ES8103755A1 - Un procedimiento para preparar compuestos de cefem - Google Patents
Un procedimiento para preparar compuestos de cefemInfo
- Publication number
- ES8103755A1 ES8103755A1 ES492002A ES492002A ES8103755A1 ES 8103755 A1 ES8103755 A1 ES 8103755A1 ES 492002 A ES492002 A ES 492002A ES 492002 A ES492002 A ES 492002A ES 8103755 A1 ES8103755 A1 ES 8103755A1
- Authority
- ES
- Spain
- Prior art keywords
- unsubstituted
- hydrogen
- cephem compounds
- protecting group
- hal
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/587—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with aliphatic hydrocarbon radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms, said aliphatic radicals being substituted in the alpha-position to the ring by a hetero atom, e.g. with m >= 0, Z being a singly or a doubly bound hetero atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cephalosporin Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
PROCEDIMIENTO PARA PREPARAR COMPUESTOS DE CEMEN DE FORMULA: *FORMULA* Y SUS SALES Y ESTERES FARMACEUTICAMENTE ACEPTABLES. DONDE X ES HALOGENO, R ELEVADO A 1 ES HIDROGENO O UN GRUPO PROTECTOR DE GRUPO AMINO, R ELEVADO A 2 DE ALCOHILO INFERIOR Y R ELEVADO A 3 ES HIDROGENO O UN GRUPO PROTECTOR DEL GRUPO CARBOXI. CONSISTE EN SOMETER UN COMPUESTO DE FORMULA: A LA ACCION DE UN REACTIVO REDUCTOR O DE CALOR PARA DE ESTA FORMA OBTENER EL COMPUESTO DESEADO. X1 ES FORMILO, HALOGENO O SULFONILOXI. LA TEMPERATURA DE REACCION ESTA COMPRENDIDA ENTRE -20 Y -50GC. ESTOS COMPUESTOS TIENEN APLICACION ANTIBACTERIANA.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP11549878A JPS5543011A (en) | 1978-09-20 | 1978-09-20 | 7-halothiazolylalkoxyiminoacetamido-3-cephem compound |
Publications (2)
Publication Number | Publication Date |
---|---|
ES8103755A1 true ES8103755A1 (es) | 1981-03-16 |
ES492002A0 ES492002A0 (es) | 1981-03-16 |
Family
ID=14663989
Family Applications (4)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES484270A Granted ES484270A0 (es) | 1978-09-20 | 1979-09-19 | Un procedimiento para preparar compuestos de cefem |
ES492001A Expired ES8103754A1 (es) | 1978-09-20 | 1980-05-30 | Un procedimiento para preparar compuestos de cefem |
ES492003A Granted ES492003A0 (es) | 1978-09-20 | 1980-05-30 | Un procedimiento para preparar compuestos de cefem |
ES492002A Granted ES492002A0 (es) | 1978-09-20 | 1980-05-30 | Un procedimiento para preparar compuestos de cefem |
Family Applications Before (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES484270A Granted ES484270A0 (es) | 1978-09-20 | 1979-09-19 | Un procedimiento para preparar compuestos de cefem |
ES492001A Expired ES8103754A1 (es) | 1978-09-20 | 1980-05-30 | Un procedimiento para preparar compuestos de cefem |
ES492003A Granted ES492003A0 (es) | 1978-09-20 | 1980-05-30 | Un procedimiento para preparar compuestos de cefem |
Country Status (12)
Country | Link |
---|---|
US (1) | US4254119A (es) |
JP (1) | JPS5543011A (es) |
AU (1) | AU528117B2 (es) |
CA (1) | CA1127632A (es) |
CH (1) | CH644129A5 (es) |
DE (1) | DE2937868A1 (es) |
ES (4) | ES484270A0 (es) |
FR (1) | FR2436787A1 (es) |
GB (1) | GB2031425B (es) |
IE (1) | IE48942B1 (es) |
IT (1) | IT7968839A0 (es) |
SE (1) | SE7907764L (es) |
Families Citing this family (15)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
PH17188A (en) * | 1977-03-14 | 1984-06-14 | Fujisawa Pharmaceutical Co | New cephem and cepham compounds and their pharmaceutical compositions and method of use |
US4372952A (en) * | 1978-07-31 | 1983-02-08 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds |
US4703046A (en) * | 1978-09-08 | 1987-10-27 | Fujisawa Pharmaceutical Co., Ltd. | Cephem compounds and processes for preparation thereof |
GR78221B (es) * | 1980-02-01 | 1984-09-26 | Ciba Geigy Ag | |
GB2111043B (en) * | 1980-12-12 | 1985-02-06 | Ciba Geigy Ag | Novel cephalosporin esters |
ES507942A0 (es) * | 1980-12-15 | 1983-02-01 | Fujisawa Pharmaceutical Co | Un procedimiento para preparar derivados del acido 7-acilaminocefalosporanico . |
JPS57154190A (en) * | 1980-12-22 | 1982-09-22 | Fujisawa Pharmaceut Co Ltd | 7-substituted cephalosporanic acid derivative and its preparation |
JPS57131794A (en) * | 1980-12-31 | 1982-08-14 | Fujisawa Pharmaceut Co Ltd | Novel cephem compound or salt thereof, preparation of the same and preventing agent and remedy for microbism containing the same as active constituent |
DE3177090D1 (en) | 1980-12-31 | 1989-09-28 | Fujisawa Pharmaceutical Co | 7-acylaminocephalosporanic acid derivatives and processes for the preparation thereof |
GB9519883D0 (en) * | 1995-09-29 | 1995-11-29 | Fujisawa Pharmaceutical Co | New cephem compounds |
US8247400B2 (en) * | 2009-02-23 | 2012-08-21 | Dedhiya Mahendra G | Cephem compounds useful for the treatment of bacterial infections |
USD644380S1 (en) | 2010-01-11 | 2011-08-30 | Soldier Technology and Armor Research Industries, LLC | Upper arm protection system |
USD630385S1 (en) | 2010-01-11 | 2011-01-04 | Soldier Technology and Armor Research Industries, LLC | Shin guard protection system |
USD628753S1 (en) | 2010-01-11 | 2010-12-07 | Soldier Technology and Armor Research Industries, LLC | Forearm protection system |
USD638583S1 (en) | 2010-01-11 | 2011-05-24 | Soldier Technology and Armor Research Industries, LLC | Torso protection assembly |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4152433A (en) * | 1976-03-12 | 1979-05-01 | Fujisawa Pharmaceutical Co., Ltd. | 2-Lower alkyl-7-substituted-2 or 3-cephem-4-carboxylic acid compounds and pharmaceutical compositions |
-
1978
- 1978-09-20 JP JP11549878A patent/JPS5543011A/ja active Pending
-
1979
- 1979-08-30 CA CA334,808A patent/CA1127632A/en not_active Expired
- 1979-09-06 AU AU50644/79A patent/AU528117B2/en not_active Ceased
- 1979-09-11 US US06/074,811 patent/US4254119A/en not_active Expired - Lifetime
- 1979-09-19 DE DE19792937868 patent/DE2937868A1/de not_active Withdrawn
- 1979-09-19 IT IT7968839A patent/IT7968839A0/it unknown
- 1979-09-19 GB GB7932466A patent/GB2031425B/en not_active Expired
- 1979-09-19 ES ES484270A patent/ES484270A0/es active Granted
- 1979-09-19 IE IE1777/79A patent/IE48942B1/en unknown
- 1979-09-19 FR FR7923354A patent/FR2436787A1/fr active Granted
- 1979-09-19 CH CH846779A patent/CH644129A5/de not_active IP Right Cessation
- 1979-09-19 SE SE7907764A patent/SE7907764L/xx not_active Application Discontinuation
-
1980
- 1980-05-30 ES ES492001A patent/ES8103754A1/es not_active Expired
- 1980-05-30 ES ES492003A patent/ES492003A0/es active Granted
- 1980-05-30 ES ES492002A patent/ES492002A0/es active Granted
Also Published As
Publication number | Publication date |
---|---|
CA1127632A (en) | 1982-07-13 |
IE48942B1 (en) | 1985-06-26 |
IT7968839A0 (it) | 1979-09-19 |
US4254119A (en) | 1981-03-03 |
JPS5543011A (en) | 1980-03-26 |
FR2436787B1 (es) | 1983-07-18 |
ES8103756A1 (es) | 1981-03-16 |
ES8100300A1 (es) | 1980-11-01 |
ES492002A0 (es) | 1981-03-16 |
SE7907764L (sv) | 1980-03-21 |
ES492001A0 (es) | 1981-03-16 |
GB2031425A (en) | 1980-04-23 |
CH644129A5 (de) | 1984-07-13 |
AU528117B2 (en) | 1983-04-14 |
DE2937868A1 (de) | 1980-04-03 |
GB2031425B (en) | 1983-02-02 |
ES484270A0 (es) | 1980-11-01 |
IE791777L (en) | 1980-03-20 |
AU5064479A (en) | 1980-03-27 |
ES8103754A1 (es) | 1981-03-16 |
ES492003A0 (es) | 1981-03-16 |
FR2436787A1 (fr) | 1980-04-18 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FD1A | Patent lapsed |
Effective date: 19990601 |