ES529349A0 - Un procedimiento para la preparacion de derivados de acilmorfinano - Google Patents
Un procedimiento para la preparacion de derivados de acilmorfinanoInfo
- Publication number
- ES529349A0 ES529349A0 ES529349A ES529349A ES529349A0 ES 529349 A0 ES529349 A0 ES 529349A0 ES 529349 A ES529349 A ES 529349A ES 529349 A ES529349 A ES 529349A ES 529349 A0 ES529349 A0 ES 529349A0
- Authority
- ES
- Spain
- Prior art keywords
- acilmorfinan
- derivatives
- procedure
- preparation
- acilmorfinan derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
- C07D221/22—Bridged ring systems
- C07D221/28—Morphinans
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/06—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/319,482 US4374139A (en) | 1981-11-09 | 1981-11-09 | Levorotatory N-substituted acylmorphinans useful as analgesic agents |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8506635A1 ES8506635A1 (es) | 1985-08-01 |
| ES529349A0 true ES529349A0 (es) | 1985-08-01 |
Family
ID=23242421
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES517222A Granted ES517222A0 (es) | 1981-11-09 | 1982-11-08 | Un procedimiento para la preparacion de derivados de acilmorrfinano. |
| ES529349A Granted ES529349A0 (es) | 1981-11-09 | 1984-02-01 | Un procedimiento para la preparacion de derivados de acilmorfinano |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES517222A Granted ES517222A0 (es) | 1981-11-09 | 1982-11-08 | Un procedimiento para la preparacion de derivados de acilmorrfinano. |
Country Status (18)
| Country | Link |
|---|---|
| US (1) | US4374139A (es) |
| EP (1) | EP0079556A3 (es) |
| JP (1) | JPS5888364A (es) |
| KR (1) | KR840002357A (es) |
| AU (1) | AU9027682A (es) |
| CA (1) | CA1195324A (es) |
| DK (1) | DK491582A (es) |
| ES (2) | ES517222A0 (es) |
| FI (1) | FI823824L (es) |
| GR (1) | GR78317B (es) |
| HU (1) | HU187425B (es) |
| IL (1) | IL67180A0 (es) |
| MC (1) | MC1490A1 (es) |
| NO (1) | NO823707L (es) |
| NZ (1) | NZ202404A (es) |
| PH (1) | PH18458A (es) |
| PT (1) | PT75815B (es) |
| ZA (1) | ZA827905B (es) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4423221A (en) * | 1982-06-10 | 1983-12-27 | Sisa Pharmaceutical Laboratories, Inc. | 7-Carboethoxy-morphinan-6-one compounds |
| US4454141A (en) * | 1982-09-23 | 1984-06-12 | Sisa Pharmaceutical Laboratories, Inc. | Trans-B/C-7-(1-hydroxypentyl)-3-methoxy-17 methyl-6,7-didehydromorphinans, and methods of relieving pain with them |
| EP0184041A1 (en) * | 1984-11-13 | 1986-06-11 | Miles Inc. | 6-Methylene morphinan purification technique |
| US4929622A (en) * | 1987-09-24 | 1990-05-29 | Hoechst-Roussel Pharmaceuticals, Inc. | 2,6-Methanopyrrolo-3-benzazocines |
| DE4304450A1 (de) * | 1993-02-13 | 1994-08-18 | Boehringer Mannheim Gmbh | System zur Zubereitung von Flüssigkeiten |
| CA2426942C (en) * | 2000-10-31 | 2014-06-03 | Mark P. Wentland | 8-carboxamido-2,6-methano-3-benzazocines |
| AU2002322720B2 (en) | 2001-07-25 | 2008-11-13 | Raptor Pharmaceutical Inc. | Compositions and methods for modulating blood-brain barrier transport |
| US20040204862A1 (en) * | 2003-04-11 | 2004-10-14 | Wainer Irving W. | Computer-based model for identification and characterization for non-competitive inhibitors of nicotinic acetylcholine receptors and related ligand-gated ion channel receptors |
| EP2392258B1 (en) | 2005-04-28 | 2014-10-08 | Proteus Digital Health, Inc. | Pharma-informatics system |
| MX2009002893A (es) | 2006-09-18 | 2009-07-10 | Raptor Pharmaceutical Inc | Tratamiento de trastornos hepaticos mediante la administracion de conjugados de la proteina asociada al receptor (rap). |
| TR201908314T4 (tr) | 2009-02-20 | 2019-06-21 | 2 Bbb Medicines B V | Glutatyon bazlı ilaç dağıtım sistemi. |
| IL295075A (en) | 2009-05-06 | 2022-09-01 | Laboratory Skin Care Inc | Preparations for administration through the skin that include complexes of an active substance with calcium phosphate and methods of using them |
| HUE043963T2 (hu) | 2009-12-04 | 2019-09-30 | Alkermes Pharma Ireland Ltd | Morfinán származékok gyógyszer-túladagolás kezelésére |
| EP2550253B9 (en) | 2010-03-22 | 2016-09-21 | Rensselaer Polytechnic Institute | Morphinane derivatives containing a carboxamide group as opioid receptor ligands |
| US20120077778A1 (en) | 2010-09-29 | 2012-03-29 | Andrea Bourdelais | Ladder-Frame Polyether Conjugates |
| WO2013003720A1 (en) | 2011-06-29 | 2013-01-03 | Alkermes, Inc. | Peripherally acting opioid compounds |
| US9211293B2 (en) | 2011-12-15 | 2015-12-15 | Alkermes Pharma Ireland Limited | Opioid agonist antagonist combinations |
| WO2014190271A2 (en) | 2013-05-24 | 2014-11-27 | Alkermes Pharma Ireland Limted | Methods for treating depressive symptoms |
| JP2016519161A (ja) | 2013-05-24 | 2016-06-30 | アルカームス ファーマ アイルランド リミテッド | モルファン及びモルフィナン類似物及び使用の方法 |
| WO2018125716A1 (en) * | 2017-01-02 | 2018-07-05 | Purdue Pharma L.P. | Morphinan derivatives and use thereof |
| EP4243768A1 (en) | 2020-11-12 | 2023-09-20 | Alkermes Pharma Ireland Limited | Immediate release multilayer tablet |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3723437A (en) * | 1970-09-15 | 1973-03-27 | American Home Prod | 4,10-(methaniminomethano phenanthrene derivatives |
| ZA73988B (en) * | 1972-03-10 | 1973-10-31 | Hoffmann La Roche | Morphinan derivatives |
| US3914233A (en) * | 1972-10-20 | 1975-10-21 | Hoffmann La Roche | 4-Hydroxy-N-substituted morphinan derivatives |
-
1981
- 1981-11-09 US US06/319,482 patent/US4374139A/en not_active Expired - Fee Related
- 1981-12-29 GR GR69729A patent/GR78317B/el unknown
-
1982
- 1982-10-28 ZA ZA827905A patent/ZA827905B/xx unknown
- 1982-11-05 IL IL67180A patent/IL67180A0/xx unknown
- 1982-11-05 NZ NZ202404A patent/NZ202404A/en unknown
- 1982-11-05 DK DK491582A patent/DK491582A/da not_active Application Discontinuation
- 1982-11-08 HU HU823578A patent/HU187425B/hu unknown
- 1982-11-08 MC MC821609A patent/MC1490A1/xx unknown
- 1982-11-08 JP JP57194799A patent/JPS5888364A/ja active Pending
- 1982-11-08 CA CA000415102A patent/CA1195324A/en not_active Expired
- 1982-11-08 ES ES517222A patent/ES517222A0/es active Granted
- 1982-11-08 PT PT75815A patent/PT75815B/pt unknown
- 1982-11-08 NO NO823707A patent/NO823707L/no unknown
- 1982-11-08 PH PH28105A patent/PH18458A/en unknown
- 1982-11-08 FI FI823824A patent/FI823824L/fi not_active Application Discontinuation
- 1982-11-08 EP EP82110285A patent/EP0079556A3/de not_active Ceased
- 1982-11-09 KR KR1019820005066A patent/KR840002357A/ko unknown
- 1982-11-09 AU AU90276/82A patent/AU9027682A/en not_active Abandoned
-
1984
- 1984-02-01 ES ES529349A patent/ES529349A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| EP0079556A3 (de) | 1983-08-24 |
| FI823824L (fi) | 1983-05-10 |
| ES8506635A1 (es) | 1985-08-01 |
| DK491582A (da) | 1983-05-10 |
| NZ202404A (en) | 1985-11-08 |
| NO823707L (no) | 1983-05-10 |
| ZA827905B (en) | 1983-08-31 |
| JPS5888364A (ja) | 1983-05-26 |
| US4374139A (en) | 1983-02-15 |
| IL67180A0 (en) | 1983-03-31 |
| CA1195324A (en) | 1985-10-15 |
| ES8500948A1 (es) | 1984-12-01 |
| KR840002357A (ko) | 1984-06-25 |
| AU9027682A (en) | 1983-05-19 |
| PT75815A (en) | 1982-12-01 |
| MC1490A1 (fr) | 1983-09-12 |
| FI823824A0 (fi) | 1982-11-08 |
| PH18458A (en) | 1985-07-18 |
| EP0079556A2 (de) | 1983-05-25 |
| PT75815B (en) | 1986-01-21 |
| ES517222A0 (es) | 1984-12-01 |
| GR78317B (es) | 1984-09-26 |
| HU187425B (en) | 1986-01-28 |
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