ES428213A1 - Dialkylaminoalkyl esters of penicillin and process for the preparation thereof - Google Patents

Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Info

Publication number
ES428213A1
ES428213A1 ES428213A ES428213A ES428213A1 ES 428213 A1 ES428213 A1 ES 428213A1 ES 428213 A ES428213 A ES 428213A ES 428213 A ES428213 A ES 428213A ES 428213 A1 ES428213 A1 ES 428213A1
Authority
ES
Spain
Prior art keywords
penicillin
preparation
dialkylaminoalkyl esters
dialkylaminoalkyl
esters
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES428213A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dr Andreu SA
Original Assignee
Dr Andreu SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dr Andreu SA filed Critical Dr Andreu SA
Priority to ES428213A priority Critical patent/ES428213A1/en
Priority to GB2833075A priority patent/GB1470154A/en
Priority to AR259481A priority patent/AR214390A1/en
Priority to CH899975A priority patent/CH595386A5/xx
Priority to FR7521914A priority patent/FR2277582A1/en
Priority to DE2531144A priority patent/DE2531144C3/en
Priority to CA231,318A priority patent/CA1055928A/en
Publication of ES428213A1 publication Critical patent/ES428213A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring

Abstract

Procedure for obtaining dialkylaminoalkyl esters of penicillin, of general formula: ** (See formula) ** where: R, can be a hydrogen, a lower alkyl radical, hydroxy, methoxy, ethoxy, etc. R'is an alkyl group n, can be 0 or 1 r, is between 1 and 10 characterized in that, in an anhydrous medium, an alkaline salt of a penicillin is reacted with an alkyl ester of chloroform acid, then decomposing the mixed anhydride generated with an N, N-disubstituted aninoalcohol. (Machine-translation by Google Translate, not legally binding)
ES428213A 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof Expired ES428213A1 (en)

Priority Applications (7)

Application Number Priority Date Filing Date Title
ES428213A ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
GB2833075A GB1470154A (en) 1974-07-12 1975-07-04 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
AR259481A AR214390A1 (en) 1974-07-12 1975-07-04 PROCEDURE FOR OBTAINING DALKYLAMINEALKYL ESTERS OF 7- (PHENILLACETIL) OR 7-BENZOYL PENICILLIN
CH899975A CH595386A5 (en) 1974-07-12 1975-07-10
FR7521914A FR2277582A1 (en) 1974-07-12 1975-07-11 PENICILLIN DIALKYLAMINOALKYL ESTERS, THEIR PREPARATION PROCESS AND THEIR APPLICATION
DE2531144A DE2531144C3 (en) 1974-07-12 1975-07-11 2,6-Dimethoxyphenylpenicillindiethylaminoäthylester and process for its preparation
CA231,318A CA1055928A (en) 1974-07-12 1975-07-11 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES428213A ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Publications (1)

Publication Number Publication Date
ES428213A1 true ES428213A1 (en) 1976-07-16

Family

ID=8467134

Family Applications (1)

Application Number Title Priority Date Filing Date
ES428213A Expired ES428213A1 (en) 1974-07-12 1974-07-12 Dialkylaminoalkyl esters of penicillin and process for the preparation thereof

Country Status (7)

Country Link
AR (1) AR214390A1 (en)
CA (1) CA1055928A (en)
CH (1) CH595386A5 (en)
DE (1) DE2531144C3 (en)
ES (1) ES428213A1 (en)
FR (1) FR2277582A1 (en)
GB (1) GB1470154A (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1569421A (en) * 1976-06-11 1980-06-18 Beecham Group Ltd Penicillin compositions
US4150157A (en) * 1976-06-11 1979-04-17 Beecham Group Limited Penicillin compositions
US4215120A (en) * 1977-07-14 1980-07-29 Beecham Group Limited Penicillin esters and their preparation
WO2008072032A1 (en) * 2006-12-10 2008-06-19 Chongxi Yu Transdermal delivery systems of beta-lactam antibiotics
US9969751B2 (en) 2009-06-10 2018-05-15 Techfields Pharma Co., Ltd. High penetration prodrug compositions of antimicrobials and antimicrobial-related compounds
EP2849738B1 (en) 2012-05-16 2023-12-06 Techfields Pharma Co., Ltd. High penetration prodrug compositions and pharmaceutical composition thereof for treatment of pulmonary conditions

Also Published As

Publication number Publication date
DE2531144A1 (en) 1976-01-29
AR214390A1 (en) 1979-06-15
DE2531144B2 (en) 1978-02-23
FR2277582B1 (en) 1978-12-01
DE2531144C3 (en) 1978-09-28
FR2277582A1 (en) 1976-02-06
GB1470154A (en) 1977-04-14
CH595386A5 (en) 1978-02-15
CA1055928A (en) 1979-06-05

Similar Documents

Publication Publication Date Title
GB1511366A (en) Aliphatic carboxylic acid esters of vitamin e and process for preparation thereof
FR2405245A1 (en) BENZYL-PYRROLYL-METHYL CARBOXYLATE INSECTICIDES AND ACARICIDES
ES450536A1 (en) Chroman-4-ones and process for preparing same
ES482415A1 (en) Process for making 4-aminohex-5-enoic acid
ES428213A1 (en) Dialkylaminoalkyl esters of penicillin and process for the preparation thereof
ES454086A1 (en) Procedure for the preparation of N- (r-tetrahydrofurfuril) -noroximorphone and N- (s-tetrahydrofurfuril) -norosimorphone new. (Machine-translation by Google Translate, not legally binding)
ES449130A1 (en) Method for the preparation of 2-hydroxybenzanthrone compounds
ES478126A1 (en) Compounds of the pregnane series with an oxygen function in the 19-position, processes for their manufacture and pharmaceutical preparations containing these compounds
ES459079A1 (en) Production of chrysanthemic acid esters and homologues thereof
ES444957A1 (en) Glycyrrhetinic acid derivatives
ES434026A1 (en) Hydroxy and ether containing phenothiazine derivatives
ES417164A1 (en) Cardenolide-3-(2'-desoxy-glycosides)+0 and process for their manufacture
ES436218A1 (en) Phenoxyalkanol derivatives and a process for their preparation
ES443115A1 (en) Novel ester of 19-nor-testosterone
ES456325A1 (en) Quinoline carboxalic acid esters
JPS51127068A (en) A process for preparing 8-azaprostanoic acid derivatives.
JPS5427546A (en) Liquid crystal compound
JPS5210218A (en) Preparation of beta-sulfenylacrylamides
JPS5217447A (en) Process for preparation of trans-4- aminomethylcyclohexane-carboxylic acid ester
ES433453A1 (en) Arylpiperazine derivatives of adenine
JPS52263A (en) Process for preparation of 1-alkanesulfonyloxy alkyl-2-alkyl-3-dipheny lmethylenepyrrolidine and its salts
JPS51127080A (en) A process for preparing quisqualic acid.
ES458893A1 (en) Pharmaceutical spasmolytic composition
JPS5210219A (en) Preparation of beta-sulfonylacrylic beta-sulfonylacrylic their esters and acids their esters and amides
GB1519690A (en) Phenoxyalkane carboxylic acid derivatives

Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19960205