ES395260A1 - Imidazo-4,5-b-pyridine derivatives - Google Patents

Imidazo-4,5-b-pyridine derivatives

Info

Publication number
ES395260A1
ES395260A1 ES395260A ES395260A ES395260A1 ES 395260 A1 ES395260 A1 ES 395260A1 ES 395260 A ES395260 A ES 395260A ES 395260 A ES395260 A ES 395260A ES 395260 A1 ES395260 A1 ES 395260A1
Authority
ES
Spain
Prior art keywords
imidazo
general formula
carbon atoms
formula
alkyl radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES395260A
Other languages
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Rhone Poulenc SA
Original Assignee
Rhone Poulenc SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7034133A external-priority patent/FR2105060A1/en
Priority claimed from FR7130825A external-priority patent/FR2150236A2/en
Application filed by Rhone Poulenc SA filed Critical Rhone Poulenc SA
Publication of ES395260A1 publication Critical patent/ES395260A1/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Procedure for the preparation of imidazo [4,5-b] pyridine of general formula: ** (See formula) ** wherein R represents a hydrogen atom or an alkyl radical containing from 1 to 4 carbon atoms and R1 represents an alkyl radical containing from 1 to 4 carbon atoms, characterized in that a diamino pyridine of general formula is reacted : ** (See formula) ** in which R is defined as above, on an isothiourea of general formula: ** (See formula) ** wherein R1 is defined as above, and then the product obtained is optionally transformed into an addition salt with an acid or a quaternary ammonium salt. (Machine-translation by Google Translate, not legally binding)
ES395260A 1970-09-21 1971-09-21 Imidazo-4,5-b-pyridine derivatives Expired ES395260A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7034133A FR2105060A1 (en) 1970-09-21 1970-09-21 Anthelmintic imidazo (4,5-b) pyridine derivs - with low mammalian toxicity,for oral human and veterinary use
FR7130825A FR2150236A2 (en) 1971-08-25 1971-08-25 Anthelmintic imidazo (4,5-b) pyridine derivs - with low mammalian toxicity,for oral human and veterinary use

Publications (1)

Publication Number Publication Date
ES395260A1 true ES395260A1 (en) 1973-12-01

Family

ID=26215952

Family Applications (2)

Application Number Title Priority Date Filing Date
ES395260A Expired ES395260A1 (en) 1970-09-21 1971-09-21 Imidazo-4,5-b-pyridine derivatives
ES403910A Expired ES403910A1 (en) 1970-09-21 1972-06-15 Imidazo-4,5-b-pyridine derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
ES403910A Expired ES403910A1 (en) 1970-09-21 1972-06-15 Imidazo-4,5-b-pyridine derivatives

Country Status (13)

Country Link
AU (1) AU453067B2 (en)
BE (1) BE772835A (en)
CA (1) CA940131A (en)
CH (1) CH532600A (en)
DE (1) DE2147103C3 (en)
DK (1) DK131345B (en)
ES (2) ES395260A1 (en)
GB (1) GB1318859A (en)
HU (1) HU163150B (en)
IL (1) IL37752A (en)
LU (1) LU63927A1 (en)
NL (1) NL145553B (en)
SE (1) SE368828B (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000057870A2 (en) 1999-03-31 2000-10-05 The Procter & Gamble Company Viral treatment
US6593466B1 (en) 1999-07-07 2003-07-15 Isis Pharmaceuticals, Inc. Guanidinium functionalized nucleotides and precursors thereof
US6384049B1 (en) * 2000-05-25 2002-05-07 The Procter & Gamble Company Cancer treatment

Also Published As

Publication number Publication date
AU3373571A (en) 1973-03-29
DE2147103B2 (en) 1974-11-14
LU63927A1 (en) 1972-06-27
DE2147103A1 (en) 1972-03-23
DK131345C (en) 1975-11-24
IL37752A0 (en) 1971-11-29
IL37752A (en) 1974-10-22
HU163150B (en) 1973-06-28
CH532600A (en) 1973-01-15
AU453067B2 (en) 1974-09-19
DK131345B (en) 1975-06-30
GB1318859A (en) 1973-05-31
SE368828B (en) 1974-07-22
BE772835A (en) 1972-03-20
DE2147103C3 (en) 1975-07-17
NL7112971A (en) 1972-03-23
ES403910A1 (en) 1975-05-01
NL145553B (en) 1975-04-15
CA940131A (en) 1974-01-15

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