ES449777A1 - Substituted pyrimido-quinoline derivatives and pharmaceutical compositions containing them - Google Patents

Substituted pyrimido-quinoline derivatives and pharmaceutical compositions containing them

Info

Publication number
ES449777A1
ES449777A1 ES449777A ES449777A ES449777A1 ES 449777 A1 ES449777 A1 ES 449777A1 ES 449777 A ES449777 A ES 449777A ES 449777 A ES449777 A ES 449777A ES 449777 A1 ES449777 A1 ES 449777A1
Authority
ES
Spain
Prior art keywords
pharmaceutical compositions
compositions containing
quinoline derivatives
formula
substituted pyrimido
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES449777A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of ES449777A1 publication Critical patent/ES449777A1/en
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/08Antiallergic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

A process for the production of pharmaceutically active compounds of the formula: ** (See formula) ** wherein R1 and R2 are each independently selected from hydrogen, C1-5 alkyl, C1-5 alkoxy, fluorine and chlorine or R1 and R2 in combination may form a group -O-CH2-CH2-O- or - O-CH2-O- and R3 is selected from chlorine, bromine and C1-5 alkoxy, characterized in that a coupling is carried out with dehydration of an acid of the formula ** (See formula) ** with a 5-amino-tetrazole. (Machine-translation by Google Translate, not legally binding)
ES449777A 1975-08-01 1976-07-12 Substituted pyrimido-quinoline derivatives and pharmaceutical compositions containing them Expired ES449777A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US60103975A 1975-08-01 1975-08-01

Publications (1)

Publication Number Publication Date
ES449777A1 true ES449777A1 (en) 1977-08-16

Family

ID=24406004

Family Applications (1)

Application Number Title Priority Date Filing Date
ES449777A Expired ES449777A1 (en) 1975-08-01 1976-07-12 Substituted pyrimido-quinoline derivatives and pharmaceutical compositions containing them

Country Status (31)

Country Link
JP (1) JPS5231098A (en)
AR (1) AR213099A1 (en)
AT (1) AT351028B (en)
AU (1) AU497412B2 (en)
BE (1) BE843952A (en)
BG (1) BG31229A3 (en)
CA (1) CA1060441A (en)
CH (1) CH616679A5 (en)
CS (1) CS195731B2 (en)
DD (1) DD126735A5 (en)
DE (1) DE2630469C2 (en)
DK (1) DK311276A (en)
EG (1) EG12424A (en)
ES (1) ES449777A1 (en)
FI (1) FI59409C (en)
FR (1) FR2319363A1 (en)
GB (1) GB1500666A (en)
GR (1) GR60549B (en)
HU (1) HU172063B (en)
IE (1) IE43028B1 (en)
IL (1) IL49924A (en)
LU (1) LU75369A1 (en)
NL (1) NL163514C (en)
NO (1) NO139786C (en)
NZ (1) NZ181317A (en)
PH (1) PH12132A (en)
PT (1) PT65349B (en)
SE (1) SE414175B (en)
SU (1) SU685156A3 (en)
YU (1) YU185076A (en)
ZA (1) ZA763876B (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2720085A1 (en) 1977-05-05 1978-11-16 Hoechst Ag PYRIMIDO (6.1-A) ISOCHINOLIN-2-ON DERIVATIVES
US4127720A (en) * 1977-09-21 1978-11-28 Bristol-Myers Company Pyrimido[2,1-a]isoquinoline derivatives having antiallergy activity
US4192944A (en) * 1978-04-03 1980-03-11 Bristol-Myers Company Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents
JPS55138593U (en) * 1979-03-27 1980-10-02
AU5533996A (en) * 1996-04-04 1997-10-29 University Of Nebraska Board Of Regents Synthetic triple helix-forming compounds

Also Published As

Publication number Publication date
PH12132A (en) 1978-11-07
IL49924A0 (en) 1976-08-31
AT351028B (en) 1979-07-10
AU1578476A (en) 1978-01-12
HU172063B (en) 1978-05-28
NO139786C (en) 1979-05-09
PT65349A (en) 1976-08-01
FI762016A (en) 1977-02-02
CA1060441A (en) 1979-08-14
PT65349B (en) 1978-01-06
NZ181317A (en) 1978-03-06
IL49924A (en) 1979-03-12
JPS5231098A (en) 1977-03-09
LU75369A1 (en) 1977-04-04
SE7607099L (en) 1977-02-02
NO139786B (en) 1979-01-29
YU185076A (en) 1982-06-30
DK311276A (en) 1977-02-02
IE43028L (en) 1977-02-01
AR213099A1 (en) 1978-12-15
CS195731B2 (en) 1980-02-29
ATA512676A (en) 1978-12-15
GR60549B (en) 1978-06-14
AU497412B2 (en) 1978-12-14
DE2630469A1 (en) 1977-02-17
DD126735A5 (en) 1977-08-10
FI59409B (en) 1981-04-30
CH616679A5 (en) 1980-04-15
FR2319363A1 (en) 1977-02-25
NL163514C (en) 1980-09-15
EG12424A (en) 1979-03-31
SU685156A3 (en) 1979-09-05
DE2630469C2 (en) 1982-04-08
NL7607618A (en) 1977-02-03
NL163514B (en) 1980-04-15
FR2319363B1 (en) 1978-11-17
FI59409C (en) 1981-08-10
BE843952A (en) 1977-01-10
BG31229A3 (en) 1981-11-16
GB1500666A (en) 1978-02-08
IE43028B1 (en) 1980-12-03
NO762411L (en) 1977-02-02
ZA763876B (en) 1977-05-25
SE414175B (en) 1980-07-14

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19980302