EP2307016A4 - Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate - Google Patents
Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonateInfo
- Publication number
- EP2307016A4 EP2307016A4 EP09803180A EP09803180A EP2307016A4 EP 2307016 A4 EP2307016 A4 EP 2307016A4 EP 09803180 A EP09803180 A EP 09803180A EP 09803180 A EP09803180 A EP 09803180A EP 2307016 A4 EP2307016 A4 EP 2307016A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- bisphosphonate
- salt
- preventing
- pharmaceutical composition
- treating osteoporosis
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 229940122361 Bisphosphonate Drugs 0.000 title 1
- 208000001132 Osteoporosis Diseases 0.000 title 1
- 150000003937 benzamidines Chemical class 0.000 title 1
- 150000004663 bisphosphonates Chemical class 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/66—Phosphorus compounds
- A61K31/662—Phosphorus acids or esters thereof having P—C bonds, e.g. foscarnet, trichlorfon
- A61K31/663—Compounds having two or more phosphorus acid groups or esters thereof, e.g. clodronic acid, pamidronic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Physical Education & Sports Medicine (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
KR20080075791 | 2008-08-01 | ||
KR1020090007774A KR20100014090A (ko) | 2008-08-01 | 2009-01-31 | 벤즈아미딘 유도체 또는 이의 염, 및 비스포스포네이트를 포함하는 골다공증의 예방 또는 치료용 약학 조성물 |
PCT/KR2009/004295 WO2010013975A2 (fr) | 2008-08-01 | 2009-07-31 | Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate |
Publications (2)
Publication Number | Publication Date |
---|---|
EP2307016A2 EP2307016A2 (fr) | 2011-04-13 |
EP2307016A4 true EP2307016A4 (fr) | 2011-12-28 |
Family
ID=42087985
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP09803180A Withdrawn EP2307016A4 (fr) | 2008-08-01 | 2009-07-31 | Composition pharmaceutique pour prévenir ou traiter l'ostéoporose comprenant un dérivé de benzamidine ou un sel de celui-ci, et du bisphosphonate |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP2307016A4 (fr) |
JP (1) | JP2011529876A (fr) |
KR (2) | KR20100014090A (fr) |
CN (1) | CN102149381A (fr) |
CA (1) | CA2732864A1 (fr) |
WO (1) | WO2010013975A2 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9187485B2 (en) | 2007-02-02 | 2015-11-17 | Baylor College Of Medicine | Methods and compositions for the treatment of cancer and related hyperproliferative disorders |
WO2010013969A2 (fr) * | 2008-08-01 | 2010-02-04 | Dong Wha Pharmaceutical Co., Ltd. | Composition pharmaceutique pour prévenir ou traiter l'ostéoporose à base de dérivés de benzamidine ou de sels de ceux-ci, et d'acide alendronique ou de sels de celui-ci |
JP2016534124A (ja) * | 2013-08-29 | 2016-11-04 | ベイラー カレッジ オブ メディスンBaylor College Of Medicine | 代謝並びに体重関連疾患の処置のための組成物および方法 |
WO2016054105A1 (fr) | 2014-09-29 | 2016-04-07 | A123 Systems, LLC | Anodes de silicium pré-lithiées avec liant pvdf |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001001991A1 (fr) * | 1999-07-01 | 2001-01-11 | Merck & Co., Inc. | Comprimes pharmaceutiques |
WO2004056373A1 (fr) * | 2002-12-20 | 2004-07-08 | F. Hoffmann-La Roche Ag | Formulation d'ibandronate a forte dose |
WO2007089101A1 (fr) * | 2006-01-31 | 2007-08-09 | Dong Wha Pharmaceutical Ind.Co., Ltd. | Nouveaux dérivés de benzamidine, procédé de fabrication et composition pharmaceutique les renfermant |
WO2009017222A1 (fr) * | 2007-08-02 | 2009-02-05 | Teijin Pharma Limited | Agent préventif ou agent thérapeutique pour une maladie provoquée par un métabolisme osseux anormal |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5451700A (en) * | 1991-06-11 | 1995-09-19 | Ciba-Geigy Corporation | Amidino compounds, their manufacture and methods of treatment |
CA2278190A1 (fr) * | 1997-02-04 | 1998-08-06 | Hong-Suk Suh | Derive 3-amino-1,2-benzoisoxazole, procede de preparation et utilisation |
US5998390A (en) * | 1998-09-28 | 1999-12-07 | The Research Foundation Of State University Of New York | Combination of bisphosphonate and tetracycline |
KR100317935B1 (ko) * | 1999-10-20 | 2001-12-22 | 유승필 | 대사성 골질환 치료용 약제조성물 및 이의 제조방법 |
KR100454767B1 (ko) * | 2001-07-19 | 2004-11-03 | 동화약품공업주식회사 | 4-[(4-티아졸릴)페녹시]알콕시-벤즈아미딘 유도체의골다공증 예방 및 치료제로서의 용도 |
JP2003292453A (ja) * | 2002-04-02 | 2003-10-15 | Asahi Kasei Corp | 骨疾患治療用医薬複合剤 |
JPWO2005002590A1 (ja) * | 2003-07-01 | 2006-08-10 | アステラス製薬株式会社 | 骨量増加誘導剤 |
CA2528805A1 (fr) * | 2003-08-13 | 2005-05-06 | Chiron Corporation | Inhibiteurs de gsk-3 et utilisations |
CN1950086A (zh) * | 2004-04-28 | 2007-04-18 | 默克公司 | 作为雄激素受体调节剂的氟化的4-氮杂甾族化合物 |
JP4657296B2 (ja) * | 2004-07-05 | 2011-03-23 | ドン ファ ファーマシューティカル カンパニー リミテッド | 骨折治療用薬学的組成物 |
JP2009017222A (ja) * | 2007-07-04 | 2009-01-22 | Panasonic Corp | 色調整装置、色調整方法および色調整装置の集積回路 |
WO2010013969A2 (fr) * | 2008-08-01 | 2010-02-04 | Dong Wha Pharmaceutical Co., Ltd. | Composition pharmaceutique pour prévenir ou traiter l'ostéoporose à base de dérivés de benzamidine ou de sels de ceux-ci, et d'acide alendronique ou de sels de celui-ci |
-
2009
- 2009-01-31 KR KR1020090007774A patent/KR20100014090A/ko unknown
- 2009-07-31 WO PCT/KR2009/004295 patent/WO2010013975A2/fr active Application Filing
- 2009-07-31 EP EP09803180A patent/EP2307016A4/fr not_active Withdrawn
- 2009-07-31 CN CN2009801335866A patent/CN102149381A/zh active Pending
- 2009-07-31 JP JP2011521047A patent/JP2011529876A/ja active Pending
- 2009-07-31 KR KR1020090070538A patent/KR20100014174A/ko not_active Application Discontinuation
- 2009-07-31 CA CA2732864A patent/CA2732864A1/fr not_active Abandoned
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2001001991A1 (fr) * | 1999-07-01 | 2001-01-11 | Merck & Co., Inc. | Comprimes pharmaceutiques |
WO2004056373A1 (fr) * | 2002-12-20 | 2004-07-08 | F. Hoffmann-La Roche Ag | Formulation d'ibandronate a forte dose |
WO2007089101A1 (fr) * | 2006-01-31 | 2007-08-09 | Dong Wha Pharmaceutical Ind.Co., Ltd. | Nouveaux dérivés de benzamidine, procédé de fabrication et composition pharmaceutique les renfermant |
WO2009017222A1 (fr) * | 2007-08-02 | 2009-02-05 | Teijin Pharma Limited | Agent préventif ou agent thérapeutique pour une maladie provoquée par un métabolisme osseux anormal |
Also Published As
Publication number | Publication date |
---|---|
WO2010013975A3 (fr) | 2010-06-03 |
CN102149381A (zh) | 2011-08-10 |
CA2732864A1 (fr) | 2010-02-04 |
KR20100014090A (ko) | 2010-02-10 |
EP2307016A2 (fr) | 2011-04-13 |
WO2010013975A2 (fr) | 2010-02-04 |
KR20100014174A (ko) | 2010-02-10 |
JP2011529876A (ja) | 2011-12-15 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 20110201 |
|
AK | Designated contracting states |
Kind code of ref document: A2 Designated state(s): AT BE BG CH CY CZ DE DK EE ES FI FR GB GR HR HU IE IS IT LI LT LU LV MC MK MT NL NO PL PT RO SE SI SK SM TR |
|
AX | Request for extension of the european patent |
Extension state: AL BA RS |
|
DAX | Request for extension of the european patent (deleted) | ||
A4 | Supplementary search report drawn up and despatched |
Effective date: 20111124 |
|
RIC1 | Information provided on ipc code assigned before grant |
Ipc: A61K 45/06 20060101ALI20111118BHEP Ipc: A61K 31/663 20060101ALI20111118BHEP Ipc: A61P 19/10 20060101ALI20111118BHEP Ipc: A61K 31/426 20060101AFI20111118BHEP |
|
GRAP | Despatch of communication of intention to grant a patent |
Free format text: ORIGINAL CODE: EPIDOSNIGR1 |
|
STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20130802 |