ES434079A1 - Procedimiento para la obtencion de compuestos indolicos sus-tituidos. - Google Patents
Procedimiento para la obtencion de compuestos indolicos sus-tituidos.Info
- Publication number
- ES434079A1 ES434079A1 ES434079A ES434079A ES434079A1 ES 434079 A1 ES434079 A1 ES 434079A1 ES 434079 A ES434079 A ES 434079A ES 434079 A ES434079 A ES 434079A ES 434079 A1 ES434079 A1 ES 434079A1
- Authority
- ES
- Spain
- Prior art keywords
- substituted
- group
- indole
- residue
- aliphatic hydrocarbon
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
CH104774 | 1974-01-25 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES434079A1 true ES434079A1 (es) | 1977-03-01 |
Family
ID=4201215
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES434079A Expired ES434079A1 (es) | 1974-01-25 | 1975-01-23 | Procedimiento para la obtencion de compuestos indolicos sus-tituidos. |
Country Status (14)
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4999186A (en) * | 1986-06-27 | 1991-03-12 | The Procter & Gamble Company | Novel sunscreen agents, sunscreen compositions and methods for preventing sunburn |
CA2407677A1 (en) * | 2000-04-28 | 2002-10-28 | Baxter Healthcare Sa | 2-acyl indol derivatives and their use as anti-tumour agents |
DE10152306A1 (de) * | 2001-10-26 | 2003-07-24 | Asta Medica Ag | 2-Acylindolderivate mit neuen therapeutisch wertvollen Eigenschaften |
EP2207547A4 (en) * | 2007-10-05 | 2010-11-17 | Amira Pharmaceuticals Inc | PROTEIN INHIBITORS THAT ACTIVATE 5-LIPOXYGENASE |
DK2448938T5 (en) | 2009-06-29 | 2015-10-05 | Incyte Corp | Pyrimidinones AS PI3K inhibitors |
WO2011075643A1 (en) | 2009-12-18 | 2011-06-23 | Incyte Corporation | Substituted heteroaryl fused derivatives as pi3k inhibitors |
TW201130842A (en) | 2009-12-18 | 2011-09-16 | Incyte Corp | Substituted fused aryl and heteroaryl derivatives as PI3K inhibitors |
WO2011130342A1 (en) | 2010-04-14 | 2011-10-20 | Incyte Corporation | FUSED DERIVATIVES AS ΡI3Κδ INHIBITORS |
WO2011163195A1 (en) | 2010-06-21 | 2011-12-29 | Incyte Corporation | Fused pyrrole derivatives as pi3k inhibitors |
JP5961187B2 (ja) | 2010-12-20 | 2016-08-02 | インサイト・ホールディングス・コーポレイションIncyte Holdings Corporation | Pi3k阻害剤としてのn−(1−(置換フェニル)エチル)−9h−プリン−6−アミン |
US9108984B2 (en) | 2011-03-14 | 2015-08-18 | Incyte Corporation | Substituted diamino-pyrimidine and diamino-pyridine derivatives as PI3K inhibitors |
US9126948B2 (en) | 2011-03-25 | 2015-09-08 | Incyte Holdings Corporation | Pyrimidine-4,6-diamine derivatives as PI3K inhibitors |
EP3513793B1 (en) | 2011-09-02 | 2021-03-10 | Incyte Holdings Corporation | Heterocyclylamines as pi3k inhibitors |
AR090548A1 (es) | 2012-04-02 | 2014-11-19 | Incyte Corp | Azaheterociclobencilaminas biciclicas como inhibidores de pi3k |
US10077277B2 (en) | 2014-06-11 | 2018-09-18 | Incyte Corporation | Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors |
HUE053025T2 (hu) | 2015-02-27 | 2021-06-28 | Incyte Corp | Sók és eljárások PI3K inhibitor elõállítására |
WO2016183060A1 (en) | 2015-05-11 | 2016-11-17 | Incyte Corporation | Process for the synthesis of a phosphoinositide 3-kinase inhibitor |
US9988401B2 (en) | 2015-05-11 | 2018-06-05 | Incyte Corporation | Crystalline forms of a PI3K inhibitor |
-
1975
- 1975-01-08 DK DK3375*BA patent/DK3375A/da unknown
- 1975-01-10 SE SE7500262A patent/SE7500262L/xx unknown
- 1975-01-16 DE DE19752501468 patent/DE2501468A1/de active Pending
- 1975-01-16 NL NL7500535A patent/NL7500535A/xx unknown
- 1975-01-23 FR FR7502129A patent/FR2258853B1/fr not_active Expired
- 1975-01-23 GB GB299475A patent/GB1472342A/en not_active Expired
- 1975-01-23 AU AU77563/75A patent/AU7756375A/en not_active Expired
- 1975-01-23 ES ES434079A patent/ES434079A1/es not_active Expired
- 1975-01-24 ZA ZA00750522A patent/ZA75522B/xx unknown
- 1975-01-24 IE IE137/75A patent/IE40368B1/xx unknown
- 1975-01-24 IL IL46505A patent/IL46505A0/xx unknown
- 1975-01-24 AT AT53175A patent/ATA53175A/de not_active IP Right Cessation
- 1975-01-24 BE BE152675A patent/BE824742A/xx unknown
- 1975-01-25 JP JP50010179A patent/JPS50106969A/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
DK3375A (US06265458-20010724-C00056.png) | 1975-09-15 |
SE7500262L (US06265458-20010724-C00056.png) | 1975-07-28 |
AU7756375A (en) | 1976-07-29 |
IL46505A0 (en) | 1975-04-25 |
BE824742A (fr) | 1975-07-24 |
FR2258853A1 (US06265458-20010724-C00056.png) | 1975-08-22 |
FR2258853B1 (US06265458-20010724-C00056.png) | 1978-06-30 |
GB1472342A (en) | 1977-05-04 |
IE40368B1 (en) | 1979-05-09 |
DE2501468A1 (de) | 1975-07-31 |
ATA53175A (de) | 1977-08-15 |
IE40368L (en) | 1975-07-25 |
NL7500535A (nl) | 1975-07-29 |
JPS50106969A (US06265458-20010724-C00056.png) | 1975-08-22 |
ZA75522B (en) | 1976-01-28 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
ES434079A1 (es) | Procedimiento para la obtencion de compuestos indolicos sus-tituidos. | |
ES320294A1 (es) | Procedimiento para la preparacion de nuevos derivados del indol. | |
ES401623A1 (es) | Procedimiento para la obtencion de derivados de adenosina. | |
ES390979A1 (es) | Procedimiento para la obtencion de derivados del acido n- fluordiclorometiltio-sulfamidico. | |
ES394562A1 (es) | Un procedimiento para la preparacion de nuevos imidazoles. | |
ES372536A1 (es) | Procedimiento para la obtencion de 6-amino - 4,5 - dihidro - isotiazolo (4,5-d) pirimidinas. | |
ES328674A1 (es) | Procedimiento para la produccion de alcaloides. | |
ES378206A1 (es) | Procedimiento para la preparacion de nuevos 2-amino-5-ni- trotiazoles. | |
ES394533A1 (es) | Procedimiento para la obtencion de compuestos de 2-hidroxi-4'-fenoxibenzofenona. | |
ES369751A1 (es) | Procedimiento para la preparacion de nuevos derivados de indol. | |
ES430417A1 (es) | Procedimiento para preparar bromuro de amidoalquil-trifenil-fosfonio. | |
ES402117A1 (es) | Procedimiento para la obtencion de derivados de 2-fenil-2- imidazolina. | |
ES462774A1 (es) | Procedimiento para la obtencion de nuevos ftalil derivados de sulfamidas. | |
ES382623A1 (es) | Procedimiento para la preparacion de nuevos derivados de i-midazolidinona. | |
ES460932A3 (es) | Un procedimiento para la preparacion de compuestos derivadosde indol. | |
ES289751A1 (es) | Procedimiento para la obtenciën de granulados minusculos | |
ES382612A1 (es) | Procedimiento para la preparacion de nuevos derivados de imidazolidinona. | |
ES433843A1 (es) | Procedimiento para la obtencion de nuevos compuestos micro-bicidas. | |
ES351328A1 (es) | Procedimiento para la preparacion de los derivados de pros-cilaridina a. | |
ES313506A1 (es) | Procedimiento para la obtencion de derivados hidracinicos. | |
ES378756A1 (es) | Procedimiento para la preparacion de nuevos derivados de isoquinoleina. | |
ES398186A1 (es) | Procedimiento para la preparacion de 3-slfoalquil-6-hidro- xi-piridonas-(2). | |
ES325525A1 (es) | Un procedimiento para la sintesis de compuestos piridazinicos. | |
ES396389A1 (es) | Procedimiento para la obtencion de compuestos de acido 7-a-cilamino-cef-3-em-4-carboxilico. | |
ES377601A2 (es) | Procedimiento para la obtencion e acidos carboxilicos alfa-(amino-fenil)-alifaticos |