ES2171997T3 - Procedimiento de conversion de heteroaromaticos hidroxi en arilaminas. - Google Patents

Procedimiento de conversion de heteroaromaticos hidroxi en arilaminas.

Info

Publication number
ES2171997T3
ES2171997T3 ES97941552T ES97941552T ES2171997T3 ES 2171997 T3 ES2171997 T3 ES 2171997T3 ES 97941552 T ES97941552 T ES 97941552T ES 97941552 T ES97941552 T ES 97941552T ES 2171997 T3 ES2171997 T3 ES 2171997T3
Authority
ES
Spain
Prior art keywords
procedure
arilaminas
hetroaromatic
hidroxi
conversion
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES97941552T
Other languages
English (en)
Inventor
Norton P Peet
John J Weidner
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Aventis Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharmaceuticals Inc filed Critical Aventis Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2171997T3 publication Critical patent/ES2171997T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/40—Nitrogen atoms attached in position 8
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/38—Nitrogen atoms
    • C07D215/42—Nitrogen atoms attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D219/00—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems
    • C07D219/04—Heterocyclic compounds containing acridine or hydrogenated acridine ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the ring system
    • C07D219/08—Nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE DESCRIBE UN PROCEDIMIENTO PARA CONVERTIR UN COMPUESTO HIDROXI - HETEROAROMATICO EN UNA ARILAMINA, QUE COMPRENDE LOS PASOS DE: 1) TRATAR UNA SAL DE UN COMPUESTO HIDROXIHETEROAROMATICO CON UN AGENTE ALQUILANTE, Y 2) TRATAR LA MEZCLA DE LA REACCION CON UN SISTEMA DISOLVENTE DE SMILES Y ELEVAR LA TEMPERATURA DE LA MEZCLA DE REACCION; Y UN COMPUESTO REALIZADO DE ACUERDO CON EL CITADO PROCEDIMIENTO.
ES97941552T 1996-11-27 1997-09-12 Procedimiento de conversion de heteroaromaticos hidroxi en arilaminas. Expired - Lifetime ES2171997T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US75366396A 1996-11-27 1996-11-27

Publications (1)

Publication Number Publication Date
ES2171997T3 true ES2171997T3 (es) 2002-09-16

Family

ID=25031624

Family Applications (1)

Application Number Title Priority Date Filing Date
ES97941552T Expired - Lifetime ES2171997T3 (es) 1996-11-27 1997-09-12 Procedimiento de conversion de heteroaromaticos hidroxi en arilaminas.

Country Status (18)

Country Link
EP (1) EP0944600B1 (es)
JP (1) JP4213769B2 (es)
KR (1) KR100503845B1 (es)
CN (1) CN1122024C (es)
AT (1) ATE212620T1 (es)
AU (1) AU732411B2 (es)
BR (1) BR9713553A (es)
CA (1) CA2269547C (es)
DE (1) DE69710217T2 (es)
DK (1) DK0944600T3 (es)
ES (1) ES2171997T3 (es)
HU (1) HUP0000144A3 (es)
IL (1) IL130081A (es)
NO (1) NO311296B1 (es)
NZ (1) NZ335209A (es)
PT (1) PT944600E (es)
SI (1) SI0944600T1 (es)
WO (1) WO1998023589A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103130652B (zh) * 2012-05-09 2014-12-10 浙江大学 从酚类化合物出发制备芳香伯胺类化合物的方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2166981T3 (es) * 1996-03-21 2002-05-01 Aventis Pharma Inc Procedimiento de alquilacion y de transposicion de smiles de aromaticos hidroxilados.

Also Published As

Publication number Publication date
IL130081A (en) 2004-07-25
PT944600E (pt) 2002-06-28
EP0944600B1 (en) 2002-01-30
NO992534D0 (no) 1999-05-26
KR20000057252A (ko) 2000-09-15
BR9713553A (pt) 2000-01-25
ATE212620T1 (de) 2002-02-15
DE69710217T2 (de) 2002-08-08
AU4343797A (en) 1998-06-22
DE69710217D1 (de) 2002-03-14
SI0944600T1 (en) 2002-06-30
JP2001508410A (ja) 2001-06-26
JP4213769B2 (ja) 2009-01-21
CN1122024C (zh) 2003-09-24
IL130081A0 (en) 2000-02-29
DK0944600T3 (da) 2002-04-02
HUP0000144A3 (en) 2002-01-28
CA2269547A1 (en) 1998-06-04
AU732411B2 (en) 2001-04-26
NO311296B1 (no) 2001-11-12
NO992534L (no) 1999-05-26
CA2269547C (en) 2003-12-16
HUP0000144A2 (hu) 2000-06-28
NZ335209A (en) 2000-11-24
CN1238763A (zh) 1999-12-15
KR100503845B1 (ko) 2005-07-26
WO1998023589A1 (en) 1998-06-04
EP0944600A1 (en) 1999-09-29

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