ES478011A1 - Un procedimiento de preparacion de nuevos derivados de la bencenopropanamina. - Google Patents
Un procedimiento de preparacion de nuevos derivados de la bencenopropanamina.Info
- Publication number
- ES478011A1 ES478011A1 ES478011A ES478011A ES478011A1 ES 478011 A1 ES478011 A1 ES 478011A1 ES 478011 A ES478011 A ES 478011A ES 478011 A ES478011 A ES 478011A ES 478011 A1 ES478011 A1 ES 478011A1
- Authority
- ES
- Spain
- Prior art keywords
- hydrogen
- group
- bromine
- chlorine
- alkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/16—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by singly-bound oxygen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Abstract
Un procedimiento de preparación de nuevos derivados de la benceno-propanamina, así como de sus sales de adición con los ácidos minerales u orgánicos, que responden a la fórmula general (I''): **(Fórmula)** en la cual X representa un átomo de hidrógeno, un átomo de flúor, de cloro o de bromo, R1 representa un átomo de hidrógeno o un radical alcohilo que contiene de 1 a 5 átomos de carbono, R2 representa un radical alcohilo que contiene de 1 a 5 átomos de carbono, y R3 representa un átomo de hidrógeno, un átomo de cloro o de bromo, un radical trifluorometilo, un radical metilo o un radical metoxi y R4 representa un radical nitro, o bien R3 representa un radical amino o acetamido y R4 representa un átomo de hidrógeno.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7805335A FR2432500A1 (fr) | 1978-02-24 | 1978-02-24 | Nouveaux derives de la benzene propanamine et leurs sels, procede de preparation et application a titre de medicaments |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES478011A1 true ES478011A1 (es) | 1979-07-01 |
Family
ID=9205011
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES478011A Expired ES478011A1 (es) | 1978-02-24 | 1979-02-23 | Un procedimiento de preparacion de nuevos derivados de la bencenopropanamina. |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US4296126A (es) |
| JP (1) | JPS54122236A (es) |
| AT (1) | AT362347B (es) |
| BE (1) | BE874416A (es) |
| CA (1) | CA1116635A (es) |
| CH (1) | CH639637A5 (es) |
| DE (1) | DE2907217C2 (es) |
| ES (1) | ES478011A1 (es) |
| FR (1) | FR2432500A1 (es) |
| GB (1) | GB2017681B (es) |
| IT (1) | IT1114717B (es) |
| NL (1) | NL7901457A (es) |
Families Citing this family (25)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4692469A (en) * | 1982-09-07 | 1987-09-08 | Ciba-Geigy Corporation | Propylamine derivatives |
| US4824868A (en) * | 1982-09-07 | 1989-04-25 | Ciba-Geigy Corporation | Propylamine derivatives useful for the treatment of dementia |
| JPH056143Y2 (es) * | 1986-10-09 | 1993-02-17 | ||
| DK630987D0 (da) * | 1987-12-01 | 1987-12-01 | Ferrosan As | Aryloxyphenylpropylaminer, deres fremstilling og anvendelse |
| US5166437A (en) * | 1989-03-03 | 1992-11-24 | Orion-Yhtyma Oy | Process for the preparation of fluoxetine |
| DK258389D0 (da) * | 1989-05-26 | 1989-05-26 | Ferrosan As | Aryloxyphenylpropylaminer, deres fremstilling og anvendelse |
| US5320825A (en) * | 1991-05-01 | 1994-06-14 | Trustees Of The University Of Pennsylvania | Serotonin reuptake inhibitors for S.P.E.C.T. imaging |
| EP0576766A1 (en) * | 1992-06-29 | 1994-01-05 | Novo Nordisk A/S | Propanolamine derivatives, their preparation and use |
| GB0004152D0 (en) * | 2000-02-23 | 2000-04-12 | Astrazeneca Uk Ltd | Novel compounds |
| GB0004153D0 (en) * | 2000-02-23 | 2000-04-12 | Astrazeneca Uk Ltd | Novel use |
| GB0004151D0 (en) * | 2000-02-23 | 2000-04-12 | Astrazeneca Uk Ltd | Novel use |
| GB0004149D0 (en) * | 2000-02-23 | 2000-04-12 | Astrazeneca Uk Ltd | Novel compounds |
| US6313350B1 (en) | 2001-01-31 | 2001-11-06 | Grayson Walker Stowell | Form a of fluoxetine hydrochloride |
| US6258853B1 (en) | 2001-01-31 | 2001-07-10 | Grayson Walker Stowell | Form a of fluoxetine hydrochloride |
| US6316672B1 (en) | 2001-01-31 | 2001-11-13 | Grayson Walker Stowell | Form a of fluoxetine hydrochloride |
| US6310251B1 (en) | 2001-01-31 | 2001-10-30 | Grayson Walker Stowell | Form a of fluoxetine hydrochloride |
| US6310250B1 (en) | 2001-01-31 | 2001-10-30 | Grayson Walker Stowell | Form A of fluoxetine hydrochloride |
| JP2004525912A (ja) * | 2001-03-06 | 2004-08-26 | イーライ・リリー・アンド・カンパニー | モノアミン取込の阻害剤 |
| AR035700A1 (es) * | 2001-05-08 | 2004-06-23 | Astrazeneca Ab | Derivados de arilheteroalquilamina, composicion farmaceutica, usos de estos derivados para la fabricacion de medicamentos, metodos de tratamiento, y proceso para la preparacion de estos derivados |
| SE0102640D0 (sv) * | 2001-07-31 | 2001-07-31 | Astrazeneca Ab | Novel compounds |
| SE0203304D0 (sv) * | 2002-11-07 | 2002-11-07 | Astrazeneca Ab | Novel Coumpounds |
| US6846957B2 (en) * | 2002-11-22 | 2005-01-25 | Board Of Regents, The University Of Texas System | Synthesis of 3-aminomethyl-1-propanol, a fluoxetine precursor |
| WO2008081477A1 (en) * | 2007-01-04 | 2008-07-10 | Natco Pharma Limited | 3-aryloxy 3-substituted propanamines |
| EP2161998B1 (en) * | 2007-06-04 | 2015-09-02 | Intra-Cellular Therapies, Inc. | Pyridine derivatives as NET/SERT modulators |
| WO2014046544A1 (en) * | 2012-09-21 | 2014-03-27 | Aapa B.V. | Substituted 3-heteroaryloxy-3-(hetero)aryl-propylamines as serotonin transporter and serotonin ht2c receptor modulators |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2683742A (en) * | 1951-02-23 | 1954-07-13 | Searle & Co | Nu, nu-disubstituted omega-arylmethoxy-omega-arylalkylamine derivatives |
| ES251290A1 (es) * | 1958-08-21 | 1960-04-01 | Parke Davis & Co | Un procedimiento para la producciën de alcohilaminas arilsustituidas |
| US3496195A (en) * | 1966-05-11 | 1970-02-17 | Chinoin Gyogyszer Es Vegyeszet | D-o-bromo-phenyl-isopropyl-methylpropinylamine and its salts |
| GB1343527A (en) * | 1971-07-30 | 1974-01-10 | Cerm Cent Europ Rech Mauvernay | Amino-propanol derivatives |
| US4314081A (en) * | 1974-01-10 | 1982-02-02 | Eli Lilly And Company | Arloxyphenylpropylamines |
| US4018895A (en) * | 1974-01-10 | 1977-04-19 | Eli Lilly And Company | Aryloxyphenylpropylamines in treating depression |
-
1978
- 1978-02-24 FR FR7805335A patent/FR2432500A1/fr active Granted
-
1979
- 1979-02-22 US US06/013,831 patent/US4296126A/en not_active Expired - Lifetime
- 1979-02-23 IT IT48102/79A patent/IT1114717B/it active
- 1979-02-23 AT AT143379A patent/AT362347B/de not_active IP Right Cessation
- 1979-02-23 CA CA000322221A patent/CA1116635A/fr not_active Expired
- 1979-02-23 DE DE2907217A patent/DE2907217C2/de not_active Expired
- 1979-02-23 CH CH181979A patent/CH639637A5/fr not_active IP Right Cessation
- 1979-02-23 NL NL7901457A patent/NL7901457A/xx not_active Application Discontinuation
- 1979-02-23 JP JP1989479A patent/JPS54122236A/ja active Granted
- 1979-02-23 BE BE0/193668A patent/BE874416A/xx not_active IP Right Cessation
- 1979-02-23 ES ES478011A patent/ES478011A1/es not_active Expired
- 1979-02-26 GB GB7906712A patent/GB2017681B/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| CH639637A5 (fr) | 1983-11-30 |
| IT1114717B (it) | 1986-01-27 |
| DE2907217A1 (de) | 1979-08-30 |
| JPS54122236A (en) | 1979-09-21 |
| US4296126A (en) | 1981-10-20 |
| FR2432500B1 (es) | 1981-01-16 |
| GB2017681B (en) | 1982-08-04 |
| AT362347B (de) | 1981-05-11 |
| CA1116635A (fr) | 1982-01-19 |
| GB2017681A (en) | 1979-10-10 |
| NL7901457A (nl) | 1979-08-28 |
| IT7948102A0 (it) | 1979-02-23 |
| JPS638935B2 (es) | 1988-02-25 |
| DE2907217C2 (de) | 1985-12-12 |
| FR2432500A1 (fr) | 1980-02-29 |
| ATA143379A (de) | 1980-10-15 |
| BE874416A (fr) | 1979-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Patent lapsed |
Effective date: 19960506 |