lab Nouveaux derives de benzothiazine et de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2856064B1 (fr) * 2003-06-13 2005-08-19 Servier Lab Nouveaux derives de benzothiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2856065B1 (fr) * 2003-06-13 2005-08-19 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2877338B1 (fr) 2004-11-03 2007-01-26 Servier Lab Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2877342B1 (fr) 2004-11-03 2007-01-26 Servier Lab Nouveaux derives de benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2879201B1 (fr) 2004-12-10 2007-02-16 Servier Lab Nouveaux derives de benzothiazine et benzothiadiazine, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2933698A1 (fr) 2008-07-09 2010-01-15 Servier Lab Nouveaux derives de benzothiadiazines cycloalkylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
FR2955107B1 (fr) 2010-01-08 2012-03-02 Servier Lab Nouveaux derives thiochromanes, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
FR2955106B1 (fr) 2010-01-08 2011-12-23 Servier Lab Nouveaux derives de benzothiadiazines cyclopropylees, leur procede de preparation et les compositions pharmaceutiques qui les contiennent

Also Published As

Publication number Publication date
AU684367B2 (en) 1997-12-11
CN1043645C (zh) 1999-06-16
FR2722502A1 (fr) 1996-01-19
AU2491395A (en) 1996-01-25
DK0692484T3 (da) 1999-10-18
JP3159894B2 (ja) 2001-04-23
FI953384A (sv) 1996-01-13
EP0692484A1 (fr) 1996-01-17
NZ272543A (en) 1996-04-26
GR3029847T3 (en) 1999-07-30
ATE178332T1 (de) 1999-04-15
CA2153549A1 (fr) 1996-01-13
CA2153549C (fr) 2003-07-08
DE69508667D1 (de) 1999-05-06
ZA955793B (en) 1996-03-05
CN1121921A (zh) 1996-05-08
NO306116B1 (no) 1999-09-20
NO952743D0 (no) 1995-07-11
US5536719A (en) 1996-07-16
ES2132556T3 (es) 1999-08-16
FI953384A0 (sv) 1995-07-11
DE69508667T2 (de) 1999-10-28
CY2161B1 (en) 2002-08-23
NO952743L (no) 1996-01-15
JPH0841072A (ja) 1996-02-13
FR2722502B1 (fr) 1996-08-23
EP0692484B1 (fr) 1999-03-31

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