ES535625A0 - Un procedimiento para la preparacion de 9-deoxo-9a-metil-9a-aza-9a-homoeritromicina d o una sal de la misma - Google Patents

Un procedimiento para la preparacion de 9-deoxo-9a-metil-9a-aza-9a-homoeritromicina d o una sal de la misma

Info

Publication number
ES535625A0
ES535625A0 ES535625A ES535625A ES535625A0 ES 535625 A0 ES535625 A0 ES 535625A0 ES 535625 A ES535625 A ES 535625A ES 535625 A ES535625 A ES 535625A ES 535625 A0 ES535625 A0 ES 535625A0
Authority
ES
Spain
Prior art keywords
homoerythromycin
deoxo
aza
methyl
salt
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES535625A
Other languages
English (en)
Other versions
ES8604256A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES535625A0 publication Critical patent/ES535625A0/es
Publication of ES8604256A1 publication Critical patent/ES8604256A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
ES535625A 1983-09-06 1984-09-04 Un procedimiento para la preparacion de 9-deoxo-9a-metil-9a-aza-9a-homoeritromicina d o una sal de la misma Expired ES8604256A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/529,828 US4465674A (en) 1983-09-06 1983-09-06 Azahomoerythromycin D derivative and intermediates therefor

Publications (2)

Publication Number Publication Date
ES535625A0 true ES535625A0 (es) 1986-01-16
ES8604256A1 ES8604256A1 (es) 1986-01-16

Family

ID=24111406

Family Applications (1)

Application Number Title Priority Date Filing Date
ES535625A Expired ES8604256A1 (es) 1983-09-06 1984-09-04 Un procedimiento para la preparacion de 9-deoxo-9a-metil-9a-aza-9a-homoeritromicina d o una sal de la misma

Country Status (7)

Country Link
US (1) US4465674A (es)
EP (1) EP0136830A3 (es)
JP (1) JPS6072897A (es)
CA (1) CA1240320A (es)
DK (1) DK157877C (es)
ES (1) ES8604256A1 (es)
GR (1) GR80278B (es)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4518590A (en) * 1984-04-13 1985-05-21 Pfizer Inc. 9α-Aza-9α-homoerythromycin compounds, pharmaceutical compositions and therapeutic method
MX13723A (es) * 1987-11-10 1993-05-01 Pfizer Procedimiento para preparar derivados de 9-desoxo-9a-alil- y propargil-9a-aza-9a-homoeritromicina a
US5075289A (en) * 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
US5912331A (en) * 1991-03-15 1999-06-15 Merck & Co., Inc. Process for the preparation of 9-deoxo-9(Z)-hydroxyiminoerythromycin A
US5985844A (en) * 1992-03-26 1999-11-16 Merck & Co., Inc. Homoerythromycin A derivatives modified at the 4"-and 8A-positions
US5189159A (en) * 1992-04-02 1993-02-23 Merck & Co., Inc. 8a-AZA-8a-homoerythromycin cyclic iminoethers
US5215980A (en) * 1992-01-17 1993-06-01 Merck & Co., Inc. 10-AZA-9-deoxo-11-deoxy-erythromycin A and derivatives thereof
US5210235A (en) * 1992-08-26 1993-05-11 Merck & Co., Inc. Methods of elaborating erythromycin fragments into amine-containing fragments of azalide antibiotics
US5332807A (en) * 1993-04-14 1994-07-26 Merck & Co., Inc. Process of producing 8A- and 9A-azalide antibiotics
EP1313749B1 (en) * 2000-08-23 2005-10-12 Wockhardt Limited Process for preparation of anhydrous azithromycin
US20040067898A1 (en) * 2001-11-27 2004-04-08 John Somberg Synthesis and separation of optically active isomers of erythromycin and their biological actions
US6861413B2 (en) * 2001-05-22 2005-03-01 Pfizer Inc. Stable non-dihydrate azithromycin oral suspensions
EA007618B1 (ru) * 2001-05-22 2006-12-29 Пфайзер Продактс Инк. Кристаллический полуторогидрат азитромицина, содержащая его фармацевтическая композиция и способ лечения на его основе
US7468428B2 (en) * 2004-03-17 2008-12-23 App Pharmaceuticals, Llc Lyophilized azithromycin formulation
US20060116336A1 (en) * 2004-03-17 2006-06-01 American Pharmaceutical Partners, Inc. Lyophilized azithromycin formulation
JP4762648B2 (ja) * 2005-08-30 2011-08-31 三和シヤッター工業株式会社 窓装置のロック装置

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3736313A (en) * 1971-02-26 1973-05-29 Abbott Lab Erythromycin derivatives
YU43116B (en) * 1979-04-02 1989-04-30 Pliva Pharm & Chem Works Process for preparing 11-aza-4-o-cladinosyl-6-o-desosaminyl-15-ethyl-7,13,14-trihydroxy-3,5,7,9,12,14-hexamethyl-oxacyclopentadecane-2-one(11-aza-10-deox
SI8110592A8 (en) * 1981-03-06 1996-06-30 Pliva Pharm & Chem Works Process for preparing of n-methyl-11-aza-10-deoxo-10-dihydroerythromycine a and derivatives thereof
US4496546A (en) * 1982-04-12 1985-01-29 Pfizer Inc. Erythromycin D and esters thereof
US4474768A (en) * 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
PH19293A (en) * 1982-11-15 1986-03-04 Pfizer Epimeric azahomoerythromycin,pharmaceutical composition containing the same and method of use thereof

Also Published As

Publication number Publication date
DK423184D0 (da) 1984-09-05
DK157877C (da) 1990-07-23
EP0136830A3 (en) 1986-03-19
ES8604256A1 (es) 1986-01-16
DK157877B (da) 1990-02-26
JPS6072897A (ja) 1985-04-24
EP0136830A2 (en) 1985-04-10
DK423184A (da) 1985-03-07
GR80278B (en) 1985-01-04
CA1240320A (en) 1988-08-09
US4465674A (en) 1984-08-14

Similar Documents

Publication Publication Date Title
ES533753A0 (es) Un procedimiento para la preparacion de nuevas fenoxialquil-1-2-4-triazolonas.
ES548672A0 (es) Un procedimiento para la preparacion de un derivado de dihi-dropiridina
ES529171A0 (es) Un procedimiento para la preparacion de una cefalosporina.
ES521728A0 (es) Un procedimiento para la preparacion de una sal de adicion de un acido bencenosulfonico de la sultamicilina.
ES535625A0 (es) Un procedimiento para la preparacion de 9-deoxo-9a-metil-9a-aza-9a-homoeritromicina d o una sal de la misma
ES541386A0 (es) Un procedimiento para la preparacion de un compuesto
ES543646A0 (es) Un procedimiento para la preparacion de derivados esteroida-les
ES530418A0 (es) Un procedimiento para la preparacion de pirazolopiridinas.
ES537487A0 (es) Un procedimiento para la preparacion de oxazolidinas
ES529462A0 (es) Un procedimiento para la preparacion de nuevos derivados de benzotiazina
ES538829A0 (es) Procedimiento para la preparacion de una 5-pirimidincarboxamida o tiocarboxamida
ES530081A0 (es) Un procedimiento para la preparacion de una macrolida
MX156049A (es) Un procedimiento para la preparacion de una n - piperazinilalcanolanilida
ES530153A0 (es) Un procedimiento para la preparacion de compuestos de beta-lactama
ES543491A0 (es) Un procedimiento para la preparacion de una sal metalica de un monoalquilfosfato.
ES532172A0 (es) Un procedimiento para la preparacion de derivados de pirimidona
ES537349A0 (es) Un procedimiento para la preparacion de un aminotiol cuaternario
ES531792A0 (es) Un procedimiento para la preparacion de un compuesto.
ES530973A0 (es) Un procedimiento para la preparacion de benzoquinolicinas
ES544640A0 (es) Un procedimiento para la preparacion de una cefalosporina
ES535493A0 (es) Un procedimiento para la preparacion de un compuesto de b-lactama
ES535392A0 (es) Un procedimiento para la preparacion de derivados de imidazobenzodiacepina
ES515237A0 (es) Un procedimiento para la preparacion de una sal de amonio cuaternario.
ES546356A0 (es) Un procedimiento para la preparacion de nuevos derivados delacido tiazolilacetico
ES528985A0 (es) Un procedimiento para la preparacion de una b- lactama

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19970401