ES2021048B3 - Un metodo para la preparacion de un derivado de 2,4-diamino-3oxi-pirimidina. - Google Patents

Un metodo para la preparacion de un derivado de 2,4-diamino-3oxi-pirimidina.

Info

Publication number
ES2021048B3
ES2021048B3 ES87306305T ES87306305T ES2021048B3 ES 2021048 B3 ES2021048 B3 ES 2021048B3 ES 87306305 T ES87306305 T ES 87306305T ES 87306305 T ES87306305 T ES 87306305T ES 2021048 B3 ES2021048 B3 ES 2021048B3
Authority
ES
Spain
Prior art keywords
3oxi
pirimidina
diamino
derivative
preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
ES87306305T
Other languages
English (en)
Inventor
Jyrki Lamsa
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Orion Oyj
Original Assignee
Orion Yhtyma Oy
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Orion Yhtyma Oy filed Critical Orion Yhtyma Oy
Application granted granted Critical
Publication of ES2021048B3 publication Critical patent/ES2021048B3/es
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48Two nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
ES87306305T 1986-10-07 1987-07-16 Un metodo para la preparacion de un derivado de 2,4-diamino-3oxi-pirimidina. Expired - Lifetime ES2021048B3 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FI864046A FI864046A (fi) 1986-10-07 1986-10-07 Foerfarande foer framstaellning av en terapeutiskt aktiv foerening.

Publications (1)

Publication Number Publication Date
ES2021048B3 true ES2021048B3 (es) 1991-10-16

Family

ID=8523270

Family Applications (1)

Application Number Title Priority Date Filing Date
ES87306305T Expired - Lifetime ES2021048B3 (es) 1986-10-07 1987-07-16 Un metodo para la preparacion de un derivado de 2,4-diamino-3oxi-pirimidina.

Country Status (18)

Country Link
US (1) US4866174A (es)
EP (1) EP0270201B1 (es)
JP (1) JPS6396175A (es)
KR (1) KR880005095A (es)
AT (1) ATE61584T1 (es)
AU (1) AU590431B2 (es)
CA (1) CA1268766A (es)
DE (1) DE3768617D1 (es)
DK (1) DK348687A (es)
ES (1) ES2021048B3 (es)
FI (2) FI864046A (es)
FR (1) FR2604707B1 (es)
HU (1) HUT44533A (es)
IL (1) IL83351A0 (es)
NO (1) NO872810L (es)
NZ (1) NZ221011A (es)
PT (1) PT85392B (es)
ZA (1) ZA875174B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FI871773A0 (fi) * 1987-04-22 1987-04-22 Farmos Oy Foerfarande foer framstaellning av en terapeutiskt aktiv foerening.
FR2636840B1 (fr) * 1988-09-23 1990-12-21 Norchim Sarl Sel du 6-piperidino-2,4-diaminopyrimidine-3-oxyde et de l'acide aceturique, leur preparation et leur application dermatocosmetologiques
NZ244301A (en) * 1991-09-20 1994-08-26 Merck & Co Inc Preparation of 2-pyridylmethylsulphinylbenzimidazole and pyridoimidazole derivatives from the corresponding sulphenyl compounds
FR2697251B1 (fr) * 1992-10-22 1994-12-02 Synthelabo N-oxydes de dérivés de 1-(4-chlorophényl)-2-[4-[(4-fluorophényl)méthyl] pipéridin-1-yl]éthanol, leur procédé de préparation et leur application en thérapeutique.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3644364A (en) * 1970-03-31 1972-02-22 Upjohn Co Compounds and process
US3998827A (en) * 1971-04-07 1976-12-21 The Upjohn Company 6-amino-4-(substituted piperidino)-1,2-dihydro-1-hydroxy-2-iminopyrimidines
HU177601B (en) * 1978-10-27 1981-11-28 Egyt Gyogyszervegyeszeti Gyar New process for preparing 6-piperidino-2,4-diamino-pyrimidine-3-oxide
EP0027693B2 (en) * 1979-10-18 1988-05-11 Interox Chemicals Limited Magnesium salts of peroxycarboxylic acids, processes for their preparation and their use as bleaching agents in washing compositions, and processes
US4483781A (en) * 1983-09-02 1984-11-20 The Procter & Gamble Company Magnesium salts of peroxycarboxylic acids

Also Published As

Publication number Publication date
DE3768617D1 (de) 1991-04-18
DK348687A (da) 1988-04-08
FI78910B (fi) 1989-06-30
FI873933A (fi) 1988-04-08
PT85392A (en) 1987-08-01
ZA875174B (en) 1988-01-20
FI78910C (fi) 1989-10-10
PT85392B (en) 1990-01-04
FI864046A0 (fi) 1986-10-07
CA1268766A (en) 1990-05-08
EP0270201A1 (en) 1988-06-08
KR880005095A (ko) 1988-06-28
FR2604707A1 (fr) 1988-04-08
NZ221011A (en) 1990-05-28
NO872810L (no) 1988-04-08
US4866174A (en) 1989-09-12
EP0270201B1 (en) 1991-03-13
DK348687D0 (da) 1987-07-07
HUT44533A (en) 1988-03-28
FR2604707B1 (fr) 1989-06-09
IL83351A0 (en) 1987-12-31
FI873933A0 (fi) 1987-09-11
FI864046A (fi) 1988-04-08
NO872810D0 (no) 1987-07-06
ATE61584T1 (de) 1991-03-15
AU590431B2 (en) 1989-11-02
JPS6396175A (ja) 1988-04-27
AU7551787A (en) 1988-04-14

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