EP4232149A2 - Compounds and methods for the treatment of ocular disorders - Google Patents
Compounds and methods for the treatment of ocular disordersInfo
- Publication number
- EP4232149A2 EP4232149A2 EP21882226.0A EP21882226A EP4232149A2 EP 4232149 A2 EP4232149 A2 EP 4232149A2 EP 21882226 A EP21882226 A EP 21882226A EP 4232149 A2 EP4232149 A2 EP 4232149A2
- Authority
- EP
- European Patent Office
- Prior art keywords
- substituted
- alkyl
- radical
- heteroalkyl
- compound
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
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- 125000004404 heteroalkyl group Chemical group 0.000 claims description 362
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- OABOXRPGTFRBFZ-IMJSIDKUSA-N Cys-Cys Chemical compound SC[C@H](N)C(=O)N[C@@H](CS)C(O)=O OABOXRPGTFRBFZ-IMJSIDKUSA-N 0.000 claims description 10
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Classifications
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
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|---|---|---|---|
| US202063094793P | 2020-10-21 | 2020-10-21 | |
| US202163170988P | 2021-04-05 | 2021-04-05 | |
| PCT/IB2021/000707 WO2022084738A2 (en) | 2020-10-21 | 2021-10-20 | Compounds and methods for the treatment of ocular disorders |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| EP4232149A2 true EP4232149A2 (en) | 2023-08-30 |
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Family Applications (1)
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|---|---|---|---|
| EP21882226.0A Pending EP4232149A2 (en) | 2020-10-21 | 2021-10-20 | Compounds and methods for the treatment of ocular disorders |
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| EP (1) | EP4232149A2 (ko) |
| JP (1) | JP2023546453A (ko) |
| KR (1) | KR20230110515A (ko) |
| AU (1) | AU2021363702A1 (ko) |
| CA (1) | CA3196145A1 (ko) |
| IL (1) | IL302173A (ko) |
| MX (1) | MX2023004537A (ko) |
| WO (1) | WO2022084738A2 (ko) |
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| JP2022530322A (ja) | 2019-04-18 | 2022-06-29 | アズーラ オフサルミックス エルティーディー． | 眼障害を処置するための化合物および方法 |
| US11459351B1 (en) | 2021-04-05 | 2022-10-04 | Azura Ophthalmics Ltd. | Compounds and methods for the treatment of ocular disorders |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2003070173A2 (en) * | 2002-02-15 | 2003-08-28 | Sympore Gmbh | Conjugates of biologically active compounds, methods for their preparation and use, formulation and pharmaceutical applications thereof |
| CN114007625A (zh) * | 2019-04-18 | 2022-02-01 | 阿祖拉眼科有限公司 | 用于治疗眼病的化合物和方法 |
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2021
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- 2021-10-20 CA CA3196145A patent/CA3196145A1/en active Pending
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Also Published As
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| IL302173A (en) | 2023-06-01 |
| AU2021363702A9 (en) | 2024-02-08 |
| WO2022084738A3 (en) | 2022-06-30 |
| CA3196145A1 (en) | 2022-04-28 |
| MX2023004537A (es) | 2023-06-15 |
| JP2023546453A (ja) | 2023-11-02 |
| KR20230110515A (ko) | 2023-07-24 |
| WO2022084738A2 (en) | 2022-04-28 |
| AU2021363702A1 (en) | 2023-06-15 |
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