ES428213A1 - Dialkylaminoalkyl esters of penicillin and process for the preparation thereof - Google Patents

Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Info

Publication number
ES428213A1
ES428213A1 ES428213A ES428213A ES428213A1 ES 428213 A1 ES428213 A1 ES 428213A1 ES 428213 A ES428213 A ES 428213A ES 428213 A ES428213 A ES 428213A ES 428213 A1 ES428213 A1 ES 428213A1
Authority
ES
Spain
Prior art keywords
penicillin
preparation
dialkylaminoalkyl esters
dialkylaminoalkyl
esters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES428213A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dr Andreu SA
Original Assignee
Dr Andreu SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Andreu SA filed Critical Dr Andreu SA
Priority to ES428213A priority Critical patent/ES428213A1/en
Priority to AR259481A priority patent/AR214390A1/en
Priority to GB2833075A priority patent/GB1470154A/en
Priority to CH899975A priority patent/CH595386A5/xx
Priority to CA231,318A priority patent/CA1055928A/en
Priority to FR7521914A priority patent/FR2277582A1/en
Priority to DE2531144A priority patent/DE2531144C3/en
Publication of ES428213A1 publication Critical patent/ES428213A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Procedure for obtaining dialkylaminoalkyl esters of penicillin, of general formula: ** (See formula) ** where: R, can be a hydrogen, a lower alkyl radical, hydroxy, methoxy, ethoxy, etc. R'is an alkyl group n, can be 0 or 1 r, is between 1 and 10 characterized in that, in an anhydrous medium, an alkaline salt of a penicillin is reacted with an alkyl ester of chloroform acid, then decomposing the mixed anhydride generated with an N, N-disubstituted aninoalcohol. (Machine-translation by Google Translate, not legally binding)
ES428213A 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof Expired ES428213A1 (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
ES428213A ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
AR259481A AR214390A1 (en) 1974-07-12 1975-07-04 PROCEDURE FOR OBTAINING DALKYLAMINEALKYL ESTERS OF 7- (PHENILLACETIL) OR 7-BENZOYL PENICILLIN
GB2833075A GB1470154A (en) 1974-07-12 1975-07-04 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
CH899975A CH595386A5 (en) 1974-07-12 1975-07-10
CA231,318A CA1055928A (en) 1974-07-12 1975-07-11 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
FR7521914A FR2277582A1 (en) 1974-07-12 1975-07-11 PENICILLIN DIALKYLAMINOALKYL ESTERS, THEIR PREPARATION PROCESS AND THEIR APPLICATION
DE2531144A DE2531144C3 (en) 1974-07-12 1975-07-11 2,6-Dimethoxyphenylpenicillindiethylaminoäthylester and process for its preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES428213A ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Publications (1)

Publication Number Publication Date
ES428213A1 true ES428213A1 (en) 1976-07-16

Family

ID=8467134

Family Applications (1)

Application Number Title Priority Date Filing Date
ES428213A Expired ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Country Status (7)

Country Link
AR (1) AR214390A1 (en)
CA (1) CA1055928A (en)
CH (1) CH595386A5 (en)
DE (1) DE2531144C3 (en)
ES (1) ES428213A1 (en)
FR (1) FR2277582A1 (en)
GB (1) GB1470154A (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4150157A (en) * 1976-06-11 1979-04-17 Beecham Group Limited Penicillin compositions
GB1569421A (en) * 1976-06-11 1980-06-18 Beecham Group Ltd Penicillin compositions
US4215120A (en) * 1977-07-14 1980-07-29 Beecham Group Limited Penicillin esters and their preparation
JP5324463B2 (en) * 2006-12-10 2013-10-23 チョンシー ユー Transdermal delivery system for β-lactam antibiotics
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
IN2014KN02583A (en) 2012-05-16 2015-05-08 Techfields Pharma Co Ltd

Also Published As

Publication number Publication date
FR2277582A1 (en) 1976-02-06
AR214390A1 (en) 1979-06-15
DE2531144A1 (en) 1976-01-29
DE2531144B2 (en) 1978-02-23
CA1055928A (en) 1979-06-05
FR2277582B1 (en) 1978-12-01
CH595386A5 (en) 1978-02-15
DE2531144C3 (en) 1978-09-28
GB1470154A (en) 1977-04-14

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19960205