EP1790636A4 - Piperidinderivate und deren anwendung - Google Patents

Piperidinderivate und deren anwendung

Info

Publication number
EP1790636A4
EP1790636A4 EP05785870A EP05785870A EP1790636A4 EP 1790636 A4 EP1790636 A4 EP 1790636A4 EP 05785870 A EP05785870 A EP 05785870A EP 05785870 A EP05785870 A EP 05785870A EP 1790636 A4 EP1790636 A4 EP 1790636A4
Authority
EP
European Patent Office
Prior art keywords
optionally substituted
salts
piperidine derivatives
compounds
preventive
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP05785870A
Other languages
English (en)
French (fr)
Japanese (ja)
Other versions
EP1790636A1 (de
Inventor
Yoshinori Ikeura
T Hashimoto
Haruyuki Nishida
Junya Shirai
N Sakauchi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Takeda Pharmaceutical Co Ltd
Original Assignee
Takeda Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical Co Ltd filed Critical Takeda Pharmaceutical Co Ltd
Publication of EP1790636A1 publication Critical patent/EP1790636A1/de
Publication of EP1790636A4 publication Critical patent/EP1790636A4/de
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D211/40—Oxygen atoms
    • C07D211/44—Oxygen atoms attached in position 4
    • C07D211/46—Oxygen atoms attached in position 4 having a hydrogen atom as the second substituent in position 4
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    • C07D401/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
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    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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EP05785870A 2004-09-17 2005-09-16 Piperidinderivate und deren anwendung Withdrawn EP1790636A4 (de)

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JP2004272639 2004-09-17
PCT/JP2005/017538 WO2006030975A1 (ja) 2004-09-17 2005-09-16 ピペリジン誘導体およびその用途

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TW200526626A (en) 2003-09-13 2005-08-16 Astrazeneca Ab Chemical compounds
CN101061095A (zh) * 2004-11-22 2007-10-24 默克公司 环烷基哌啶速激肽受体拮抗剂
US20080076783A1 (en) * 2004-11-22 2008-03-27 Merck & Co., Inc. Cycloalkyl Keto Piperidine Tachykinin Receptor Antagonists
EP1817302A4 (de) * 2004-11-22 2009-07-01 Merck & Co Inc Piperidinylpiperidin-tachykinin-rezeptorantagonisten
US20080161306A1 (en) * 2005-02-18 2008-07-03 Brian Sherer Pyrrole Derivatives as Dna Gyrase and Topoisomerase Inhibitors
CN101163693B (zh) 2005-02-18 2013-03-06 阿斯利康(瑞典)有限公司 抗菌哌啶衍生物
TW200716603A (en) * 2005-04-21 2007-05-01 Takeda Pharmaceuticals Co Piperidine derivative crystal, process for producing the same, and use
WO2006115285A1 (ja) * 2005-04-21 2006-11-02 Takeda Pharmaceutical Company Limited 医薬組成物
JP2009502739A (ja) * 2005-08-04 2009-01-29 武田薬品工業株式会社 タキキニン受容体拮抗剤としてのピペリジン誘導体
USRE49686E1 (en) 2008-09-19 2023-10-10 Takeda Pharmaceutical Company Limited Nitrogen-containing heterocyclic compound and use of same
WO2010091411A1 (en) * 2009-02-09 2010-08-12 Glaxosmithkline Llc Piperidinyl cyclic amido antiviral agents
DE20168827T1 (de) 2017-06-30 2021-01-21 Gtx Medical B.V. System zur neuromodulierung
DE18205821T1 (de) 2018-11-13 2020-12-24 Gtx Medical B.V. Steuerungssystem zur bewegungsrekonstruktion und/oder wiederherstellung für einen patienten
EP3695878B1 (de) 2019-02-12 2023-04-19 ONWARD Medical N.V. System zur neuromodulierung
DE19211698T1 (de) 2019-11-27 2021-09-02 Onward Medical B.V. Neuromodulation system

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WO2006057921A2 (en) * 2004-11-22 2006-06-01 Merck & Co., Inc. Piperidinyl piperidine tachykinin receptor antagonists
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