ES500870A0 - Un procedimiento para la preparacion de nuevos derivados de triariltiazol. - Google Patents

Un procedimiento para la preparacion de nuevos derivados de triariltiazol.

Info

Publication number
ES500870A0
ES500870A0 ES500870A ES500870A ES500870A0 ES 500870 A0 ES500870 A0 ES 500870A0 ES 500870 A ES500870 A ES 500870A ES 500870 A ES500870 A ES 500870A ES 500870 A0 ES500870 A0 ES 500870A0
Authority
ES
Spain
Prior art keywords
triariltiazole
derivatives
procedure
preparation
new
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES500870A
Other languages
English (en)
Other versions
ES8205210A1 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Publication of ES8205210A1 publication Critical patent/ES8205210A1/es
Publication of ES500870A0 publication Critical patent/ES500870A0/es
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/24Radicals substituted by oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/63Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by introduction of halogen; by substitution of halogen atoms by other halogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
ES500870A 1980-04-02 1981-03-30 Un procedimiento para la preparacion de nuevos derivados de triariltiazol. Granted ES500870A0 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/136,591 US4322428A (en) 1980-04-02 1980-04-02 2(4-Fluorophenyl)-4,5,-bis(4-methoxyphenyl)thiazole and method of use

Publications (2)

Publication Number Publication Date
ES8205210A1 ES8205210A1 (es) 1982-06-01
ES500870A0 true ES500870A0 (es) 1982-06-01

Family

ID=22473504

Family Applications (1)

Application Number Title Priority Date Filing Date
ES500870A Granted ES500870A0 (es) 1980-04-02 1981-03-30 Un procedimiento para la preparacion de nuevos derivados de triariltiazol.

Country Status (24)

Country Link
US (1) US4322428A (es)
EP (1) EP0037274A1 (es)
JP (1) JPS56152469A (es)
AR (1) AR226098A1 (es)
AU (1) AU6881081A (es)
BG (1) BG35045A3 (es)
CA (1) CA1157864A (es)
CS (1) CS217994B2 (es)
DD (1) DD157799A5 (es)
DK (1) DK142381A (es)
ES (1) ES500870A0 (es)
FI (1) FI810935L (es)
GB (1) GB2073189A (es)
GR (1) GR73694B (es)
HU (1) HU182705B (es)
IL (1) IL62491A0 (es)
NZ (1) NZ196625A (es)
PH (1) PH16945A (es)
PL (1) PL128570B1 (es)
PT (1) PT72757B (es)
RO (1) RO81686B (es)
SU (1) SU957765A3 (es)
YU (1) YU80281A (es)
ZA (1) ZA812019B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4533666A (en) * 1983-06-22 1985-08-06 Eli Lilly And Company 6-Phenyl-2,3-bis-(4-methoxyphenyl)-pyridine derivatives having anti-inflammatory activity
US4500533A (en) * 1983-06-22 1985-02-19 Eli Lilly And Company 2,4,5-Triaryl pyrimidines and a method of treating pain, fever, thrombosis, inflammation and arthritis
US4495202A (en) * 1983-06-22 1985-01-22 Eli Lilly And Company Terphenyl derivatives and pharmaceutical uses thereof
US4659726A (en) * 1984-04-19 1987-04-21 Kanebo, Ltd. Novel 4,5-Bis (4-methoxyphenyl)-2-(pyrrol-2-yl) thiazoles and pharmaceutical composition containing the same
DE69132944T2 (de) 1990-11-30 2002-11-21 Otsuka Pharmaceutical Co., Ltd. Azolederivate als Inhibitor von Superoxide-Radikalen
MY128323A (en) 1996-09-30 2007-01-31 Otsuka Pharma Co Ltd Thiazole derivatives for inhibition of cytokine production and of cell adhesion
CN100383131C (zh) * 2005-06-15 2008-04-23 浙江大学 2-对三氟甲苯-4-甲基-5-噻唑甲酸乙酯的合成方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3560514A (en) * 1966-09-26 1971-02-02 Upjohn Co 2-(lithiummethyl)-4,5-dianisylthiazole
US3558644A (en) * 1966-09-26 1971-01-26 Upjohn Co 2-substituted-4,5-dianisylthiazoles
US3458526A (en) * 1966-09-26 1969-07-29 Upjohn Co Certain 2-amino-4,5-bis(p-methoxyphenyl)thiazoles
GB1145884A (en) * 1966-11-18 1969-03-19 Wyeth John & Brother Ltd Thiazole derivatives
IE32084B1 (en) * 1967-06-07 1973-04-04 Wyeth John & Brother Ltd Thiazole derivatives
GB1539450A (en) * 1976-06-08 1979-01-31 Wyeth John & Brother Ltd Thiazole derivatives
US4197306A (en) * 1977-06-30 1980-04-08 Uniroyal, Inc. Aryl-substituted thiazoles
US4168315A (en) * 1977-09-28 1979-09-18 The Upjohn Company Dianisyl thiazole compound, compositions and method of antithrombotic treatment

Also Published As

Publication number Publication date
JPS56152469A (en) 1981-11-26
CS217994B2 (en) 1983-02-25
RO81686A (ro) 1983-04-29
RO81686B (ro) 1983-04-30
BG35045A3 (en) 1984-01-16
ES8205210A1 (es) 1982-06-01
PL230426A1 (es) 1981-12-23
IL62491A0 (en) 1981-05-20
FI810935L (fi) 1981-10-03
GR73694B (es) 1984-04-03
NZ196625A (en) 1983-09-30
CA1157864A (en) 1983-11-29
YU80281A (en) 1983-09-30
GB2073189A (en) 1981-10-14
EP0037274A1 (en) 1981-10-07
DD157799A5 (de) 1982-12-08
DK142381A (da) 1981-10-03
PH16945A (en) 1984-04-24
ZA812019B (en) 1982-11-24
US4322428A (en) 1982-03-30
SU957765A3 (ru) 1982-09-07
PT72757A (en) 1981-04-01
HU182705B (en) 1984-03-28
PT72757B (en) 1982-03-23
AR226098A1 (es) 1982-05-31
AU6881081A (en) 1981-10-08
PL128570B1 (en) 1984-02-29

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