ES2125162A1 - Procedimiento para preparar un compuesto farmaceuticamente activo. - Google Patents

Procedimiento para preparar un compuesto farmaceuticamente activo.

Info

Publication number
ES2125162A1
ES2125162A1 ES09600694A ES9600694A ES2125162A1 ES 2125162 A1 ES2125162 A1 ES 2125162A1 ES 09600694 A ES09600694 A ES 09600694A ES 9600694 A ES9600694 A ES 9600694A ES 2125162 A1 ES2125162 A1 ES 2125162A1
Authority
ES
Spain
Prior art keywords
preparing
active compound
pharmaceutically active
salts
amide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
ES09600694A
Other languages
English (en)
Other versions
ES2125162B1 (es
Inventor
Victor Wiltold Jacewics
Alan David Jones
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
SmithKline Beecham Ltd
Original Assignee
SmithKline Beecham Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by SmithKline Beecham Ltd filed Critical SmithKline Beecham Ltd
Publication of ES2125162A1 publication Critical patent/ES2125162A1/es
Application granted granted Critical
Publication of ES2125162B1 publication Critical patent/ES2125162B1/es
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Procedimiento para reparar un compuesto farmacéuticamente activo, especialmente granisetrón, que comprende hacer reaccionar ácido 1-metilindazol-3-carboxílico o un derivado reactivo del mismo o una de sus sales con un derivado activo de una amida de la estructura (3) o una de sus sales, en que R es un grupo alquilo, aralquilo, arilo o heteroarilo opcionalmente sustituido, seguido, si es necesario, de la descomposición de la bis-amida formada.
ES9600694A 1995-03-25 1996-03-22 Procedimiento para preparar un compuesto farmaceuticamente activo. Expired - Fee Related ES2125162B1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB9506119.8A GB9506119D0 (en) 1995-03-25 1995-03-25 Chemical process

Publications (2)

Publication Number Publication Date
ES2125162A1 true ES2125162A1 (es) 1999-02-16
ES2125162B1 ES2125162B1 (es) 1999-11-16

Family

ID=10771889

Family Applications (1)

Application Number Title Priority Date Filing Date
ES9600694A Expired - Fee Related ES2125162B1 (es) 1995-03-25 1996-03-22 Procedimiento para preparar un compuesto farmaceuticamente activo.

Country Status (3)

Country Link
AT (1) AT406678B (es)
ES (1) ES2125162B1 (es)
GB (1) GB9506119D0 (es)

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0200444A2 (en) * 1985-04-27 1986-11-05 Beecham Group Plc Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity
EP0214772A1 (en) * 1985-08-16 1987-03-18 Beecham Group Plc Novel compounds
EP0223385A2 (en) * 1985-10-21 1987-05-27 Beecham Group Plc 8-Azabicyclo[3,2,1]octane and 9-azabicyclo[3,3,1]nonane derivatives
WO1991001316A1 (en) * 1989-07-21 1991-02-07 Beecham Group Plc New 9-azabicyclo[3.3.1]nonane-derivate
WO1995023799A1 (en) * 1994-03-03 1995-09-08 Smithkline Beecham Plc Process for the preparation of an indazole-3-carboxamide derivative

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9602866D0 (en) * 1996-02-13 1996-04-10 Smithkline Beecham Plc Novel process

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0200444A2 (en) * 1985-04-27 1986-11-05 Beecham Group Plc Azabicyclononyl-indazole-carboxamide having 5-HT antagonist activity
EP0214772A1 (en) * 1985-08-16 1987-03-18 Beecham Group Plc Novel compounds
EP0223385A2 (en) * 1985-10-21 1987-05-27 Beecham Group Plc 8-Azabicyclo[3,2,1]octane and 9-azabicyclo[3,3,1]nonane derivatives
WO1991001316A1 (en) * 1989-07-21 1991-02-07 Beecham Group Plc New 9-azabicyclo[3.3.1]nonane-derivate
WO1995023799A1 (en) * 1994-03-03 1995-09-08 Smithkline Beecham Plc Process for the preparation of an indazole-3-carboxamide derivative

Also Published As

Publication number Publication date
AT406678B (de) 2000-07-25
ES2125162B1 (es) 1999-11-16
GB9506119D0 (en) 1995-05-10
ATA53196A (de) 1999-12-15

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