ES382550A1 - Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino-tieno (3,2-d) pirimidinas. - Google Patents

Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino-tieno (3,2-d) pirimidinas.

Info

Publication number
ES382550A1
ES382550A1 ES382550A ES382550A ES382550A1 ES 382550 A1 ES382550 A1 ES 382550A1 ES 382550 A ES382550 A ES 382550A ES 382550 A ES382550 A ES 382550A ES 382550 A1 ES382550 A1 ES 382550A1
Authority
ES
Spain
Prior art keywords
carboxylic acid
imide
carbon atoms
amino
atom
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES382550A
Other languages
English (en)
Spanish (es)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Original Assignee
Dr Karl Thomae GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE19691940572 external-priority patent/DE1940572A1/de
Priority claimed from DE19702032686 external-priority patent/DE2032686A1/de
Priority claimed from DE19702032687 external-priority patent/DE2032687A1/de
Application filed by Dr Karl Thomae GmbH filed Critical Dr Karl Thomae GmbH
Publication of ES382550A1 publication Critical patent/ES382550A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D495/00Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04Ortho-condensed systems
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Slide Fasteners (AREA)
ES382550A 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino-tieno (3,2-d) pirimidinas. Expired ES382550A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19691940572 DE1940572A1 (de) 1969-08-08 1969-08-08 Neue 2-Aminoalkylamino-thieno[3,2-d]pyrimidine und Verfahren zu ihrer Herstellung
DE19702032686 DE2032686A1 (de) 1970-07-02 1970-07-02 Verfahren zur Herstellung von neuen 2 Aminoalkylamino thieno eckige Klammer auf 3,2 d eckige Klammer zu Pynmidinen
DE19702032687 DE2032687A1 (en) 1970-07-02 1970-07-02 Cardiovascular 2-aminoalkylamino-thienopyrimidines - and 4-morpholino derivatives from 4-diethanolamino-compounds by intramolecular cyclisa

Publications (1)

Publication Number Publication Date
ES382550A1 true ES382550A1 (es) 1973-04-16

Family

ID=27182086

Family Applications (5)

Application Number Title Priority Date Filing Date
ES382550A Expired ES382550A1 (es) 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino-tieno (3,2-d) pirimidinas.
ES382552A Expired ES382552A1 (es) 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino tieno (3,2-d) pirimidinas.
ES382548A Expired ES382548A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.
ES382551A Expired ES382551A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)pirimidinas.
ES382549A Expired ES382549A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.

Family Applications After (4)

Application Number Title Priority Date Filing Date
ES382552A Expired ES382552A1 (es) 1969-08-08 1970-08-07 Procedimiento para la preparacion de nuevas 2-aminoalcohi- lamino tieno (3,2-d) pirimidinas.
ES382548A Expired ES382548A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.
ES382551A Expired ES382551A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)pirimidinas.
ES382549A Expired ES382549A1 (es) 1969-08-08 1970-08-07 Un procedimiento para la preparacion de nuevas 2-amino-al- cohil-amino-tieno (3,2-d)piridinas.

Country Status (14)

Country Link
US (1) US3838121A (enrdf_load_html_response)
JP (1) JPS519759B1 (enrdf_load_html_response)
BE (1) BE754606A (enrdf_load_html_response)
BG (1) BG17591A3 (enrdf_load_html_response)
CH (5) CH547301A (enrdf_load_html_response)
ES (5) ES382550A1 (enrdf_load_html_response)
FI (1) FI51939C (enrdf_load_html_response)
FR (1) FR2068478B1 (enrdf_load_html_response)
IE (1) IE34687B1 (enrdf_load_html_response)
IL (1) IL35078A (enrdf_load_html_response)
NL (1) NL7011592A (enrdf_load_html_response)
NO (1) NO130538C (enrdf_load_html_response)
PH (1) PH9574A (enrdf_load_html_response)
SE (1) SE386449B (enrdf_load_html_response)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6187777B1 (en) 1998-02-06 2001-02-13 Amgen Inc. Compounds and methods which modulate feeding behavior and related diseases
EP1608652A1 (en) * 2003-03-31 2005-12-28 Vernalis (Cambridge) Limited Pyrazolopyrimidine compounds and their use in medicine
GB0423653D0 (en) 2004-10-25 2004-11-24 Piramed Ltd Pharmaceutical compounds
CA2605161A1 (en) * 2005-04-21 2006-10-26 Boehringer Ingelheim International Gmbh Dihydrothienopyrimidines for the treatment of inflammatory diseases
EP1847543A1 (de) 2006-04-19 2007-10-24 Boehringer Ingelheim Pharma GmbH & Co. KG Dihydrothienopyrimidine zur Behandlung von entzündlichen Erkrankungen
UA95799C2 (en) 2006-04-26 2011-09-12 Ф. Хоффманн-Ля Рош Аг Pharmaceutical compounds
WO2007127183A1 (en) * 2006-04-26 2007-11-08 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and pharmaceutical compositions containing them
AU2007243457B2 (en) 2006-04-26 2012-02-23 F. Hoffmann-La Roche Ag Pharmaceutical compounds
TWI499420B (zh) 2006-12-07 2015-09-11 Hoffmann La Roche 肌醇磷脂3-激酶抑制劑化合物及使用方法
CA2671845C (en) * 2006-12-07 2015-03-24 Genentech, Inc. Phosphoinositide 3-kinase inhibitor compounds and methods of use
NZ585346A (en) * 2007-10-19 2011-09-30 Boehringer Ingelheim Int Substituted piperidino-dihydrothienopyrimidines
KR20100075930A (ko) 2007-10-19 2010-07-05 베링거 인겔하임 인터내셔날 게엠베하 헤테로사이클-치환된 피페라지노-디하이드로티에노피리미딘
JP5563466B2 (ja) 2007-10-19 2014-07-30 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング 新規ピペラジノ−ジヒドロチエノピリミジン誘導体
GB0721095D0 (en) * 2007-10-26 2007-12-05 Piramed Ltd Pharmaceutical compounds
EP2451811A1 (en) * 2009-05-27 2012-05-16 F. Hoffmann-La Roche AG Bicyclic indole-pyrimidine pi3k inhibitor compounds selective for p110 delta, and methods of use
JP5781066B2 (ja) 2009-05-27 2015-09-16 ジェネンテック, インコーポレイテッド p110δに対して選択的な二環式ピリミジンPI3K阻害剤化合物及び使用方法
AU2010314287A1 (en) * 2009-10-12 2012-05-03 F. Hoffmann-La Roche Ag Combinations of a PI3K inhibitor and a MEK inhibitor
US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma

Also Published As

Publication number Publication date
NO130538C (enrdf_load_html_response) 1975-01-08
ES382549A1 (es) 1973-04-01
NL7011592A (enrdf_load_html_response) 1971-02-10
CH547299A (de) 1974-03-29
IL35078A (en) 1974-09-10
FR2068478A1 (enrdf_load_html_response) 1971-08-27
CH547301A (de) 1974-03-29
CH546251A (de) 1974-02-28
US3838121A (en) 1974-09-24
CH547300A (de) 1974-03-29
IE34687B1 (en) 1975-07-23
JPS519759B1 (enrdf_load_html_response) 1976-03-30
PH9574A (en) 1976-01-16
FI51939C (fi) 1977-05-10
IL35078A0 (en) 1970-10-30
BE754606A (fr) 1971-02-08
FI51939B (enrdf_load_html_response) 1977-01-31
ES382552A1 (es) 1973-04-16
FR2068478B1 (enrdf_load_html_response) 1974-08-30
ES382551A1 (es) 1973-04-01
ES382548A1 (es) 1973-04-01
NO130538B (enrdf_load_html_response) 1974-09-23
CH547304A (de) 1974-03-29
BG17591A3 (bg) 1973-11-10
IE34687L (en) 1971-02-08
SE386449B (sv) 1976-08-09

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