ES2629690T3 - Inhibidores de aminopirimidina quinasa - Google Patents
Inhibidores de aminopirimidina quinasa Download PDFInfo
- Publication number
- ES2629690T3 ES2629690T3 ES12780393.0T ES12780393T ES2629690T3 ES 2629690 T3 ES2629690 T3 ES 2629690T3 ES 12780393 T ES12780393 T ES 12780393T ES 2629690 T3 ES2629690 T3 ES 2629690T3
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- alkyl
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- aryl
- heteroatoms
- heteroaryl
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Classifications
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- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C07—ORGANIC CHEMISTRY
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Landscapes
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201161555617P | 2011-11-04 | 2011-11-04 | |
| US201161555617P | 2011-11-04 | ||
| PCT/US2012/061597 WO2013066684A1 (en) | 2011-11-04 | 2012-10-24 | Aminopyrimidine kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ES2629690T3 true ES2629690T3 (es) | 2017-08-14 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES12780393.0T Active ES2629690T3 (es) | 2011-11-04 | 2012-10-24 | Inhibidores de aminopirimidina quinasa |
Country Status (14)
| Country | Link |
|---|---|
| US (3) | US8927525B2 (https=) |
| EP (1) | EP2776432B1 (https=) |
| JP (1) | JP6215832B2 (https=) |
| KR (1) | KR101990605B1 (https=) |
| CN (1) | CN104011046B (https=) |
| AU (1) | AU2012332931B2 (https=) |
| BR (1) | BR112014010563B1 (https=) |
| CA (1) | CA2853454C (https=) |
| ES (1) | ES2629690T3 (https=) |
| IL (1) | IL232234A0 (https=) |
| MX (1) | MX347191B (https=) |
| PL (1) | PL2776432T3 (https=) |
| RU (1) | RU2674017C2 (https=) |
| WO (1) | WO2013066684A1 (https=) |
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| PL2516425T3 (pl) * | 2009-12-23 | 2016-03-31 | Jasco Pharmaceuticals Llc | Inhibitory kinaz aminopirydynowych |
| EP2699569B1 (en) * | 2011-04-22 | 2017-08-30 | Jasco Pharmaceuticals, LLC | Aminopyrimidine kinase inhibitors |
| KR101990605B1 (ko) | 2011-11-04 | 2019-06-18 | 자스코 파머수티컬스, 엘엘씨 | 아미노피리미딘 키나아제 억제제 |
| ES2649156T3 (es) | 2013-01-14 | 2018-01-10 | Incyte Holdings Corporation | Compuestos bicíclicos de carboxamida aromática útiles como inhibidores de quinasas Pim |
| PE20191245A1 (es) | 2013-01-15 | 2019-09-18 | Incyte Holdings Corp | Compuestos de tiazolcarboxamidas y piridinacarboxamida utiles como inhibidores de quinasa pim |
| EA201690458A1 (ru) | 2013-08-23 | 2016-07-29 | Инсайт Корпорейшн | Фуро- и тиенопиридинкарбоксамиды, используемые в качестве ингибиторов pim-киназы |
| US9822124B2 (en) | 2014-07-14 | 2017-11-21 | Incyte Corporation | Bicyclic heteroaromatic carboxamide compounds useful as Pim kinase inhibitors |
| US9580418B2 (en) | 2014-07-14 | 2017-02-28 | Incyte Corporation | Bicyclic aromatic carboxamide compounds useful as Pim kinase inhibitors |
| WO2016196244A1 (en) | 2015-05-29 | 2016-12-08 | Incyte Corporation | Pyridineamine compounds useful as pim kinase inhibitors |
| US10376511B2 (en) * | 2015-08-04 | 2019-08-13 | Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. | Pyrazole pyrimidine derivative and uses thereof |
| TWI734699B (zh) | 2015-09-09 | 2021-08-01 | 美商英塞特公司 | Ｐｉｍ激酶抑制劑之鹽 |
| US9920032B2 (en) | 2015-10-02 | 2018-03-20 | Incyte Corporation | Heterocyclic compounds useful as pim kinase inhibitors |
| MX394556B (es) | 2017-02-01 | 2025-03-24 | Yissum Res Dev Co Of Hebrew Univ Jerusalem Ltd | Derivados de n1-(4-(5-(ciclopropilmetil)-1-metil-1h-pirazol-4-il) piridin-2-il) ciclohexano-1,4-diamina y compuestos relacionados como inhibidores de ck1 y/o irak1 para tratar cáncer. |
| WO2019113487A1 (en) | 2017-12-08 | 2019-06-13 | Incyte Corporation | Low dose combination therapy for treatment of myeloproliferative neoplasms |
| UY38911A (es) | 2019-10-09 | 2021-05-31 | Bayer Ag | Compuestos de heteroarilo-triazol como pesticidas, formulaciones, usos y métodos de uso de los mismos |
| WO2025132870A1 (en) * | 2023-12-21 | 2025-06-26 | Glaxosmithkline Intellectual Property (No.4) Limited | Chemical compounds and uses thereof |
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| TW245716B (https=) | 1992-12-28 | 1995-04-21 | Takeda Pharm Industry Co | |
| US5955481A (en) | 1994-03-28 | 1999-09-21 | Nissan Chemical Industries, Ltd. | Pyridine type thiazolidines |
| TW420669B (en) * | 1994-03-28 | 2001-02-01 | Nissan Chemical Ind Ltd | Pyridine type thiazolidines |
| ATE238297T1 (de) | 1994-10-20 | 2003-05-15 | Nippon Chemiphar Co | Chinolinderivat |
| KR20070027584A (ko) | 2004-06-17 | 2007-03-09 | 와이어쓰 | 고나도트로핀 방출 호르몬 수용체 길항제 |
| CN101052640B (zh) | 2004-09-03 | 2011-05-11 | 默克雪兰诺有限公司 | 吡啶亚甲基唑烷酮类及其作为磷酸肌醇抑制剂的用途 |
| ZA200702435B (en) | 2004-10-12 | 2008-06-25 | Serono Lab | PI3 Kinase gamma inhibitors for the treatment of anaemia |
| EP1916249A1 (en) | 2006-10-10 | 2008-04-30 | LEK Pharmaceuticals D.D. | 3-(benzo[d][1,3]dioxol-5-ylmethyl)-4-(thio)oxo-2-(thio)oxo-azolidin-5-ylidene derivatives as antibacterial agents |
| EP2217235A4 (en) * | 2007-11-15 | 2011-01-12 | Musc Found For Res Dev | INHIBITORS OF PIM PROTEIN KINASES, COMPOSITIONS AND METHOD FOR THE TREATMENT OF CANCER |
| US8252823B2 (en) | 2008-01-28 | 2012-08-28 | New York University | Oxazole and thiazole compounds as beta-catenin modulators and uses thereof |
| RU2011121655A (ru) | 2008-10-29 | 2012-12-10 | Сертрис Фармасьютикалз, Инк. | Производные пиридина, бициклические производные пиридина и родственные аналоги в качестве модуляторов сиртуина |
| WO2010148351A1 (en) * | 2009-06-18 | 2010-12-23 | Cylene Pharmaceuticals, Inc. | Rhodanines and related heterocycles as kinase inhibitors |
| PL2516425T3 (pl) | 2009-12-23 | 2016-03-31 | Jasco Pharmaceuticals Llc | Inhibitory kinaz aminopirydynowych |
| EP2699569B1 (en) | 2011-04-22 | 2017-08-30 | Jasco Pharmaceuticals, LLC | Aminopyrimidine kinase inhibitors |
| KR101990605B1 (ko) | 2011-11-04 | 2019-06-18 | 자스코 파머수티컬스, 엘엘씨 | 아미노피리미딘 키나아제 억제제 |
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| AU2012332931B2 (en) | 2017-08-03 |
| JP6215832B2 (ja) | 2017-10-18 |
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| CA2853454C (en) | 2020-01-21 |
| US20130310342A1 (en) | 2013-11-21 |
| BR112014010563A2 (pt) | 2017-04-25 |
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| MX347191B (es) | 2017-04-19 |
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| EP2776432A1 (en) | 2014-09-17 |
| MX2014005052A (es) | 2015-03-19 |
| RU2674017C2 (ru) | 2018-12-04 |
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| US9629840B2 (en) | 2017-04-25 |
| KR20140098105A (ko) | 2014-08-07 |
| US20150202205A1 (en) | 2015-07-23 |
| WO2013066684A1 (en) | 2013-05-10 |
| PL2776432T3 (pl) | 2017-10-31 |
| US10336743B2 (en) | 2019-07-02 |
| KR101990605B1 (ko) | 2019-06-18 |
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