ES527711A0 - Un procedimiento para la preparacion de derivados de -lactama - Google Patents
Un procedimiento para la preparacion de derivados de -lactamaInfo
- Publication number
- ES527711A0 ES527711A0 ES527711A ES527711A ES527711A0 ES 527711 A0 ES527711 A0 ES 527711A0 ES 527711 A ES527711 A ES 527711A ES 527711 A ES527711 A ES 527711A ES 527711 A0 ES527711 A0 ES 527711A0
- Authority
- ES
- Spain
- Prior art keywords
- procedure
- preparation
- lactam derivatives
- lactam
- derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
- C07D231/22—One oxygen atom attached in position 3 or 5 with aryl radicals attached to ring nitrogen atoms
- C07D231/26—1-Phenyl-3-methyl-5- pyrazolones, unsubstituted or substituted on the phenyl ring
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8209426 | 1982-03-31 |
Publications (2)
Publication Number | Publication Date |
---|---|
ES527711A0 true ES527711A0 (es) | 1986-02-01 |
ES8604511A1 ES8604511A1 (es) | 1986-02-01 |
Family
ID=10529420
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES521192A Granted ES521192A0 (es) | 1982-03-31 | 1983-03-30 | Un procedimiento para la preparacion de derivados de b-lactama. |
ES527711A Expired ES8604511A1 (es) | 1982-03-31 | 1983-12-01 | Un procedimiento para la preparacion de derivados de -lactama |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES521192A Granted ES521192A0 (es) | 1982-03-31 | 1983-03-30 | Un procedimiento para la preparacion de derivados de b-lactama. |
Country Status (7)
Country | Link |
---|---|
US (1) | US4537886A (es) |
EP (1) | EP0090656A1 (es) |
JP (1) | JPS58183692A (es) |
AU (1) | AU1294383A (es) |
ES (2) | ES521192A0 (es) |
NZ (1) | NZ203734A (es) |
ZA (1) | ZA832226B (es) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8409986D0 (en) * | 1984-04-17 | 1984-05-31 | Beecham Group Plc | Beta-lactam antibacterial agents |
DE3508258A1 (de) * | 1985-03-08 | 1986-09-18 | Bayer Ag, 5090 Leverkusen | Ss-lactamantibiotika, verfahren zur herstellung und ihre verwendung als und in arzneimitteln |
DE3509618A1 (de) * | 1985-03-16 | 1986-09-18 | Bayer Ag, 5090 Leverkusen | Ss-lactam-antibiotika, verfahren zur herstellung und ihre verwendung als arzneimittel |
US4870168A (en) * | 1987-02-26 | 1989-09-26 | Bristol-Myers Company | 3-Unsaturated alkyl cephems from 3-triflyl cephems |
DE3803169A1 (de) * | 1988-02-03 | 1989-08-17 | Bayer Ag | Ss-lactam-antibiotika, verfahren zu ihrer herstellung und ihre verwendung als und in arzneimitteln |
US5128336A (en) * | 1988-03-23 | 1992-07-07 | Eli Lilly And Company | 3-(substituted)-1-carba(dethia)-3-cephems |
US20050245498A1 (en) * | 2002-05-14 | 2005-11-03 | Shoichet Brian K | Sterically-awkward beta-lactamase inhibitors |
US20080146535A1 (en) * | 2003-04-30 | 2008-06-19 | Tomasz Glinka | Compositions comprising carbacephem beta-lactam antibiotics and beta-lactamase inhibitors |
EA201070504A1 (ru) * | 2007-10-25 | 2010-12-30 | Эйкеоджен, Инк. | КАРБАЦЕФЕМ β-ЛАКТАМОВЫЕ АНТИБИОТИКИ |
WO2010030810A1 (en) * | 2008-09-10 | 2010-03-18 | Achaogen, Inc. | Carbacephem beta-lactam antibiotics |
WO2017106064A1 (en) * | 2015-12-15 | 2017-06-22 | Merck Sharp & Dohme Corp. | Biaryl monobactam compounds and methods of use thereof for the treatment of bacterial infections |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE2448966A1 (de) * | 1973-10-19 | 1975-04-30 | Yamanouchi Pharma Co Ltd | Penicillinderivate |
JPS5195090A (en) * | 1975-02-14 | 1976-08-20 | 66 * dd22 * 33 hidorokishipiridajin 44 karubokishiamido * 22 * paraahidorokishifueniru * asetoamido * penishiransanno seiho | |
DE2720579A1 (de) * | 1977-05-07 | 1978-11-09 | Bayer Ag | Beta-lactam-verbindungen, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel |
DE2810083A1 (de) * | 1978-03-08 | 1979-09-20 | Bayer Ag | Beta-lactam-verbindungen |
JPS5616489A (en) * | 1979-07-20 | 1981-02-17 | Ajinomoto Co Inc | Imidazolecarboxylic acid derivative |
-
1983
- 1983-03-29 AU AU12943/83A patent/AU1294383A/en not_active Abandoned
- 1983-03-29 ZA ZA832226A patent/ZA832226B/xx unknown
- 1983-03-29 NZ NZ203734A patent/NZ203734A/en unknown
- 1983-03-29 US US06/479,953 patent/US4537886A/en not_active Expired - Fee Related
- 1983-03-30 ES ES521192A patent/ES521192A0/es active Granted
- 1983-03-30 EP EP83301786A patent/EP0090656A1/en not_active Ceased
- 1983-03-30 JP JP58054989A patent/JPS58183692A/ja active Pending
- 1983-12-01 ES ES527711A patent/ES8604511A1/es not_active Expired
Also Published As
Publication number | Publication date |
---|---|
EP0090656A1 (en) | 1983-10-05 |
NZ203734A (en) | 1986-03-14 |
ES8405411A1 (es) | 1984-06-01 |
ES8604511A1 (es) | 1986-02-01 |
JPS58183692A (ja) | 1983-10-26 |
ES521192A0 (es) | 1984-06-01 |
AU1294383A (en) | 1983-10-06 |
US4537886A (en) | 1985-08-27 |
ZA832226B (en) | 1984-02-29 |
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