ES2153584T3 - Piridiniminil-1,2-benzisoxazol y -benzisotiazol como antipsicoticos. - Google Patents

Piridiniminil-1,2-benzisoxazol y -benzisotiazol como antipsicoticos.

Info

Publication number
ES2153584T3
ES2153584T3 ES96920335T ES96920335T ES2153584T3 ES 2153584 T3 ES2153584 T3 ES 2153584T3 ES 96920335 T ES96920335 T ES 96920335T ES 96920335 T ES96920335 T ES 96920335T ES 2153584 T3 ES2153584 T3 ES 2153584T3
Authority
ES
Spain
Prior art keywords
piridiniminil
benzisotiazol
benzisoxazol
antipsychotics
benzisoxazoles
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES96920335T
Other languages
English (en)
Inventor
David M Fink
Barbara E Kurys
Gregory M Shutske
John D Tomer Iv
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharmaceuticals Inc
Original Assignee
Aventis Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharmaceuticals Inc filed Critical Aventis Pharmaceuticals Inc
Application granted granted Critical
Publication of ES2153584T3 publication Critical patent/ES2153584T3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D231/00Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56Benzopyrazoles; Hydrogenated benzopyrazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D261/00Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/20Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

Abstract

SE DESCRIBEN NUEVOS PIRIDINIMINIL - 1,2 - BENZISOXAZOLES Y BENZISOTIAZOLES Y PROCEDIMIENTOS PARA SU PREPARACION, Y PROCEDIMIENTOS PARA ALIVIAR LA DISFUNCION DE LA MEMORIA Y PARA TRATAR LA DEPRESION UTILIZANDO LOS 1,2 - BENZISOXAZOLES Y BENZISOTIAZOLES Y LOS INTERMEDIOS, O COMPOSICIONES DE LOS MISMOS.
ES96920335T 1995-06-06 1996-05-14 Piridiniminil-1,2-benzisoxazol y -benzisotiazol como antipsicoticos. Expired - Lifetime ES2153584T3 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46602195A 1995-06-06 1995-06-06
US08/637,091 US5668154A (en) 1995-06-06 1996-05-02 Pyridiniminyl-1,2-benzisoxazoles and -benzisothiazoles

Publications (1)

Publication Number Publication Date
ES2153584T3 true ES2153584T3 (es) 2001-03-01

Family

ID=23850131

Family Applications (1)

Application Number Title Priority Date Filing Date
ES96920335T Expired - Lifetime ES2153584T3 (es) 1995-06-06 1996-05-14 Piridiniminil-1,2-benzisoxazol y -benzisotiazol como antipsicoticos.

Country Status (17)

Country Link
US (3) US5668154A (es)
EP (1) EP0848713B1 (es)
KR (1) KR100309215B1 (es)
AR (1) AR002204A1 (es)
AT (1) ATE197153T1 (es)
AU (1) AU708843B2 (es)
CA (1) CA2224171A1 (es)
DE (1) DE69610778T2 (es)
DK (1) DK0848713T3 (es)
ES (1) ES2153584T3 (es)
GR (1) GR3035249T3 (es)
HU (1) HUP9802571A3 (es)
NO (1) NO975682L (es)
NZ (1) NZ308831A (es)
PT (1) PT848713E (es)
TW (1) TW355710B (es)
ZA (1) ZA964565B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6083932A (en) * 1997-04-18 2000-07-04 Cv Technologies Inc. Pharmaceutical compositions derived from ginseng and methods of treatment using same
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US6123554A (en) * 1999-05-28 2000-09-26 Berg Technology, Inc. Connector cover with board stiffener
US9907751B2 (en) * 2016-03-10 2018-03-06 RxOMEG Therapeutics LLC Composition and method of use of colchicine oral liquid
US10226423B1 (en) 2017-12-20 2019-03-12 RxOMEG Therapeutics LLC Colchicine drug-to-drug interactions
CN110117278B (zh) * 2018-02-07 2022-07-19 石家庄以岭药业股份有限公司 烷氧基苯并五元(六元)杂环胺类化合物及其药物用途
WO2023083445A1 (en) 2021-11-10 2023-05-19 Symrise Ag Compositions comprising trpm8 agonistic cooling agents

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5328920A (en) * 1991-04-17 1994-07-12 Hoechst-Roussel Pharmaceuticals Incorporated Substituted (pyridinylamino)-indoles
US5177088A (en) * 1991-04-17 1993-01-05 Hoechst-Roussel Pharmaceuticals Incorporated Substituted 3-(pyridinylamino)-indoles
US5494908A (en) * 1992-11-23 1996-02-27 Hoechst-Roussel Pharmaceutical Incorporated Substituted 3-(aminoalkylamino)-1,2-benzisoxazoles and related compounds

Also Published As

Publication number Publication date
DK0848713T3 (da) 2000-12-18
CA2224171A1 (en) 1996-12-12
ZA964565B (en) 1996-12-12
US5728717A (en) 1998-03-17
AU708843B2 (en) 1999-08-12
MX9709450A (es) 1998-06-28
KR100309215B1 (ko) 2001-12-28
KR19990022265A (ko) 1999-03-25
AR002204A1 (es) 1998-01-07
EP0848713B1 (en) 2000-10-25
HUP9802571A2 (hu) 1999-08-30
DE69610778D1 (de) 2000-11-30
GR3035249T3 (en) 2001-04-30
US5668154A (en) 1997-09-16
EP0848713A1 (en) 1998-06-24
AU5867796A (en) 1996-12-24
DE69610778T2 (de) 2001-06-13
TW355710B (en) 1999-04-11
US5948798A (en) 1999-09-07
NO975682D0 (no) 1997-12-05
HUP9802571A3 (en) 1999-11-29
PT848713E (pt) 2001-02-28
NO975682L (no) 1998-02-05
NZ308831A (en) 1998-11-25
ATE197153T1 (de) 2000-11-15

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