ES8501233A1 - Un procedimiento para la preparacion de nuevos derivados de benzoxazolinona sustituidos - Google Patents
Un procedimiento para la preparacion de nuevos derivados de benzoxazolinona sustituidosInfo
- Publication number
- ES8501233A1 ES8501233A1 ES527521A ES527521A ES8501233A1 ES 8501233 A1 ES8501233 A1 ES 8501233A1 ES 527521 A ES527521 A ES 527521A ES 527521 A ES527521 A ES 527521A ES 8501233 A1 ES8501233 A1 ES 8501233A1
- Authority
- ES
- Spain
- Prior art keywords
- radical
- benzoxazolinones
- ethyl
- amino
- substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- OJDFTWCVSPXNCS-UHFFFAOYSA-N 2-(1-aminoethyl)-2h-1,3-benzoxazol-6-one Chemical class O=C1C=CC2=NC(C(N)C)OC2=C1 OJDFTWCVSPXNCS-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- -1 alkyl radical Chemical class 0.000 abstract 4
- 229910052739 hydrogen Inorganic materials 0.000 abstract 3
- 239000001257 hydrogen Substances 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- SLRMQYXOBQWXCR-UHFFFAOYSA-N 2154-56-5 Chemical compound [CH2]C1=CC=CC=C1 SLRMQYXOBQWXCR-UHFFFAOYSA-N 0.000 abstract 1
- 206010019280 Heart failures Diseases 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- CIUQDSCDWFSTQR-UHFFFAOYSA-N [C]1=CC=CC=C1 Chemical compound [C]1=CC=CC=C1 CIUQDSCDWFSTQR-UHFFFAOYSA-N 0.000 abstract 1
- 125000003545 alkoxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 150000002431 hydrogen Chemical class 0.000 abstract 1
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
- 230000000147 hypnotic effect Effects 0.000 abstract 1
- 229910052757 nitrogen Inorganic materials 0.000 abstract 1
- 125000004433 nitrogen atom Chemical group N* 0.000 abstract 1
- 125000002023 trifluoromethyl group Chemical group FC(F)(F)* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/02—Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Heart & Thoracic Surgery (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Anesthesiology (AREA)
- Hospice & Palliative Care (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Compositions Of Macromolecular Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR8219812A FR2536749A1 (fr) | 1982-11-25 | 1982-11-25 | (amino-2 ethyl)-6 benzoxazolinones substituees, leur preparation et leurs applications en therapeutique |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES527521A0 ES527521A0 (es) | 1984-12-01 |
| ES8501233A1 true ES8501233A1 (es) | 1984-12-01 |
Family
ID=9279533
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES527521A Expired ES8501233A1 (es) | 1982-11-25 | 1983-11-24 | Un procedimiento para la preparacion de nuevos derivados de benzoxazolinona sustituidos |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US4558060A (enExample) |
| EP (1) | EP0110781B1 (enExample) |
| JP (1) | JPS59112976A (enExample) |
| KR (1) | KR910000416B1 (enExample) |
| AT (1) | ATE26270T1 (enExample) |
| AU (1) | AU562113B2 (enExample) |
| CA (1) | CA1208220A (enExample) |
| DE (1) | DE3370624D1 (enExample) |
| DK (1) | DK539983A (enExample) |
| ES (1) | ES8501233A1 (enExample) |
| FI (1) | FI78079C (enExample) |
| FR (1) | FR2536749A1 (enExample) |
| GR (1) | GR81294B (enExample) |
| HU (1) | HU190635B (enExample) |
| IE (1) | IE56285B1 (enExample) |
| PT (1) | PT77735B (enExample) |
| ZA (1) | ZA838684B (enExample) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4554284A (en) * | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones |
| MX173362B (es) * | 1987-03-02 | 1994-02-23 | Pfizer | Compuestos de piperazinil heterociclicos y procedimiento para su preparacion |
| US4883795A (en) * | 1988-01-22 | 1989-11-28 | Pfizer Inc. | Piperazinyl-heterocyclic compounds |
| FR2637286A1 (fr) * | 1988-10-04 | 1990-04-06 | Adir | Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent |
| FR2643634A1 (fr) * | 1989-02-28 | 1990-08-31 | Adir | Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent |
| US5182278A (en) * | 1989-02-28 | 1993-01-26 | Adir Et Compagnie | Analgesic benzoxazolinones having at the 6-position a 1-hydroxy-3-morpholinopropyl side chain |
| US5268381A (en) * | 1990-09-26 | 1993-12-07 | Adir Et Compagnie | Aminoalkyl-benzothiazolinone and -benzoxazolinone compounds having a high 5-HT1A affinity |
| FR2667068B1 (fr) * | 1990-09-26 | 1994-09-09 | Adir | Nouvelles amines alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US5147881A (en) * | 1990-11-14 | 1992-09-15 | Pfizer Inc | 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents |
| FR2674524B1 (fr) * | 1991-03-25 | 1993-05-21 | Adir | Nouveaux amides alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent. |
| US5338846A (en) * | 1992-08-26 | 1994-08-16 | Pfizer Inc. | Process for preparing aryl piperazinyl-heterocyclic compounds with a piperazine salt |
| US5206366A (en) * | 1992-08-26 | 1993-04-27 | Pfizer Inc. | Process for preparing aryl piperazinyl-heterocyclic compounds |
| FR2717810B1 (fr) * | 1994-03-22 | 1996-04-26 | Adir | Nouvelles aminoalkyl benzoxazolinones et benzothiazolinones, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
| CN1182103C (zh) * | 1997-08-07 | 2004-12-29 | 株式会社富吉摩托普拉泽兹 | 乙胺衍生物 |
| US7213005B2 (en) * | 1999-12-09 | 2007-05-01 | International Business Machines Corporation | Digital content distribution using web broadcasting services |
| US20040192669A1 (en) * | 2000-04-13 | 2004-09-30 | Rosenfeld Mark J. | Novel compounds for use in weight loss and appetite suppression in humans |
| US7794761B2 (en) * | 2000-04-13 | 2010-09-14 | Seroctin Research & Technology, Inc. | Methods for inducing anti-anxiety and calming effects in animals and humans |
| US7524877B2 (en) | 2003-11-20 | 2009-04-28 | Seroctin Research & Technology, Inc. | Compounds for use in weight loss and appetite suppression in humans |
| EP1687300A4 (en) * | 2003-11-28 | 2007-08-01 | Wockhardt Ltd | PROCESS FOR THE PREPARATION OF ZIPRASIDONE MONOHYDROCHLORIDE HYDRATE |
| KR100812310B1 (ko) * | 2005-12-27 | 2008-03-10 | 주식회사이에스이 | 위치제어용 얼라인 장치 |
| CA2968806A1 (en) | 2014-12-05 | 2016-06-09 | Semmelweis University | Use of arylalkylamine monoamine oxidase inhibitors in the treatment or prevention of cancer |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4034100A (en) * | 1976-02-13 | 1977-07-05 | Merck & Co., Inc. | Antihypertensive agents |
| FR2491066A1 (fr) * | 1980-09-29 | 1982-04-02 | Cerm Cent Europ Rech Mauvernay | Benzoxazolinones substituees en 6 par une chaine aminoalcool ou aminocetone, leur preparation et leur application en therapeutique |
| FR2491471A1 (fr) * | 1980-10-03 | 1982-04-09 | Cerm Cent Europ Rech Mauvernay | Benzoxazolinones substituees, leur preparation et leur application en therapeutique |
| JPS57123103A (en) * | 1981-01-26 | 1982-07-31 | Hokko Chem Ind Co Ltd | Agricultural and horticultural fungicide |
| JPS61231548A (ja) * | 1985-04-05 | 1986-10-15 | Konishiroku Photo Ind Co Ltd | 写真廃液の処理方法及び写真自動現像機 |
-
1982
- 1982-11-25 FR FR8219812A patent/FR2536749A1/fr active Granted
-
1983
- 1983-11-21 ZA ZA838684A patent/ZA838684B/xx unknown
- 1983-11-22 US US06/554,194 patent/US4558060A/en not_active Expired - Fee Related
- 1983-11-23 AU AU21612/83A patent/AU562113B2/en not_active Ceased
- 1983-11-24 JP JP58221350A patent/JPS59112976A/ja active Pending
- 1983-11-24 AT AT83402267T patent/ATE26270T1/de not_active IP Right Cessation
- 1983-11-24 EP EP83402267A patent/EP0110781B1/fr not_active Expired
- 1983-11-24 ES ES527521A patent/ES8501233A1/es not_active Expired
- 1983-11-24 FI FI834315A patent/FI78079C/fi not_active IP Right Cessation
- 1983-11-24 GR GR73064A patent/GR81294B/el unknown
- 1983-11-24 IE IE2756/83A patent/IE56285B1/en not_active IP Right Cessation
- 1983-11-24 DE DE8383402267T patent/DE3370624D1/de not_active Expired
- 1983-11-24 HU HU834038A patent/HU190635B/hu not_active IP Right Cessation
- 1983-11-24 CA CA000441918A patent/CA1208220A/en not_active Expired
- 1983-11-25 PT PT77735A patent/PT77735B/pt not_active IP Right Cessation
- 1983-11-25 KR KR1019830005578A patent/KR910000416B1/ko not_active Expired
- 1983-11-25 DK DK539983A patent/DK539983A/da not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| DK539983A (da) | 1984-05-26 |
| EP0110781B1 (fr) | 1987-04-01 |
| FI78079C (fi) | 1989-06-12 |
| US4558060A (en) | 1985-12-10 |
| EP0110781A1 (fr) | 1984-06-13 |
| FI834315L (fi) | 1984-05-26 |
| HU190635B (en) | 1986-09-29 |
| CA1208220A (en) | 1986-07-22 |
| IE832756L (en) | 1984-05-25 |
| ZA838684B (en) | 1984-07-25 |
| AU2161283A (en) | 1984-05-31 |
| KR840006633A (ko) | 1984-12-01 |
| AU562113B2 (en) | 1987-05-28 |
| FR2536749A1 (fr) | 1984-06-01 |
| FI834315A0 (fi) | 1983-11-24 |
| DE3370624D1 (en) | 1987-05-07 |
| FI78079B (fi) | 1989-02-28 |
| ES527521A0 (es) | 1984-12-01 |
| DK539983D0 (da) | 1983-11-25 |
| PT77735A (fr) | 1983-12-01 |
| ATE26270T1 (de) | 1987-04-15 |
| IE56285B1 (en) | 1991-06-05 |
| KR910000416B1 (ko) | 1991-01-25 |
| PT77735B (fr) | 1986-03-27 |
| FR2536749B1 (enExample) | 1985-04-26 |
| JPS59112976A (ja) | 1984-06-29 |
| GR81294B (enExample) | 1984-12-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD1A | Patent lapsed |
Effective date: 19960603 |