ES286808A1 - A procedure for the preparation of benzoxazepin derivatives (Machine-translation by Google Translate, not legally binding) - Google Patents
A procedure for the preparation of benzoxazepin derivatives (Machine-translation by Google Translate, not legally binding)Info
- Publication number
- ES286808A1 ES286808A1 ES286808A ES286808A ES286808A1 ES 286808 A1 ES286808 A1 ES 286808A1 ES 286808 A ES286808 A ES 286808A ES 286808 A ES286808 A ES 286808A ES 286808 A1 ES286808 A1 ES 286808A1
- Authority
- ES
- Spain
- Prior art keywords
- translation
- preparation
- machine
- legally binding
- google translate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
A process for the preparation of benzoxazepine derivatives, characterized in comprising the cyclization of a compound of the formula ** (See formula) ** where R1 represents hydrogen or lower alkyl, R2 represents hydrogen or halogen, R3 represents hydrogen, halogen or sulfamyl and X represents halogen, by intramolecular elimination of hydrogen halide, converting it into a compound of the formula ** (See formula) ** where R1, R2 and R3 have the same meaning as before, and, if the conversion of the latter compound into a salt is desired. (Machine-translation by Google Translate, not legally binding)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US18551262A | 1962-04-06 | 1962-04-06 |
Publications (1)
Publication Number | Publication Date |
---|---|
ES286808A1 true ES286808A1 (en) | 1963-11-16 |
Family
ID=22681287
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES0286809A Expired ES286809A1 (en) | 1962-04-06 | 1963-04-05 | Novel benzoxazepine derivatives and a process for the manufacture thereof |
ES286808A Expired ES286808A1 (en) | 1962-04-06 | 1963-04-05 | A procedure for the preparation of benzoxazepin derivatives (Machine-translation by Google Translate, not legally binding) |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES0286809A Expired ES286809A1 (en) | 1962-04-06 | 1963-04-05 | Novel benzoxazepine derivatives and a process for the manufacture thereof |
Country Status (5)
Country | Link |
---|---|
BE (1) | BE630572A (en) |
BR (1) | BR6348190D0 (en) |
CH (1) | CH428741A (en) |
ES (2) | ES286809A1 (en) |
GB (2) | GB980593A (en) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5017567A (en) * | 1983-11-25 | 1991-05-21 | Schering Corporation | Carboxyalkyl dipeptides as antiglaucoma agents |
US4906635A (en) * | 1983-11-25 | 1990-03-06 | Schering Corporation | Carboxyalkyl dipeptides as antiglaucoma agents |
US4778795A (en) * | 1983-11-25 | 1988-10-18 | Schering Corporation | Carboxyalkyl dipeptides as antiglaucoma agents |
-
1963
- 1963-03-20 CH CH350763A patent/CH428741A/en unknown
- 1963-04-03 BR BR148190/63A patent/BR6348190D0/en unknown
- 1963-04-04 GB GB13380/63A patent/GB980593A/en not_active Expired
- 1963-04-04 BE BE630572A patent/BE630572A/en unknown
- 1963-04-04 GB GB13379/63A patent/GB980592A/en not_active Expired
- 1963-04-05 ES ES0286809A patent/ES286809A1/en not_active Expired
- 1963-04-05 ES ES286808A patent/ES286808A1/en not_active Expired
Also Published As
Publication number | Publication date |
---|---|
BR6348190D0 (en) | 1973-07-03 |
GB980592A (en) | 1965-01-13 |
CH428741A (en) | 1967-01-31 |
GB980593A (en) | 1965-01-13 |
BE630572A (en) | 1963-11-04 |
ES286809A1 (en) | 1963-10-16 |
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