ES336020A1 - Procedimiento para la preparacion de nuevos derivados de imidazol. - Google Patents

Procedimiento para la preparacion de nuevos derivados de imidazol.

Info

Publication number
ES336020A1
ES336020A1 ES0336020A ES336020A ES336020A1 ES 336020 A1 ES336020 A1 ES 336020A1 ES 0336020 A ES0336020 A ES 0336020A ES 336020 A ES336020 A ES 336020A ES 336020 A1 ES336020 A1 ES 336020A1
Authority
ES
Spain
Prior art keywords
group
translation
lower alkyl
preparation
alkyl group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES0336020A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
JR Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by JR Geigy AG filed Critical JR Geigy AG
Publication of ES336020A1 publication Critical patent/ES336020A1/es
Expired legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/88Nitrogen atoms, e.g. allantoin

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES0336020A 1966-01-25 1967-01-24 Procedimiento para la preparacion de nuevos derivados de imidazol. Expired ES336020A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US52282966A 1966-01-25 1966-01-25

Publications (1)

Publication Number Publication Date
ES336020A1 true ES336020A1 (es) 1967-12-16

Family

ID=24082557

Family Applications (1)

Application Number Title Priority Date Filing Date
ES0336020A Expired ES336020A1 (es) 1966-01-25 1967-01-24 Procedimiento para la preparacion de nuevos derivados de imidazol.

Country Status (14)

Country Link
US (1) US3459763A (es)
AT (1) AT262997B (es)
BE (1) BE693079A (es)
CH (1) CH474522A (es)
DE (1) DE1695005A1 (es)
DK (1) DK121302B (es)
ES (1) ES336020A1 (es)
FR (2) FR1508888A (es)
GB (1) GB1131191A (es)
GR (1) GR36359B (es)
IL (1) IL27312A (es)
NL (1) NL6701100A (es)
NO (1) NO117129B (es)
SE (1) SE339475B (es)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3700685A (en) * 1970-05-15 1972-10-24 Merck & Co Inc Nitroimidazole derivatives
US3859302A (en) * 1973-02-05 1975-01-07 Monsanto Co Preparation of 2-imino-imidazole derivatives
FR2269341B1 (es) * 1974-04-30 1978-07-28 Castaigne Sa
US4195092A (en) * 1977-12-27 1980-03-25 Eli Lilly And Company 2-(Substituted amino)-N-(3-substituted phenyl)-2-imidazoline-1-carbothioamides
EP0656210A1 (en) * 1993-11-19 1995-06-07 Takeda Chemical Industries, Ltd. Imidazole derivatives as glutaminose inhibitors
JP3805360B2 (ja) * 1994-01-24 2006-08-02 アラーガン、インコーポレイテッド α▲下2A▼アドレナリン受容体作動剤としての芳香族2−アミノ−イミダゾール誘導体
US5922751A (en) * 1994-06-24 1999-07-13 Euro-Celtique, S.A. Aryl pyrazole compound for inhibiting phosphodiesterase IV and methods of using same
US6087361A (en) * 1995-05-12 2000-07-11 Allergan Sales, Inc. Aryl-imidazolines and aryl-imidazoles useful as α-2 adrenergic agonists without cardiovascular side effects
WO2001044203A1 (en) * 1999-12-17 2001-06-21 The Procter & Gamble Company N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
US6596739B2 (en) 2000-03-29 2003-07-22 The Procter & Gamble Company N-(1-phenylethyl)-5-phenyl-imidazole-2-amine compounds, their compositions and uses
DE10304374A1 (de) * 2003-02-04 2004-08-05 Aventis Pharma Deutschland Gmbh Neue substituierte 2-Aminoimidazole, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament
US20050054705A1 (en) 2003-02-04 2005-03-10 Aventis Pharma Deutschland Gmbh N-substituted (benzoimidazol-2-yl) phenylamines, process for their preparation, their use as medicament or diagnostic aid, and medicament comprising them
EP2101762B1 (en) 2006-12-13 2011-05-18 F. Hoffmann-La Roche AG Novel 2 -imidazoles as ligands for trace amine associated receptors (taar)
JP2010531837A (ja) 2007-07-02 2010-09-30 エフ.ホフマン−ラ ロシュ アーゲー 微量アミン関連レセプター(taar)に対して良好な親和性を有する2−イミダゾリン
KR101133862B1 (ko) 2007-07-27 2012-04-06 에프. 호프만-라 로슈 아게 Taar 리간드로서의 2-아제티딘메테인아민 및 2-피롤리딘메테인아민
CN101784515A (zh) 2007-08-03 2010-07-21 弗·哈夫曼-拉罗切有限公司 作为taar1配体的吡啶甲酰胺和苯甲酰胺衍生物
US9452980B2 (en) 2009-12-22 2016-09-27 Hoffmann-La Roche Inc. Substituted benzamides
SG10201913878YA (en) 2016-03-17 2020-03-30 Hoffmann La Roche 5-ethyl-4-methyl-pyrazole-3-carboxamide derivative having activity as agonist of taar

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2988478A (en) * 1958-12-22 1961-06-13 Pfizer & Co C Agricultural compositions and use

Also Published As

Publication number Publication date
GR36359B (el) 1969-02-03
FR6337M (es) 1968-09-30
CH474522A (de) 1969-06-30
NL6701100A (es) 1967-07-26
FR1508888A (fr) 1968-01-05
SE339475B (es) 1971-10-11
BE693079A (es) 1967-07-24
AT262997B (de) 1968-07-10
DE1695005A1 (de) 1971-02-25
GB1131191A (en) 1968-10-23
US3459763A (en) 1969-08-05
IL27312A (en) 1971-01-28
DK121302B (da) 1971-10-04
NO117129B (es) 1969-07-07

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