ES2161243T3 - Imidazolo-quinoxalinonas para el tratamiento de enfermedades del sistema nervioso central. - Google Patents

Imidazolo-quinoxalinonas para el tratamiento de enfermedades del sistema nervioso central.

Info

Publication number
ES2161243T3
ES2161243T3 ES94911933T ES94911933T ES2161243T3 ES 2161243 T3 ES2161243 T3 ES 2161243T3 ES 94911933 T ES94911933 T ES 94911933T ES 94911933 T ES94911933 T ES 94911933T ES 2161243 T3 ES2161243 T3 ES 2161243T3
Authority
ES
Spain
Prior art keywords
central nervous
pct
quinoxalinones
imidazolo
diseases
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES94911933T
Other languages
English (en)
Inventor
Hans-Joerg Treiber
Berthold Behl
Hans Peter Hofmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
BASF SE
Original Assignee
BASF SE
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by BASF SE filed Critical BASF SE
Application granted granted Critical
Publication of ES2161243T3 publication Critical patent/ES2161243T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/08Antiepileptics; Anticonvulsants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia

Abstract

SE DESCRIBE LA UTILIZACION DE IMIDAZOLO QUINOXALINONAS PARA ELABORACION DE MEDICAMENTOS PARA TRATAMIENTO DE ENFERMEDADES DEL SISTEMA NERVIOSO CENTRAL. LAS IMIDAZOLO QUINOXALINONAS POSEEN LA FORMULA (I) DONDE R{SUB,1}, R{SUP,2} Y X TIENEN EL SIGNIFICADO DADO EN LA DESCRIPCION.
ES94911933T 1993-03-31 1994-03-19 Imidazolo-quinoxalinonas para el tratamiento de enfermedades del sistema nervioso central. Expired - Lifetime ES2161243T3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4310523A DE4310523A1 (de) 1993-03-31 1993-03-31 Imidazolo-chinoxalinone zur Behandlung zentralnervöser Erkrankungen

Publications (1)

Publication Number Publication Date
ES2161243T3 true ES2161243T3 (es) 2001-12-01

Family

ID=6484366

Family Applications (1)

Application Number Title Priority Date Filing Date
ES94911933T Expired - Lifetime ES2161243T3 (es) 1993-03-31 1994-03-19 Imidazolo-quinoxalinonas para el tratamiento de enfermedades del sistema nervioso central.

Country Status (9)

Country Link
US (1) US5538972A (es)
EP (1) EP0691846B1 (es)
JP (1) JPH08508272A (es)
AT (1) ATE203671T1 (es)
CA (1) CA2156624A1 (es)
DE (2) DE4310523A1 (es)
DK (1) DK0691846T3 (es)
ES (1) ES2161243T3 (es)
WO (1) WO1994022447A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH09508632A (ja) * 1994-02-11 1997-09-02 ノボ ノルディスク アクティーゼルスカブ 複素環式化合物並びにそれらの製造及び使用
WO1996010572A1 (de) * 1994-09-30 1996-04-11 Basf Aktiengesellschaft Neue heterocyclische substituierte imidazolo-chinoxalinone, ihre herstellung und verwendung

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2448541A1 (fr) * 1979-02-09 1980-09-05 Roussel Uclaf Nouveaux derives de l'oxoimidazoquinoxaline et leurs sels, leur procede de preparation, leur application comme medicaments et les compositions pharmaceutiques les renfermant
SE441449B (sv) * 1979-02-09 1985-10-07 Roussel Uclaf Heterocykliska derivat och farmaceutiska kompositioner innehallande dessa derivat
DK160941C (da) * 1988-06-28 1991-10-21 Novo Nordisk As Kondenserede 2,3-dihydroxypyraziner, fremgangsmaade til deres fremstilling og farmaceutiske praeparater, hvori forbindelserne indgaar
US5055465A (en) * 1989-05-31 1991-10-08 Berlex Laboratories, Inc. Imidazoquinoxalinones, their aza analogs and process for their preparation
US5166344A (en) * 1989-05-31 1992-11-24 Berlex Laboratories, Inc. Process for the preparation of imidazoquinoxalinones
FR2663029B1 (fr) * 1990-06-07 1992-07-31 Rhone Poulenc Sante Derives de benzothiazole, leur preparation et les medicaments les contenant.
US5153196A (en) * 1991-06-05 1992-10-06 Eli Lilly And Company Excitatory amino acid receptor antagonists and methods for the use thereof
US5182386A (en) * 1991-08-27 1993-01-26 Neurogen Corporation Certain imidazoquinoxalinones; a new class of gaba brain receptor ligands
AU3767793A (en) * 1992-04-03 1993-11-08 Yamanouchi Pharmaceutical Co., Ltd. Fused quinoxalinone derivative and pharmaceutical composition containing the same

Also Published As

Publication number Publication date
EP0691846A1 (de) 1996-01-17
CA2156624A1 (en) 1994-10-13
EP0691846B1 (de) 2001-08-01
WO1994022447A1 (de) 1994-10-13
DK0691846T3 (da) 2001-10-08
ATE203671T1 (de) 2001-08-15
US5538972A (en) 1996-07-23
JPH08508272A (ja) 1996-09-03
DE4310523A1 (de) 1994-10-06
DE59409813D1 (de) 2001-09-06

Similar Documents

Publication Publication Date Title
KR960701051A (ko) 이미다조피리딘 및 이를 위장 질환의 치료에 사용하는 방법(imidazopyridines and their use in treating castrointestinal diseases)
ATE144420T1 (de) Verwendung von riluzol zur behandlung von parkinson und den parkinson-syndromen
AR028705A1 (es) Bis-arilsulfonas
FI961564A0 (fi) Imidatso(1,2-a)pyridiinien alkoksialkyylikarbamaatit
ES2132401T3 (es) Tetrahidro-1h-benzazepinonas y hexahidroazepinonas como antagonistas selectivos del receptor colecistoquinina-b.
ES2161243T3 (es) Imidazolo-quinoxalinonas para el tratamiento de enfermedades del sistema nervioso central.
ES2094638T3 (es) N-acilpirrolidinas y medicamentos para el tratamiento o la prevencion de los desordenes relacionados con la colecistoquinina y la gastrina.
DE69510933D1 (de) Amidderivate und ihre therapeutische anwendung
BR9509337A (pt) Pirrolil-tetra-hidro-benzo-quinoxalino-dionas uso das pirrolil-tetra-hidro-benzo-quinoxalino-dionas e processo para o tratamento de pacientes que apresentam distúrbios neurodegenerativos e distúrbios neurotóxicos do sistema nervoso central
MX9304075A (es) Composicion farmaceutica para el tratamiento o profilaxis de los desordenes trombohemorragicos consuntivos.
MX9307837A (es) Triazolo quinazolinas para el tratamiento de enfermedades del sistema nervioso central.
ES2144857T3 (es) Utilizacion de derivados benzonaftalenicos para la fabricacion de medicamentos destinados para el tratamiento de las enfermedades del sistema nervioso.
ES2123836T3 (es) Imidazo(1,5-a)quinoleinas para el tratamiento de la ansiedad y trastornos del sueño.
ES2140544T3 (es) Utilizacion de efaroxan y de sus derivados para la fabricacion de medicamentos destinados al tratamiento de las enfermedades neurodegenerativas.
ES2109512T3 (es) Macrolactama (ciclamenol) antiinflamatoria.
ATE190845T1 (de) Rektale flunisolid-zubereitung zur behandlung entzündlicher darmerkrankungen
DK0673377T3 (da) Nye triazoloquinazoliner, fremstilling og anvendelse deraf

Legal Events

Date Code Title Description
FG2A Definitive protection

Ref document number: 691846

Country of ref document: ES