ES8800917A1 - Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas - Google Patents

Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Info

Publication number
ES8800917A1
ES8800917A1 ES557045A ES557045A ES8800917A1 ES 8800917 A1 ES8800917 A1 ES 8800917A1 ES 557045 A ES557045 A ES 557045A ES 557045 A ES557045 A ES 557045A ES 8800917 A1 ES8800917 A1 ES 8800917A1
Authority
ES
Spain
Prior art keywords
image
arylmethanones
oxadiazol
medicaments
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES557045A
Other languages
English (en)
Other versions
ES557045A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Hoechst Roussel Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Roussel Pharmaceuticals Inc filed Critical Hoechst Roussel Pharmaceuticals Inc
Publication of ES557045A0 publication Critical patent/ES557045A0/es
Publication of ES8800917A1 publication Critical patent/ES8800917A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D271/00—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms
    • C07D271/02—Heterocyclic compounds containing five-membered rings having two nitrogen atoms and one oxygen atom as the only ring hetero atoms not condensed with other rings
    • C07D271/06—1,2,4-Oxadiazoles; Hydrogenated 1,2,4-oxadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

PROCEDIMIENTO PARA LA PREPARACION DE (1,2,4-OXADIAZOL-3-IL)-ARILMETANONAS, DE FORMULA GENERAL (I), Y SUS SALES DE ADICION DE ACIDOS FARMACEUTICAMENTE ACEPTABLES. CONSISTE EN HACER REACCIONAR UN COMPUESTO DE FORMULA GENERAL (II), EN LA QUE X ES HIDROGENO, HALOGENO, ALQUILO INFERIOR O ALCOXI INFERIOR, CON FENIL-MERCAPTANO, AMONIACO O CON UNA PIPERAZINA SUSTITUIDA. OPCIONALMENTE SE PUEDE OXIDAR UN COMPUESTO DE FORMULA GENERAL (I), EN LA QUE R ES UN RADICAL DE AZUFRE, CON UN COMPUESTO PEROXIDICO, PARA FORMAR UN COMPUESTO DE FORMULA GENERAL (I), EN LA QUE R ES UN RADICAL DE FORMULA GENERAL (III). DE APLICACION COMO AGENTES ANTIHIPERTENSIVOS, ANALGESICOS Y ANTIINFLAMATORIOS.
ES557045A 1985-01-22 1986-09-01 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas Expired ES8800917A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/693,509 US4562186A (en) 1985-01-22 1985-01-22 (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use

Publications (2)

Publication Number Publication Date
ES557045A0 ES557045A0 (es) 1987-12-01
ES8800917A1 true ES8800917A1 (es) 1987-12-01

Family

ID=24784962

Family Applications (2)

Application Number Title Priority Date Filing Date
ES551041A Expired ES8705868A1 (es) 1985-01-22 1986-01-20 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas
ES557045A Expired ES8800917A1 (es) 1985-01-22 1986-09-01 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Family Applications Before (1)

Application Number Title Priority Date Filing Date
ES551041A Expired ES8705868A1 (es) 1985-01-22 1986-01-20 Un procedimiento para preparar (1,2,4-oxadiazol-3-il)-arilmetanonas

Country Status (8)

Country Link
US (1) US4562186A (es)
EP (1) EP0189080A3 (es)
JP (1) JPS61167674A (es)
DK (1) DK30186A (es)
ES (2) ES8705868A1 (es)
GR (1) GR860142B (es)
IE (1) IE860177L (es)
PT (1) PT81880B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4562186A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use
US7576220B2 (en) * 2006-04-06 2009-08-18 Rikkyo Gakuin Method of producing 1,2,4-oxadiazole derivatives
WO2020070611A1 (en) * 2018-10-01 2020-04-09 Pi Industries Ltd Oxadiazoles as fungicides

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL120029C (es) * 1959-09-29
BE738276A (en) * 1968-09-01 1970-02-16 Prepn of 3-acyl-1,2,4-oxadiazoles useful in syn - of medicaments, in plant protection and as inter
GB1227978A (es) * 1968-09-13 1971-04-15
FR2053742A5 (en) * 1969-07-16 1971-04-16 Berlin Chemie Veb Prepn of 3-acyl-1,2,4-oxadiazoles useful in syn - of medicaments, in plant protection and as inter
IL42363A0 (en) * 1972-07-04 1973-07-30 Lepetit Spa 1,2,4-oxadiazole derivatives
US4160829A (en) * 1972-12-22 1979-07-10 Gist-Brocades N.V. Antibacterial 1,2,4-oxadiazolylacetamido cephalosporins
JPS58150576A (ja) * 1982-03-03 1983-09-07 Sumitomo Chem Co Ltd 新規な１，２，４−オキサジアゾ−ル誘導体
US4562187A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (Isoxazol-3-yl)arylmethanones, compositions and pharmaceutical use
US4562186A (en) * 1985-01-22 1985-12-31 Hoechst-Roussel Pharmaceuticals Inc. (1,2,4-Oxadiazol-3-yl)arylmethanones, compositions and pharmaceutical use

Also Published As

Publication number Publication date
ES557045A0 (es) 1987-12-01
ES551041A0 (es) 1987-05-16
PT81880A (en) 1986-02-01
ES8705868A1 (es) 1987-05-16
JPS61167674A (ja) 1986-07-29
DK30186D0 (da) 1986-01-21
GR860142B (en) 1986-05-16
EP0189080A2 (en) 1986-07-30
PT81880B (en) 1987-11-12
DK30186A (da) 1986-07-23
US4562186A (en) 1985-12-31
IE860177L (en) 1986-07-22
EP0189080A3 (en) 1987-07-15

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