ES8202561A1 - Un procedimiento para la produccion de 11,12-carbonato de eritromicilamina - Google Patents

Un procedimiento para la produccion de 11,12-carbonato de eritromicilamina

Info

Publication number
ES8202561A1
ES8202561A1 ES500939A ES500939A ES8202561A1 ES 8202561 A1 ES8202561 A1 ES 8202561A1 ES 500939 A ES500939 A ES 500939A ES 500939 A ES500939 A ES 500939A ES 8202561 A1 ES8202561 A1 ES 8202561A1
Authority
ES
Spain
Prior art keywords
erythromycylamine
carbonate
preparation
derivatives
carbethoxypropionyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES500939A
Other languages
English (en)
Other versions
ES500939A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES8202561A1 publication Critical patent/ES8202561A1/es
Publication of ES500939A0 publication Critical patent/ES500939A0/es
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

PROCEDIMIENTOS DE PREPARACION DE 11,12 CARBONO DE ERITROMICILAMINA Y CIERTOS DERIVADOS, ASI COMO SUS SALES DE ADICION FARMACEUTICAMENTE ACEPTABLES. CONSISTENTE EN PRODUCIR 11,12 CARBONATO DE ERITROMICILAMINA ESTERIFICANDO DIRECTAMENTE LA ERITROMICILAMINA CON UN CARBONATO DE ALQUILENO EN UN DISOLVENTE INERTE A LA REACCION Y EN PRESENCIA DE UN CARBONATO METALICO ALCALINO. EN UN PROCEDIMIENTO SE UTILIZA CARBONATO DE ETILENO PARA LA ESTERIFICACION, EN PRESENCIA DE CARBONATO POTASICO. COMO DISOLVENTES INERTES SE UTILIZAN PREFERENTEMENTE ACETATO DE ESTILO O TOUENO. LOS COMPUESTOS OBTENIDOS SE EMPLEAN COMO AGENTES ANTIBACTERIANOS.
ES500939A 1980-04-01 1981-03-31 Un procedimiento para la produccion de 11,12-carbonato de eritromicilamina Granted ES500939A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/136,197 US4283527A (en) 1980-04-01 1980-04-01 Erythromycylamine 11,12-carbonate and derivatives thereof

Publications (2)

Publication Number Publication Date
ES8202561A1 true ES8202561A1 (es) 1982-02-01
ES500939A0 ES500939A0 (es) 1982-02-01

Family

ID=22471781

Family Applications (1)

Application Number Title Priority Date Filing Date
ES500939A Granted ES500939A0 (es) 1980-04-01 1981-03-31 Un procedimiento para la produccion de 11,12-carbonato de eritromicilamina

Country Status (11)

Country Link
US (1) US4283527A (es)
EP (1) EP0037241B1 (es)
JP (1) JPS56154496A (es)
AR (1) AR226885A1 (es)
CA (1) CA1151160A (es)
DE (1) DE3165498D1 (es)
DK (1) DK152214C (es)
ES (1) ES500939A0 (es)
GR (1) GR74812B (es)
IE (1) IE51481B1 (es)
PH (1) PH16669A (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
YU43006B (en) * 1981-03-06 1989-02-28 Pliva Pharm & Chem Works Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4740502A (en) * 1986-06-20 1988-04-26 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) * 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3417077A (en) * 1966-05-16 1968-12-17 Lilly Co Eli Erythromycin derivative and process for the preparation thereof
PL76937B1 (pl) * 1971-05-06 1977-07-30 Instytut Przemysłu Farmaceutycznego Sposób wytwarzania cyklicznych węglanów estrów erytromycynowych kwasów jednokarboksylowych
US4150220A (en) * 1977-02-04 1979-04-17 Pfizer Inc. Semi-synthetic 4"-erythromycin A derivatives

Also Published As

Publication number Publication date
DE3165498D1 (en) 1984-09-20
EP0037241A1 (en) 1981-10-07
DK152214B (da) 1988-02-08
GR74812B (es) 1984-07-12
AR226885A1 (es) 1982-08-31
DK144781A (da) 1981-10-02
DK152214C (da) 1988-08-08
US4283527A (en) 1981-08-11
JPS56154496A (en) 1981-11-30
IE51481B1 (en) 1987-01-07
CA1151160A (en) 1983-08-02
ES500939A0 (es) 1982-02-01
JPS6219437B2 (es) 1987-04-28
IE810714L (en) 1981-10-01
EP0037241B1 (en) 1984-08-15
PH16669A (en) 1983-12-13

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