EP2498608A4 - Composés de benzènesulfonamide-thiazole et oxazole - Google Patents
Composés de benzènesulfonamide-thiazole et oxazoleInfo
- Publication number
- EP2498608A4 EP2498608A4 EP10830388.4A EP10830388A EP2498608A4 EP 2498608 A4 EP2498608 A4 EP 2498608A4 EP 10830388 A EP10830388 A EP 10830388A EP 2498608 A4 EP2498608 A4 EP 2498608A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- benzene sulfonamide
- oxazole compounds
- sulfonamide thiazole
- thiazole
- oxazole
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US25976809P | 2009-11-10 | 2009-11-10 | |
| PCT/US2010/051890 WO2011059610A1 (fr) | 2009-11-10 | 2010-10-08 | Composés de benzènesulfonamide-thiazole et oxazole |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EP2498608A1 EP2498608A1 (fr) | 2012-09-19 |
| EP2498608A4 true EP2498608A4 (fr) | 2013-04-24 |
Family
ID=43991933
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EP10830388.4A Withdrawn EP2498608A4 (fr) | 2009-11-10 | 2010-10-08 | Composés de benzènesulfonamide-thiazole et oxazole |
Country Status (2)
| Country | Link |
|---|---|
| EP (1) | EP2498608A4 (fr) |
| WO (1) | WO2011059610A1 (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2012015100A (es) * | 2010-06-25 | 2013-05-01 | Novartis Ag | Compuestos y composiciones de heteroarilo como inhibidores de cinasa de proteina. |
| ES2580961T3 (es) * | 2011-02-24 | 2016-08-30 | Nerviano Medical Sciences S.R.L. | Derivados Tiazolilfenil-bencenosulfonamido como Inhibidores de Cinasa |
| US9242969B2 (en) | 2013-03-14 | 2016-01-26 | Novartis Ag | Biaryl amide compounds as kinase inhibitors |
| CA2912568A1 (fr) | 2013-05-30 | 2014-12-04 | Plexxikon Inc. | Composes pour modulation de kinases, et indications correspondantes |
| UY36294A (es) | 2014-09-12 | 2016-04-29 | Novartis Ag | Compuestos y composiciones como inhibidores de quinasa |
| JP2019532944A (ja) | 2016-09-23 | 2019-11-14 | セルイプセ | Ｌｉｍｋ介在性疾患における、ｌｉｍキナーゼ阻害剤、医薬組成物および使用方法 |
| WO2020124397A1 (fr) * | 2018-12-19 | 2020-06-25 | Inventisbio Shanghai Ltd. | Inhibiteurs de kinase src c-terminale |
| WO2021110997A1 (fr) * | 2019-12-05 | 2021-06-10 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Composés de n-(3-(5-(pyrimidin-4-yl)thiazol-4-yl)phényl)sulfonamide et leurs utilisations en tant qu'inhibiteurs de braf |
| CN111320548B (zh) * | 2020-04-24 | 2022-10-18 | 浦拉司科技（上海）有限责任公司 | 抗癌药物中间体2-氟-3-氨基苯甲酸甲酯的合成方法 |
| CN114560774A (zh) * | 2020-11-27 | 2022-05-31 | 瑞博(杭州)医药科技有限公司 | 一种2-氟-3-硝基苯甲酸的合成方法 |
| WO2023070076A1 (fr) * | 2021-10-22 | 2023-04-27 | The Board Of Trustees Of The University Of Illinois | Composés contre les cancers provoqués par une mutation de braf |
| CN115850103B (zh) * | 2023-01-19 | 2023-04-28 | 北京颖泰嘉和生物科技股份有限公司 | 3-氨基-2-氟苯甲酸甲酯的制备方法 |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005116025A2 (fr) * | 2004-05-26 | 2005-12-08 | Cyclacel Limited | Composes |
| WO2009137391A2 (fr) * | 2008-05-06 | 2009-11-12 | Smithkline Beecham Corporation | Composés de benzène sulfonamide thiazole et oxazole |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110098296A1 (en) * | 2007-12-13 | 2011-04-28 | George Adjabeng | Thiazole And Oxazole Kinase Inhibitors |
-
2010
- 2010-10-08 WO PCT/US2010/051890 patent/WO2011059610A1/fr active Application Filing
- 2010-10-08 EP EP10830388.4A patent/EP2498608A4/fr not_active Withdrawn
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2005116025A2 (fr) * | 2004-05-26 | 2005-12-08 | Cyclacel Limited | Composes |
| WO2009137391A2 (fr) * | 2008-05-06 | 2009-11-12 | Smithkline Beecham Corporation | Composés de benzène sulfonamide thiazole et oxazole |
Non-Patent Citations (1)
| Title |
|---|
| See also references of WO2011059610A1 * |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011059610A1 (fr) | 2011-05-19 |
| EP2498608A1 (fr) | 2012-09-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
| 17P | Request for examination filed |
Effective date: 20120608 |
|
| AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AL AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO RS SE SI SK SM TR |
|
| DAX | Request for extension of the european patent (deleted) | ||
| A4 | Supplementary search report drawn up and despatched |
Effective date: 20130327 |
|
| RIC1 | Information provided on ipc code assigned before grant |
Ipc: A01N 43/78 20060101AFI20130321BHEP Ipc: C07D 417/14 20060101ALI20130321BHEP Ipc: C07D 413/04 20060101ALI20130321BHEP Ipc: A61K 31/425 20060101ALI20130321BHEP Ipc: C07D 417/04 20060101ALI20130321BHEP |
|
| STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
| 18D | Application deemed to be withdrawn |
Effective date: 20130503 |