ES2989433T3 - Tapentadol para usar en el tratamiento del dolor asociado con neuralgia del trigémino - Google Patents
Tapentadol para usar en el tratamiento del dolor asociado con neuralgia del trigémino Download PDFInfo
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- ES2989433T3 ES2989433T3 ES19194585T ES19194585T ES2989433T3 ES 2989433 T3 ES2989433 T3 ES 2989433T3 ES 19194585 T ES19194585 T ES 19194585T ES 19194585 T ES19194585 T ES 19194585T ES 2989433 T3 ES2989433 T3 ES 2989433T3
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- tapentadol
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- treatment
- pain
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- QORWJWZARLRLPR-UHFFFAOYSA-H tricalcium bis(phosphate) Chemical compound [Ca+2].[Ca+2].[Ca+2].[O-]P([O-])([O-])=O.[O-]P([O-])([O-])=O QORWJWZARLRLPR-UHFFFAOYSA-H 0.000 description 1
- 230000001228 trophic effect Effects 0.000 description 1
- 150000004670 unsaturated fatty acids Chemical class 0.000 description 1
- 235000021122 unsaturated fatty acids Nutrition 0.000 description 1
- 229940088594 vitamin Drugs 0.000 description 1
- 235000013343 vitamin Nutrition 0.000 description 1
- 239000011782 vitamin Substances 0.000 description 1
- 229930003231 vitamin Natural products 0.000 description 1
- 235000019156 vitamin B Nutrition 0.000 description 1
- 239000011720 vitamin B Substances 0.000 description 1
- 229940046001 vitamin b complex Drugs 0.000 description 1
- 150000003722 vitamin derivatives Chemical class 0.000 description 1
- 238000005406 washing Methods 0.000 description 1
- 239000001993 wax Substances 0.000 description 1
- 238000005303 weighing Methods 0.000 description 1
- 239000011787 zinc oxide Substances 0.000 description 1
- 235000014692 zinc oxide Nutrition 0.000 description 1
- XOOUIPVCVHRTMJ-UHFFFAOYSA-L zinc stearate Chemical compound [Zn+2].CCCCCCCCCCCCCCCCCC([O-])=O.CCCCCCCCCCCCCCCCCC([O-])=O XOOUIPVCVHRTMJ-UHFFFAOYSA-L 0.000 description 1
- 229940057977 zinc stearate Drugs 0.000 description 1
- NWONKYPBYAMBJT-UHFFFAOYSA-L zinc sulfate Chemical compound [Zn+2].[O-]S([O-])(=O)=O NWONKYPBYAMBJT-UHFFFAOYSA-L 0.000 description 1
- 229910000368 zinc sulfate Inorganic materials 0.000 description 1
- 229960001763 zinc sulfate Drugs 0.000 description 1
- 108020001612 μ-opioid receptors Proteins 0.000 description 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Emergency Medicine (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pain & Pain Management (AREA)
- Dermatology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP11002810 | 2011-04-05 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2989433T3 true ES2989433T3 (es) | 2024-11-26 |
Family
ID=44115674
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES19194585T Active ES2989433T3 (es) | 2011-04-05 | 2012-04-03 | Tapentadol para usar en el tratamiento del dolor asociado con neuralgia del trigémino |
| ES12718065T Active ES2761334T3 (es) | 2011-04-05 | 2012-04-03 | Tapentadol para uso en el tratamiento del dolor asociado con la neuralgia del trigémino |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES12718065T Active ES2761334T3 (es) | 2011-04-05 | 2012-04-03 | Tapentadol para uso en el tratamiento del dolor asociado con la neuralgia del trigémino |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20120309840A1 (https=) |
| EP (2) | EP3607943B1 (https=) |
| JP (2) | JP6040219B2 (https=) |
| ES (2) | ES2989433T3 (https=) |
| HU (1) | HUE047342T2 (https=) |
| PL (1) | PL2694050T3 (https=) |
| PT (1) | PT2694050T (https=) |
| WO (1) | WO2012136351A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP3607943B1 (en) * | 2011-04-05 | 2024-09-11 | Grünenthal GmbH | Tapentadol for use in treating pain associated with trigeminal neuralgia |
| PT3302454T (pt) * | 2015-05-26 | 2021-04-01 | Technophage Investig E Desenvolvimento Em Biotecnologia Sa | Composições para utilização no tratamento da doença de parkinson e distúrbios associados |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE4426245A1 (de) | 1994-07-23 | 1996-02-22 | Gruenenthal Gmbh | 1-Phenyl-3-dimethylamino-propanverbindungen mit pharmakologischer Wirkung |
| PE20030527A1 (es) | 2001-10-24 | 2003-07-26 | Gruenenthal Chemie | Formulacion farmaceutica con liberacion retardada que contiene 3-(3-dimetilamino-1-etil-2-metil-propil) fenol o una sal farmaceuticamente aceptable del mismo y tabletas para administracion oral que la contienen |
| JP5276982B2 (ja) * | 2005-08-26 | 2013-08-28 | ボード オブ トラスティーズ オブ ザ レランド スタンフォード ジュニア ユニバーシティ | オキシトシンの投与による頭痛の処置のための方法 |
| DE102007012165A1 (de) | 2007-03-12 | 2008-09-18 | Grünenthal GmbH | Verwendung von 1-Phenyl-3-dimethylamino-propanverbindungen zur Therapie des Neuropathieschmerzes |
| EP1985292A1 (en) * | 2007-04-23 | 2008-10-29 | Grünenthal GmbH | Titration of tapentadol |
| WO2010100477A2 (en) * | 2009-03-03 | 2010-09-10 | Shire Llc | Amino acid and peptide carbamate prodrugs of tapentadol and uses thereof |
| EP3607943B1 (en) * | 2011-04-05 | 2024-09-11 | Grünenthal GmbH | Tapentadol for use in treating pain associated with trigeminal neuralgia |
-
2012
- 2012-04-03 EP EP19194585.6A patent/EP3607943B1/en active Active
- 2012-04-03 HU HUE12718065A patent/HUE047342T2/hu unknown
- 2012-04-03 JP JP2014503020A patent/JP6040219B2/ja not_active Expired - Fee Related
- 2012-04-03 WO PCT/EP2012/001475 patent/WO2012136351A1/en not_active Ceased
- 2012-04-03 EP EP12718065.1A patent/EP2694050B1/en active Active
- 2012-04-03 ES ES19194585T patent/ES2989433T3/es active Active
- 2012-04-03 US US13/438,410 patent/US20120309840A1/en not_active Abandoned
- 2012-04-03 PL PL12718065T patent/PL2694050T3/pl unknown
- 2012-04-03 ES ES12718065T patent/ES2761334T3/es active Active
- 2012-04-03 PT PT127180651T patent/PT2694050T/pt unknown
-
2016
- 2016-11-04 JP JP2016215836A patent/JP6356763B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| PL2694050T3 (pl) | 2020-03-31 |
| WO2012136351A8 (en) | 2013-10-17 |
| EP2694050A1 (en) | 2014-02-12 |
| EP3607943B1 (en) | 2024-09-11 |
| EP3607943A1 (en) | 2020-02-12 |
| JP6040219B2 (ja) | 2016-12-07 |
| US20120309840A1 (en) | 2012-12-06 |
| PT2694050T (pt) | 2019-11-22 |
| EP3607943C0 (en) | 2024-09-11 |
| EP2694050B1 (en) | 2019-10-02 |
| JP2014510760A (ja) | 2014-05-01 |
| ES2761334T3 (es) | 2020-05-19 |
| WO2012136351A1 (en) | 2012-10-11 |
| JP2017052778A (ja) | 2017-03-16 |
| HUE047342T2 (hu) | 2020-04-28 |
| JP6356763B2 (ja) | 2018-07-11 |
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