ES2133072A1 - Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central. - Google Patents

Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central.

Info

Publication number
ES2133072A1
ES2133072A1 ES09601852A ES9601852A ES2133072A1 ES 2133072 A1 ES2133072 A1 ES 2133072A1 ES 09601852 A ES09601852 A ES 09601852A ES 9601852 A ES9601852 A ES 9601852A ES 2133072 A1 ES2133072 A1 ES 2133072A1
Authority
ES
Spain
Prior art keywords
nervous system
central nervous
therapeutic activity
glycine derivatives
substituted glycine
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES09601852A
Other languages
English (en)
Other versions
ES2133072B1 (es
Inventor
Stephen Richard Baker
John Goldsworthy
Tercero Concepcion Pedregal
Esteban Almudena Rubio
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Lilly SA
Lilly Industries Ltd
Original Assignee
Lilly SA
Lilly Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly SA, Lilly Industries Ltd filed Critical Lilly SA
Priority to ES009601852A priority Critical patent/ES2133072B1/es
Publication of ES2133072A1 publication Critical patent/ES2133072A1/es
Application granted granted Critical
Publication of ES2133072B1 publication Critical patent/ES2133072B1/es
Anticipated expiration legal-status Critical
Withdrawn - After Issue legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Derivados de glicina n-sustituidos con actividad terapéutica sobre el sistema nervioso central. Compuestos farmacéuticos de fórmula (I), en la que n es 0, 1 ó 2 y m es 1 ó 2, R sup,1 es hidrógeno, alquilo C sub,1-10 , alquenilo C sub,2-10 , alquinilo C sub,2-10 , fenilo, naftilo, alquilfenilo C sub,1-10 , alquenilfenilo C sub,2-10 o alquinilfenilo C sub,2-10 , estando dichos grupos fenilo y naftilo opcionalmente sustituidos, R sup,2 es hidrógeno o un grupo protector y Q es un grupo ácido; o una sal o éster del mismo.
ES009601852A 1996-08-27 1996-08-27 Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central. Withdrawn - After Issue ES2133072B1 (es)

Priority Applications (1)

Application Number Priority Date Filing Date Title
ES009601852A ES2133072B1 (es) 1996-08-27 1996-08-27 Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central.

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES009601852A ES2133072B1 (es) 1996-08-27 1996-08-27 Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central.

Publications (2)

Publication Number Publication Date
ES2133072A1 true ES2133072A1 (es) 1999-08-16
ES2133072B1 ES2133072B1 (es) 2000-04-01

Family

ID=8295903

Family Applications (1)

Application Number Title Priority Date Filing Date
ES009601852A Withdrawn - After Issue ES2133072B1 (es) 1996-08-27 1996-08-27 Derivados de glicina n-sustituidos con actividad terapeutica sobre el sistema nervioso central.

Country Status (1)

Country Link
ES (1) ES2133072B1 (es)

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1467138A (en) * 1975-03-18 1977-03-16 Richardson Merrell Inc Acetylene derivatives of amino acids
EP0394118A1 (fr) * 1989-04-18 1990-10-24 Roussel-Uclaf Nouveaux dérivés insaturés de l'acide 2,6-amino heptanedioique, leur procédé de préparation et leur application comme médicaments
DE3917836A1 (de) * 1989-06-01 1990-12-20 Hoechst Ag (alpha)-trifluormethyl-substituierte aminosaeuren mit acetylenfunktion, verfahren zu deren herstellung und deren verwendung

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1467138A (en) * 1975-03-18 1977-03-16 Richardson Merrell Inc Acetylene derivatives of amino acids
EP0394118A1 (fr) * 1989-04-18 1990-10-24 Roussel-Uclaf Nouveaux dérivés insaturés de l'acide 2,6-amino heptanedioique, leur procédé de préparation et leur application comme médicaments
DE3917836A1 (de) * 1989-06-01 1990-12-20 Hoechst Ag (alpha)-trifluormethyl-substituierte aminosaeuren mit acetylenfunktion, verfahren zu deren herstellung und deren verwendung

Also Published As

Publication number Publication date
ES2133072B1 (es) 2000-04-01

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Legal Events

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EC2A Search report published

Date of ref document: 19990816

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Effective date: 19990816

FA2A Application withdrawn

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