ES2003201A6 - Un procedimiento para la preparacion de esteroides aminoglicosidicos. - Google Patents

Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Info

Publication number
ES2003201A6
ES2003201A6 ES8700043A ES8700043A ES2003201A6 ES 2003201 A6 ES2003201 A6 ES 2003201A6 ES 8700043 A ES8700043 A ES 8700043A ES 8700043 A ES8700043 A ES 8700043A ES 2003201 A6 ES2003201 A6 ES 2003201A6
Authority
ES
Spain
Prior art keywords
preparation
pharmaceutical compositions
compositions containing
alkyl
sugar
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8700043A
Other languages
English (en)
Inventor
Laura Chiodini
Mauro Gobbini
Sergio Mantegani
Daniela Ruggieri
Aldemio Temperilli
Gabriella Traquandi
Patrizia Ferrari
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of ES2003201A6 publication Critical patent/ES2003201A6/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J71/00—Steroids in which the cyclopenta(a)hydrophenanthrene skeleton is condensed with a heterocyclic ring
    • C07J71/0036—Nitrogen-containing hetero ring
    • C07J71/0057—Nitrogen and oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE DESCRIBEN COMPUESTOS DE FORMULA I [R1 F H O ALQUILO C1-3, R2 F UN RESTO AMINODESOXI O AMINODIDESOXI O AMINOTRIDESOXI AZUCAR DE LA SERIE D O L SUSTITUIDO CON ALQUILO, SIENDO EL ENLACE GLICOSIDICO A O B] Y SUS SALES FARMACEUTICAMENTE ACEPTABLES, QUE SON UTILES COMO AGENTES ANTIHIPERTENSIVOS. EL PROCEDIMIENTO SE CARACTERIZA POR HACER REACCIONAR LOS DERIVADOS 3-HIDROXI CORRESPONDIENTES CON UN DERIVADO PROTEGIDO ADECUADO DE UN AMINO AZUCAR.
ES8700043A 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos. Expired ES2003201A6 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB868600490A GB8600490D0 (en) 1986-01-09 1986-01-09 Aminoglycoside norcholanic acid lactams

Publications (1)

Publication Number Publication Date
ES2003201A6 true ES2003201A6 (es) 1988-10-16

Family

ID=10591135

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8700043A Expired ES2003201A6 (es) 1986-01-09 1987-01-08 Un procedimiento para la preparacion de esteroides aminoglicosidicos.

Country Status (16)

Country Link
US (1) US4920099A (es)
EP (1) EP0253840B1 (es)
JP (1) JPS63502180A (es)
KR (1) KR880700815A (es)
AU (1) AU582945B2 (es)
DK (1) DK468487D0 (es)
ES (1) ES2003201A6 (es)
FI (1) FI873799A7 (es)
GB (1) GB8600490D0 (es)
GR (1) GR870013B (es)
HU (1) HU199158B (es)
IL (1) IL81165A (es)
NZ (1) NZ218855A (es)
PT (1) PT84073B (es)
WO (1) WO1987004168A1 (es)
ZA (1) ZA87115B (es)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8916635D0 (en) * 1989-07-20 1989-09-06 Erba Carlo Spa Cardanolactam derivatives
CZ171095A3 (en) * 1993-01-08 1996-01-17 Astra Ab Novel steroidal derivatives specific for colon or ilium
ES2146665T3 (es) * 1993-09-24 2000-08-16 Procter & Gamble Nuevos compuestos 14-aminoesteroides que contienen oligosacaridos y nuevo procedimiento en quimica de aminoesteroides diastereoselectivo.
US5922703A (en) * 1993-09-24 1999-07-13 The Procter & Gamble Company Urethane-containing aminosteroid compounds
US6372712B1 (en) 1998-05-22 2002-04-16 The Board Of Trustees Of The Leland Stanford Jr. University Synthetic bifunctional molecules containing a drug moiety and presenter protein ligand
JP4589869B2 (ja) * 2002-07-12 2010-12-01 塩野義製薬株式会社 酸触媒として機能するゼオライト類似体の簡易な製造法
US20040064050A1 (en) * 2002-09-20 2004-04-01 Jun Liu System and method for screening tissue
EP2671508B1 (en) 2005-04-28 2020-09-16 Proteus Digital Health, Inc. Pharma-informatics system
US9062126B2 (en) 2005-09-16 2015-06-23 Raptor Pharmaceuticals Inc. Compositions comprising receptor-associated protein (RAP) variants specific for CR-containing proteins and uses thereof
ES2919563T3 (es) 2009-02-20 2022-07-27 Enhanx Biopharm Inc Sistema de administración de medicamentos a base de glutatión
KR20180114970A (ko) 2009-05-06 2018-10-19 라보라토리 스킨 케어, 인크. 활성제-칼슘 포스페이트 입자 복합체를 포함하는 피부 전달 조성물 및 이들을 이용하는 방법

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3036061A (en) * 1959-08-05 1962-05-22 Ciba Geigy Corp Steroids
US3451994A (en) * 1967-11-02 1969-06-24 American Home Prod 14beta-hydroxy-16beta,21-oxidonorcholan-23-oic acid lactams and derivatives
US3462413A (en) * 1967-11-02 1969-08-19 American Home Prod 14,21-oxidonorcholan-23-oic acid lactams and derivatives
DE2254060A1 (de) * 1972-11-04 1974-05-16 Hoechst Ag Cardenolid-3-eckige klammer auf 4'-amino-2',3',4'-tridesoxy-glykoside eckige klammer zu und verfahren zu ihrer herstellung
DE2603046C2 (de) * 1976-01-28 1983-07-14 Beiersdorf Ag, 2000 Hamburg 4'α- und 4'β-Amino-4'-desoxy-oleandrine, Verfahren zu ihrer Herstellung sowie diese enthaltende pharmazeutische Präparate
JPS54135759A (en) * 1978-04-14 1979-10-22 Kureha Chem Ind Co Ltd Amino sugar-steroid hormone combination
GB8600489D0 (en) * 1986-01-09 1986-02-12 Erba Farmitalia Aminoglycoside steroids
GB8600491D0 (en) * 1986-01-09 1986-02-12 Erba Farmitalia Aminoglycoside norcholanic acid derivatives

Also Published As

Publication number Publication date
HUT46929A (en) 1988-12-28
AU6846987A (en) 1987-07-28
GB8600490D0 (en) 1986-02-12
GR870013B (en) 1987-05-08
US4920099A (en) 1990-04-24
FI873799A0 (fi) 1987-09-01
FI873799L (fi) 1987-09-01
AU582945B2 (en) 1989-04-13
FI873799A7 (fi) 1987-09-01
NZ218855A (en) 1989-06-28
DK468487D0 (da) 1987-09-08
HU199158B (en) 1990-01-29
JPS63502180A (ja) 1988-08-25
PT84073B (pt) 1989-07-31
WO1987004168A1 (en) 1987-07-16
IL81165A (en) 1991-05-12
IL81165A0 (en) 1987-08-31
PT84073A (en) 1987-02-01
EP0253840B1 (en) 1991-04-03
ZA87115B (en) 1987-09-30
KR880700815A (ko) 1988-04-12
EP0253840A1 (en) 1988-01-27
DK468487A (da) 1987-09-07

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991108