ES423827A1 - Procedimiento para preparar derivados de acidos penicilani-co y cefalosporanico. - Google Patents
Procedimiento para preparar derivados de acidos penicilani-co y cefalosporanico.Info
- Publication number
- ES423827A1 ES423827A1 ES423827A ES423827A ES423827A1 ES 423827 A1 ES423827 A1 ES 423827A1 ES 423827 A ES423827 A ES 423827A ES 423827 A ES423827 A ES 423827A ES 423827 A1 ES423827 A1 ES 423827A1
- Authority
- ES
- Spain
- Prior art keywords
- group
- symbol
- carbonylamino
- salt
- residue
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 239000002253 acid Substances 0.000 title abstract 3
- 150000007513 acids Chemical class 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 150000002148 esters Chemical group 0.000 abstract 5
- 125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 4
- 150000003839 salts Chemical class 0.000 abstract 4
- WKBOTKDWSSQWDR-UHFFFAOYSA-N Bromine atom Chemical group [Br] WKBOTKDWSSQWDR-UHFFFAOYSA-N 0.000 abstract 3
- -1 carbamoyloxy group Chemical group 0.000 abstract 3
- 125000006297 carbonyl amino group Chemical group [H]N([*:2])C([*:1])=O 0.000 abstract 3
- 229910052801 chlorine Inorganic materials 0.000 abstract 3
- 239000000460 chlorine Substances 0.000 abstract 3
- KZBUYRJDOAKODT-UHFFFAOYSA-N Chlorine Chemical compound ClCl KZBUYRJDOAKODT-UHFFFAOYSA-N 0.000 abstract 2
- 150000001408 amides Chemical class 0.000 abstract 2
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- 239000001257 hydrogen Substances 0.000 abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 2
- 125000004356 hydroxy functional group Chemical group O* 0.000 abstract 2
- 230000000269 nucleophilic effect Effects 0.000 abstract 2
- NGHVIOIJCVXTGV-ALEPSDHESA-N 6-aminopenicillanic acid Chemical compound [O-]C(=O)[C@H]1C(C)(C)S[C@@H]2[C@H]([NH3+])C(=O)N21 NGHVIOIJCVXTGV-ALEPSDHESA-N 0.000 abstract 1
- HSHGZXNAXBPPDL-HZGVNTEJSA-N 7beta-aminocephalosporanic acid Chemical compound S1CC(COC(=O)C)=C(C([O-])=O)N2C(=O)[C@@H]([NH3+])[C@@H]12 HSHGZXNAXBPPDL-HZGVNTEJSA-N 0.000 abstract 1
- ZAMOUSCENKQFHK-UHFFFAOYSA-N Chlorine atom Chemical group [Cl] ZAMOUSCENKQFHK-UHFFFAOYSA-N 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 238000010521 absorption reaction Methods 0.000 abstract 1
- 125000003668 acetyloxy group Chemical group [H]C([H])([H])C(=O)O[*] 0.000 abstract 1
- 238000005917 acylation reaction Methods 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 239000003513 alkali Substances 0.000 abstract 1
- 229910052784 alkaline earth metal Inorganic materials 0.000 abstract 1
- 150000001342 alkaline earth metals Chemical class 0.000 abstract 1
- 125000004466 alkoxycarbonylamino group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 150000001412 amines Chemical class 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- 125000004429 atom Chemical group 0.000 abstract 1
- 125000000852 azido group Chemical group *N=[N+]=[N-] 0.000 abstract 1
- GDTBXPJZTBHREO-UHFFFAOYSA-N bromine Chemical group BrBr GDTBXPJZTBHREO-UHFFFAOYSA-N 0.000 abstract 1
- 229910052794 bromium Chemical group 0.000 abstract 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 abstract 1
- 150000001768 cations Chemical class 0.000 abstract 1
- YGBFLZPYDUKSPT-MRVPVSSYSA-N cephalosporanic acid Chemical compound S1CC(COC(=O)C)=C(C(O)=O)N2C(=O)C[C@H]21 YGBFLZPYDUKSPT-MRVPVSSYSA-N 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002883 imidazolyl group Chemical group 0.000 abstract 1
- 125000000842 isoxazolyl group Chemical group 0.000 abstract 1
- 229910052751 metal Inorganic materials 0.000 abstract 1
- 239000002184 metal Substances 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 239000003960 organic solvent Substances 0.000 abstract 1
- 125000001715 oxadiazolyl group Chemical group 0.000 abstract 1
- 125000002071 phenylalkoxy group Chemical group 0.000 abstract 1
- 230000001681 protective effect Effects 0.000 abstract 1
- 125000000542 sulfonic acid group Chemical group 0.000 abstract 1
- 125000006633 tert-butoxycarbonylamino group Chemical group 0.000 abstract 1
- 125000003831 tetrazolyl group Chemical group 0.000 abstract 1
- 230000001131 transforming effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Cephalosporin Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1018973A GB1464377A (en) | 1973-03-02 | 1973-03-02 | Penicillanic and cephalosporanic acid derivatives |
| GB183674 | 1974-01-15 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES423827A1 true ES423827A1 (es) | 1976-10-16 |
Family
ID=26237021
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES423827A Expired ES423827A1 (es) | 1973-03-02 | 1974-03-02 | Procedimiento para preparar derivados de acidos penicilani-co y cefalosporanico. |
| ES423828A Expired ES423828A1 (es) | 1973-03-02 | 1974-03-02 | Procedimiento para preparar derivados de acidos aminopenici-lanico 6-sustituidos y aminocefalosparanico 7-sustituidos. |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES423828A Expired ES423828A1 (es) | 1973-03-02 | 1974-03-02 | Procedimiento para preparar derivados de acidos aminopenici-lanico 6-sustituidos y aminocefalosparanico 7-sustituidos. |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JPS5029591A (enrdf_load_stackoverflow) |
| AU (1) | AU6620274A (enrdf_load_stackoverflow) |
| DE (1) | DE2409949A1 (enrdf_load_stackoverflow) |
| ES (2) | ES423827A1 (enrdf_load_stackoverflow) |
| FR (1) | FR2219775A1 (enrdf_load_stackoverflow) |
| NL (1) | NL7402778A (enrdf_load_stackoverflow) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS54106495A (en) * | 1978-02-09 | 1979-08-21 | Dai Ichi Seiyaku Co Ltd | Cephem derivative |
| JPS6052713B2 (ja) * | 1978-04-11 | 1985-11-20 | 三共株式会社 | ７−メトキシセフアロスポリン化合物、その製法及びその化合物を主成分とする抗菌剤 |
| JPS6017368A (ja) * | 1983-07-09 | 1985-01-29 | Toyota Motor Corp | キツクレス式ケ−ブルの短絡検出方法及びその装置 |
| HU203243B (en) * | 1985-07-16 | 1991-06-28 | Biogal Gyogyszergyar | Process for producing cefalosporin derivative |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1364453A (en) * | 1970-11-06 | 1974-08-21 | Gist Brocades Nv | Penicillanic and cepholosporanic acid derivatives |
-
1974
- 1974-03-01 NL NL7402778A patent/NL7402778A/xx unknown
- 1974-03-01 AU AU66202/74A patent/AU6620274A/en not_active Expired
- 1974-03-01 FR FR7407098A patent/FR2219775A1/fr active Granted
- 1974-03-01 DE DE2409949A patent/DE2409949A1/de active Pending
- 1974-03-02 ES ES423827A patent/ES423827A1/es not_active Expired
- 1974-03-02 ES ES423828A patent/ES423828A1/es not_active Expired
- 1974-03-02 JP JP49024712A patent/JPS5029591A/ja active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| AU6620274A (en) | 1975-09-04 |
| NL7402778A (enrdf_load_stackoverflow) | 1974-09-04 |
| FR2219775A1 (en) | 1974-09-27 |
| JPS5029591A (enrdf_load_stackoverflow) | 1975-03-25 |
| ES423828A1 (es) | 1977-06-16 |
| FR2219775B1 (enrdf_load_stackoverflow) | 1978-07-28 |
| DE2409949A1 (de) | 1974-09-05 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| US4138397A (en) | 6-(2,3-Dihydro-5-benzofuranyl)acetamido penicillin derivatives | |
| KR840002407A (ko) | 세팔로스포린 유도체의 제조방법 | |
| ES423827A1 (es) | Procedimiento para preparar derivados de acidos penicilani-co y cefalosporanico. | |
| CA3041437A1 (en) | A process for preparing an intermediate for avibactam | |
| SU578876A3 (ru) | Способ получени производных пиразин-4-оксида или их солей | |
| GB1073828A (en) | O-desacetyl-o-carbamoyl-7-acylamino-cephalosporanic acids | |
| ES381577A1 (es) | Procedimiento para la preparacion de nuevos derivados de acido ariloxi y ariltio-acetico. | |
| GB1382494A (en) | Acylaminocephalosporanic acids and process for their manufacture | |
| US4229575A (en) | 7-(2,3-Dihydrobenzo-5-furanyl)-acetamido cephalosporin derivatives | |
| US3067237A (en) | Lower-alkyl mono-or bis-(alkanesulfonamido) benzoate esters | |
| US4024129A (en) | Process for the preparation of heterocyclic compounds | |
| US3479401A (en) | Guanidinoaryl and guanidinomethylaryl compounds | |
| SE7600585L (sv) | Forfarande for framstellning av 7-aminocefalosporansyraderivat | |
| US2741614A (en) | N-isobutylnormorpfflne compounds | |
| US3296250A (en) | 4-thiazolylmethylpenicillins | |
| US3666770A (en) | Process for preparing d-5,5-dimethyl-{66 {11 -thiazoline-4-carboxylic derivatives | |
| GB1473981A (en) | Hydrazino-cephalosporanic acid derivatives | |
| US3946002A (en) | Process for preparing cephalosporins | |
| US2915522A (en) | N-tbeta-methyl-mercapto-ethyl | |
| US3294783A (en) | Certain 3-and 5-substituted-4-isothiazolylmethylpenicillins | |
| US3531470A (en) | Alpha-amino-2,4,6-cycloheptatrienyl-methylpenicillins | |
| GB748724A (en) | Desdimethylamino-oxytetracycline | |
| US3280111A (en) | Penicillin derivatives | |
| GB882090A (en) | New sulphamoyl benzamides and processes for the production thereof | |
| GB727481A (en) | Improvements in or relating to the preparation of esters and amides of penicillin g and penicillin x |