AU562113B2 - Benzoxazolinones - Google Patents

Benzoxazolinones

Info

Publication number
AU562113B2
AU562113B2 AU21612/83A AU2161283A AU562113B2 AU 562113 B2 AU562113 B2 AU 562113B2 AU 21612/83 A AU21612/83 A AU 21612/83A AU 2161283 A AU2161283 A AU 2161283A AU 562113 B2 AU562113 B2 AU 562113B2
Authority
AU
Australia
Prior art keywords
radical
hydrogen
compounds
lower alkyl
represent
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU21612/83A
Other languages
English (en)
Other versions
AU2161283A (en
Inventor
Norbert Busch
Daniel-Henri Caignard
Daniel Lesieur
Charles Lespagnol
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Riom Laboratoires-Cerm Sa
Original Assignee
Centre Europeen de Recherches Mauvernay CERM
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Centre Europeen de Recherches Mauvernay CERM filed Critical Centre Europeen de Recherches Mauvernay CERM
Publication of AU2161283A publication Critical patent/AU2161283A/en
Application granted granted Critical
Publication of AU562113B2 publication Critical patent/AU562113B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/54Benzoxazoles; Hydrogenated benzoxazoles
    • C07D263/58Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cardiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Anesthesiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
AU21612/83A 1982-11-25 1983-11-23 Benzoxazolinones Ceased AU562113B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR8219812A FR2536749A1 (fr) 1982-11-25 1982-11-25 (amino-2 ethyl)-6 benzoxazolinones substituees, leur preparation et leurs applications en therapeutique
FR8219812 1982-11-25

Publications (2)

Publication Number Publication Date
AU2161283A AU2161283A (en) 1984-05-31
AU562113B2 true AU562113B2 (en) 1987-05-28

Family

ID=9279533

Family Applications (1)

Application Number Title Priority Date Filing Date
AU21612/83A Ceased AU562113B2 (en) 1982-11-25 1983-11-23 Benzoxazolinones

Country Status (17)

Country Link
US (1) US4558060A (enExample)
EP (1) EP0110781B1 (enExample)
JP (1) JPS59112976A (enExample)
KR (1) KR910000416B1 (enExample)
AT (1) ATE26270T1 (enExample)
AU (1) AU562113B2 (enExample)
CA (1) CA1208220A (enExample)
DE (1) DE3370624D1 (enExample)
DK (1) DK539983A (enExample)
ES (1) ES8501233A1 (enExample)
FI (1) FI78079C (enExample)
FR (1) FR2536749A1 (enExample)
GR (1) GR81294B (enExample)
HU (1) HU190635B (enExample)
IE (1) IE56285B1 (enExample)
PT (1) PT77735B (enExample)
ZA (1) ZA838684B (enExample)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU581020B2 (en) * 1984-09-12 1989-02-09 Smithkline Beckman Corporation 7-(2-aminoethyl)-1,3-benzthia- or oxa- zol-2(3H)-ones

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX173362B (es) * 1987-03-02 1994-02-23 Pfizer Compuestos de piperazinil heterociclicos y procedimiento para su preparacion
US4883795A (en) * 1988-01-22 1989-11-28 Pfizer Inc. Piperazinyl-heterocyclic compounds
FR2637286A1 (fr) * 1988-10-04 1990-04-06 Adir Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
FR2643634A1 (fr) * 1989-02-28 1990-08-31 Adir Nouveaux derives benzoxazolinoniques, leurs procedes de preparation et les compositions pharmaceutiques qui les contiennent
US5182278A (en) * 1989-02-28 1993-01-26 Adir Et Compagnie Analgesic benzoxazolinones having at the 6-position a 1-hydroxy-3-morpholinopropyl side chain
US5268381A (en) * 1990-09-26 1993-12-07 Adir Et Compagnie Aminoalkyl-benzothiazolinone and -benzoxazolinone compounds having a high 5-HT1A affinity
FR2667068B1 (fr) * 1990-09-26 1994-09-09 Adir Nouvelles amines alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5147881A (en) * 1990-11-14 1992-09-15 Pfizer Inc 4-(1,2-benzisoxazolyl)piperidine antipsychotic agents
FR2674524B1 (fr) * 1991-03-25 1993-05-21 Adir Nouveaux amides alkyl heterocycliques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
US5338846A (en) * 1992-08-26 1994-08-16 Pfizer Inc. Process for preparing aryl piperazinyl-heterocyclic compounds with a piperazine salt
US5206366A (en) * 1992-08-26 1993-04-27 Pfizer Inc. Process for preparing aryl piperazinyl-heterocyclic compounds
FR2717810B1 (fr) * 1994-03-22 1996-04-26 Adir Nouvelles aminoalkyl benzoxazolinones et benzothiazolinones, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
CN1182103C (zh) * 1997-08-07 2004-12-29 株式会社富吉摩托普拉泽兹 乙胺衍生物
US7213005B2 (en) * 1999-12-09 2007-05-01 International Business Machines Corporation Digital content distribution using web broadcasting services
US20040192669A1 (en) * 2000-04-13 2004-09-30 Rosenfeld Mark J. Novel compounds for use in weight loss and appetite suppression in humans
US7794761B2 (en) * 2000-04-13 2010-09-14 Seroctin Research & Technology, Inc. Methods for inducing anti-anxiety and calming effects in animals and humans
US7524877B2 (en) 2003-11-20 2009-04-28 Seroctin Research & Technology, Inc. Compounds for use in weight loss and appetite suppression in humans
EP1687300A4 (en) * 2003-11-28 2007-08-01 Wockhardt Ltd PROCESS FOR THE PREPARATION OF ZIPRASIDONE MONOHYDROCHLORIDE HYDRATE
KR100812310B1 (ko) * 2005-12-27 2008-03-10 주식회사이에스이 위치제어용 얼라인 장치
CA2968806A1 (en) 2014-12-05 2016-06-09 Semmelweis University Use of arylalkylamine monoamine oxidase inhibitors in the treatment or prevention of cancer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4034100A (en) * 1976-02-13 1977-07-05 Merck & Co., Inc. Antihypertensive agents
FR2491066A1 (fr) * 1980-09-29 1982-04-02 Cerm Cent Europ Rech Mauvernay Benzoxazolinones substituees en 6 par une chaine aminoalcool ou aminocetone, leur preparation et leur application en therapeutique
FR2491471A1 (fr) * 1980-10-03 1982-04-09 Cerm Cent Europ Rech Mauvernay Benzoxazolinones substituees, leur preparation et leur application en therapeutique
JPS57123103A (en) * 1981-01-26 1982-07-31 Hokko Chem Ind Co Ltd Agricultural and horticultural fungicide
JPS61231548A (ja) * 1985-04-05 1986-10-15 Konishiroku Photo Ind Co Ltd 写真廃液の処理方法及び写真自動現像機

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU581020B2 (en) * 1984-09-12 1989-02-09 Smithkline Beckman Corporation 7-(2-aminoethyl)-1,3-benzthia- or oxa- zol-2(3H)-ones

Also Published As

Publication number Publication date
DK539983A (da) 1984-05-26
EP0110781B1 (fr) 1987-04-01
FI78079C (fi) 1989-06-12
US4558060A (en) 1985-12-10
EP0110781A1 (fr) 1984-06-13
FI834315L (fi) 1984-05-26
HU190635B (en) 1986-09-29
CA1208220A (en) 1986-07-22
IE832756L (en) 1984-05-25
ZA838684B (en) 1984-07-25
AU2161283A (en) 1984-05-31
KR840006633A (ko) 1984-12-01
FR2536749A1 (fr) 1984-06-01
FI834315A0 (fi) 1983-11-24
DE3370624D1 (en) 1987-05-07
FI78079B (fi) 1989-02-28
ES527521A0 (es) 1984-12-01
DK539983D0 (da) 1983-11-25
ES8501233A1 (es) 1984-12-01
PT77735A (fr) 1983-12-01
ATE26270T1 (de) 1987-04-15
IE56285B1 (en) 1991-06-05
KR910000416B1 (ko) 1991-01-25
PT77735B (fr) 1986-03-27
FR2536749B1 (enExample) 1985-04-26
JPS59112976A (ja) 1984-06-29
GR81294B (enExample) 1984-12-11

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