EP2307016A4 - Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate - Google Patents

Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate

Info

Publication number
EP2307016A4
EP2307016A4 EP09803180A EP09803180A EP2307016A4 EP 2307016 A4 EP2307016 A4 EP 2307016A4 EP 09803180 A EP09803180 A EP 09803180A EP 09803180 A EP09803180 A EP 09803180A EP 2307016 A4 EP2307016 A4 EP 2307016A4
Authority
EP
European Patent Office
Prior art keywords
bisphosphonate
salt
preventing
pharmaceutical composition
treating osteoporosis
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP09803180A
Other languages
German (de)
English (en)
Other versions
EP2307016A2 (fr
Inventor
Jin Soo Lee
Yun Ha Hwang
Jei Man Ryu
Young Goo Jin
Ki Yoon Kim
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dong Wha Pharm Co Ltd
Original Assignee
Dong Wha Pharm Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dong Wha Pharm Co Ltd filed Critical Dong Wha Pharm Co Ltd
Publication of EP2307016A2 publication Critical patent/EP2307016A2/fr
Publication of EP2307016A4 publication Critical patent/EP2307016A4/fr
Withdrawn legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/662Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
    • A61K31/663Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/08Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A61P19/10Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
EP09803180A 2008-08-01 2009-07-31 Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate Withdrawn EP2307016A4 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20080075791 2008-08-01
KR1020090007774A KR20100014090A (ko) 2008-08-01 2009-01-31 벤즈아미딘 유도체 또는 이의 염, 및 비스포스포네이트를 포함하는 골다공증의 예방 또는 치료용 약학 조성물
PCT/KR2009/004295 WO2010013975A2 (fr) 2008-08-01 2009-07-31 Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate

Publications (2)

Publication Number Publication Date
EP2307016A2 EP2307016A2 (fr) 2011-04-13
EP2307016A4 true EP2307016A4 (fr) 2011-12-28

Family

ID=42087985

Family Applications (1)

Application Number Title Priority Date Filing Date
EP09803180A Withdrawn EP2307016A4 (fr) 2008-08-01 2009-07-31 Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate

Country Status (6)

Country Link
EP (1) EP2307016A4 (fr)
JP (1) JP2011529876A (fr)
KR (2) KR20100014090A (fr)
CN (1) CN102149381A (fr)
CA (1) CA2732864A1 (fr)
WO (1) WO2010013975A2 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9187485B2 (en) 2007-02-02 2015-11-17 Baylor College Of Medicine Methods and compositions for the treatment of cancer and related hyperproliferative disorders
WO2010013969A2 (fr) * 2008-08-01 2010-02-04 Dong Wha Pharmaceutical Co., Ltd. Composition pharmaceutique pour prévenir ou traiter l'ostéoporose à base de dérivés de benzamidine ou de sels de ceux-ci, et d'acide alendronique ou de sels de celui-ci
JP2016534124A (ja) * 2013-08-29 2016-11-04 ベイラー カレッジ オブ メディスンBaylor College Of Medicine 代謝並びに体重関連疾患の処置のための組成物および方法
WO2016054105A1 (fr) 2014-09-29 2016-04-07 A123 Systems, LLC Anodes de silicium pré-lithiées avec liant pvdf

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001001991A1 (fr) * 1999-07-01 2001-01-11 Merck & Co., Inc. Comprimes pharmaceutiques
WO2004056373A1 (fr) * 2002-12-20 2004-07-08 F. Hoffmann-La Roche Ag Formulation d'ibandronate a forte dose
WO2007089101A1 (fr) * 2006-01-31 2007-08-09 Dong Wha Pharmaceutical Ind.Co., Ltd. Nouveaux dérivés de benzamidine, procédé de fabrication et composition pharmaceutique les renfermant
WO2009017222A1 (fr) * 2007-08-02 2009-02-05 Teijin Pharma Limited Agent préventif ou agent thérapeutique pour une maladie provoquée par un métabolisme osseux anormal

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5451700A (en) * 1991-06-11 1995-09-19 Ciba-Geigy Corporation Amidino compounds, their manufacture and methods of treatment
CA2278190A1 (fr) * 1997-02-04 1998-08-06 Hong-Suk Suh Derive 3-amino-1,2-benzoisoxazole, procede de preparation et utilisation
US5998390A (en) * 1998-09-28 1999-12-07 The Research Foundation Of State University Of New York Combination of bisphosphonate and tetracycline
KR100317935B1 (ko) * 1999-10-20 2001-12-22 유승필 대사성 골질환 치료용 약제조성물 및 이의 제조방법
KR100454767B1 (ko) * 2001-07-19 2004-11-03 동화약품공업주식회사 4-[(4-티아졸릴)페녹시]알콕시-벤즈아미딘 유도체의골다공증 예방 및 치료제로서의 용도
JP2003292453A (ja) * 2002-04-02 2003-10-15 Asahi Kasei Corp 骨疾患治療用医薬複合剤
JPWO2005002590A1 (ja) * 2003-07-01 2006-08-10 アステラス製薬株式会社 骨量増加誘導剤
CA2528805A1 (fr) * 2003-08-13 2005-05-06 Chiron Corporation Inhibiteurs de gsk-3 et utilisations
CN1950086A (zh) * 2004-04-28 2007-04-18 默克公司 作为雄激素受体调节剂的氟化的4-氮杂甾族化合物
JP4657296B2 (ja) * 2004-07-05 2011-03-23 ドン ファ ファーマシューティカル カンパニー リミテッド 骨折治療用薬学的組成物
JP2009017222A (ja) * 2007-07-04 2009-01-22 Panasonic Corp 色調整装置、色調整方法および色調整装置の集積回路
WO2010013969A2 (fr) * 2008-08-01 2010-02-04 Dong Wha Pharmaceutical Co., Ltd. Composition pharmaceutique pour prévenir ou traiter l'ostéoporose à base de dérivés de benzamidine ou de sels de ceux-ci, et d'acide alendronique ou de sels de celui-ci

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2001001991A1 (fr) * 1999-07-01 2001-01-11 Merck & Co., Inc. Comprimes pharmaceutiques
WO2004056373A1 (fr) * 2002-12-20 2004-07-08 F. Hoffmann-La Roche Ag Formulation d'ibandronate a forte dose
WO2007089101A1 (fr) * 2006-01-31 2007-08-09 Dong Wha Pharmaceutical Ind.Co., Ltd. Nouveaux dérivés de benzamidine, procédé de fabrication et composition pharmaceutique les renfermant
WO2009017222A1 (fr) * 2007-08-02 2009-02-05 Teijin Pharma Limited Agent préventif ou agent thérapeutique pour une maladie provoquée par un métabolisme osseux anormal

Also Published As

Publication number Publication date
WO2010013975A3 (fr) 2010-06-03
CN102149381A (zh) 2011-08-10
CA2732864A1 (fr) 2010-02-04
KR20100014090A (ko) 2010-02-10
EP2307016A2 (fr) 2011-04-13
WO2010013975A2 (fr) 2010-02-04
KR20100014174A (ko) 2010-02-10
JP2011529876A (ja) 2011-12-15

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