ES2523382T8 - Un proceso para preparar derivados de fenilo trisustituido que comprenden un grupo (1H-1,2,4-triazol-1-il) alquilo - Google Patents
Un proceso para preparar derivados de fenilo trisustituido que comprenden un grupo (1H-1,2,4-triazol-1-il) alquilo Download PDFInfo
- Publication number
- ES2523382T8 ES2523382T8 ES11700054.7T ES11700054T ES2523382T8 ES 2523382 T8 ES2523382 T8 ES 2523382T8 ES 11700054 T ES11700054 T ES 11700054T ES 2523382 T8 ES2523382 T8 ES 2523382T8
- Authority
- ES
- Spain
- Prior art keywords
- triazol
- alkyl group
- phenyl derivatives
- trisubstituted phenyl
- preparing trisubstituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10150257A EP2343278A1 (en) | 2010-01-07 | 2010-01-07 | A process for preparing trisubstituted phenyl derivatives comprising a (1H-1,2,4-triazol-1-yl)alkyl group |
EP10150257 | 2010-01-07 | ||
PCT/EP2011/000018 WO2011083079A1 (en) | 2010-01-07 | 2011-01-05 | A process for preparing trisubstituted phenyl derivatives comprising a (1h-1,2,4-triazol-1-yl)alkyl group |
Publications (2)
Publication Number | Publication Date |
---|---|
ES2523382T3 ES2523382T3 (es) | 2014-11-25 |
ES2523382T8 true ES2523382T8 (es) | 2014-12-05 |
Family
ID=41650285
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ES11700054.7T Active ES2523382T3 (es) | 2010-01-07 | 2011-01-05 | Un proceso para preparar derivados de fenilo trisustituido que comprenden un grupo (1H-1,2,4-triazol-1-il) alquilo |
Country Status (3)
Country | Link |
---|---|
EP (2) | EP2343278A1 (es) |
ES (1) | ES2523382T3 (es) |
WO (1) | WO2011083079A1 (es) |
Family Cites Families (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8714013D0 (en) | 1987-06-16 | 1987-07-22 | Ici Plc | (substituted-aralkyl)heterocyclic compounds |
WO2005105762A1 (en) | 2004-05-05 | 2005-11-10 | Natco Pharma Limited | Improved process for the preparation of high purity anastrozole |
DE102005037484A1 (de) | 2004-08-09 | 2006-02-23 | Chemagis Ltd. | Neue Verfahren zur Herstellung von im Wesentlichen reinem Anastrozol |
MX2007012394A (es) | 2005-04-06 | 2007-11-07 | Sicor Inc | Procesos para la preparacion de farmacos anticancer. |
WO2007002722A2 (en) | 2005-06-27 | 2007-01-04 | Sicor, Inc. | Synthesis of anastrozole and purification of one of its intermediate |
US20080207915A1 (en) | 2005-10-05 | 2008-08-28 | Radhakrishnan Tarur Venkatasub | Process for the Preparation of 2,2'-[5-(1H-1,2,4-Triazole-1-Ylmethyl) -1,3-Phenylene] Di (2-Methylpropionitrile) |
US20070100148A1 (en) | 2005-10-31 | 2007-05-03 | Veerender Murki | Process for preparing anastrozole |
AR061016A1 (es) * | 2006-05-19 | 2008-07-30 | Synthon Bv | Proceso para la purificacion de anastrozol |
EP2066646B1 (en) | 2006-10-17 | 2012-06-13 | Cipla Limited | Process for the preparation of pure anastrozole |
-
2010
- 2010-01-07 EP EP10150257A patent/EP2343278A1/en not_active Withdrawn
-
2011
- 2011-01-05 EP EP11700054.7A patent/EP2456758B1/en not_active Not-in-force
- 2011-01-05 ES ES11700054.7T patent/ES2523382T3/es active Active
- 2011-01-05 WO PCT/EP2011/000018 patent/WO2011083079A1/en active Application Filing
Also Published As
Publication number | Publication date |
---|---|
EP2456758B1 (en) | 2014-08-06 |
WO2011083079A1 (en) | 2011-07-14 |
EP2456758A1 (en) | 2012-05-30 |
EP2343278A1 (en) | 2011-07-13 |
ES2523382T3 (es) | 2014-11-25 |
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