EP1333807A4 - ERYTHROMYCIN DERIVATIVES WITH PROLONGED RELEASE - Google Patents

ERYTHROMYCIN DERIVATIVES WITH PROLONGED RELEASE

Info

Publication number
EP1333807A4
EP1333807A4 EP01986972A EP01986972A EP1333807A4 EP 1333807 A4 EP1333807 A4 EP 1333807A4 EP 01986972 A EP01986972 A EP 01986972A EP 01986972 A EP01986972 A EP 01986972A EP 1333807 A4 EP1333807 A4 EP 1333807A4
Authority
EP
European Patent Office
Prior art keywords
extended release
erythromycin derivatives
release erythromycin
derivatives
extended
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP01986972A
Other languages
German (de)
English (en)
French (fr)
Other versions
EP1333807A2 (en
Inventor
Sandra E Wassink
Donald J Treacy Jr
Edward M Rudnic
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
MiddleBrook Pharmaceuticals Inc
Original Assignee
Advancis Pharmaceutical Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Advancis Pharmaceutical Corp filed Critical Advancis Pharmaceutical Corp
Publication of EP1333807A2 publication Critical patent/EP1333807A2/en
Publication of EP1333807A4 publication Critical patent/EP1333807A4/en
Withdrawn legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
EP01986972A 2000-10-13 2001-10-12 ERYTHROMYCIN DERIVATIVES WITH PROLONGED RELEASE Withdrawn EP1333807A4 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US689988 1991-04-23
US68998800A 2000-10-13 2000-10-13
PCT/US2001/032055 WO2002038577A2 (en) 2000-10-13 2001-10-12 Extended release erythromycin derivatives

Publications (2)

Publication Number Publication Date
EP1333807A2 EP1333807A2 (en) 2003-08-13
EP1333807A4 true EP1333807A4 (en) 2005-06-29

Family

ID=24770642

Family Applications (1)

Application Number Title Priority Date Filing Date
EP01986972A Withdrawn EP1333807A4 (en) 2000-10-13 2001-10-12 ERYTHROMYCIN DERIVATIVES WITH PROLONGED RELEASE

Country Status (6)

Country Link
EP (1) EP1333807A4 (ja)
JP (1) JP2004528272A (ja)
AU (1) AU2002239232A1 (ja)
CA (1) CA2425688A1 (ja)
MX (1) MXPA03003146A (ja)
WO (1) WO2002038577A2 (ja)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6544555B2 (en) 2000-02-24 2003-04-08 Advancis Pharmaceutical Corp. Antibiotic product, use and formulation thereof
US20020068078A1 (en) 2000-10-13 2002-06-06 Rudnic Edward M. Antifungal product, use and formulation thereof
JP2007502294A (ja) 2003-08-12 2007-02-08 アドバンシス ファーマスーティカル コーポレイション 抗生物質製剤、その使用法及び作成方法
MX2007005306A (es) 2004-11-04 2007-06-11 Xenoport Inc Formas de dosis oral de liberacion sostenida de la prodroga gabapentina.

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1991019486A1 (en) * 1990-06-14 1991-12-26 Kalmo Enterprises, Inc. Stable aqueous drug suspensions
US5707646A (en) * 1992-03-12 1998-01-13 Taisho Pharmaceutical Co., Ltd. Taste masking pharmaceutical composition
EP0826376A1 (en) * 1995-05-02 1998-03-04 Taisho Pharmaceutical Co. Ltd Composition for oral administration
US5780604A (en) * 1997-09-26 1998-07-14 Abbott Laboratories 11,12-cyclic phosphite or phosphate derivatives of erythromycin and related macrolides
US5858986A (en) * 1996-07-29 1999-01-12 Abbott Laboratories Crystal form I of clarithromycin
WO2000054811A1 (fr) * 1999-03-17 2000-09-21 Daiichi Pharmaceutical Co., Ltd. Compositions medicamenteuses
WO2000069415A2 (en) * 1999-05-19 2000-11-23 LEK, tovarna farmacevtskih in kemičnih izdelkov, d.d. Melt granulation

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3108046A (en) * 1960-11-25 1963-10-22 Smith Kline French Lab Method of preparing high dosage sustained release tablet and product of this method
JPS49107855A (ja) * 1973-02-03 1974-10-14
JP2528652B2 (ja) * 1987-03-30 1996-08-28 エスエス製薬株式会社 持効性セフラジン製剤
US4808411A (en) * 1987-06-05 1989-02-28 Abbott Laboratories Antibiotic-polymer compositions
JPH07267850A (ja) * 1994-03-28 1995-10-17 Eisai Co Ltd 不快味を防止した医薬組成物及びその製造方法
US6010718A (en) * 1997-04-11 2000-01-04 Abbott Laboratories Extended release formulations of erythromycin derivatives
JP2000169364A (ja) * 1998-09-30 2000-06-20 Taisho Pharmaceut Co Ltd 経口製剤用粒子

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1991019486A1 (en) * 1990-06-14 1991-12-26 Kalmo Enterprises, Inc. Stable aqueous drug suspensions
US5707646A (en) * 1992-03-12 1998-01-13 Taisho Pharmaceutical Co., Ltd. Taste masking pharmaceutical composition
EP0826376A1 (en) * 1995-05-02 1998-03-04 Taisho Pharmaceutical Co. Ltd Composition for oral administration
US5858986A (en) * 1996-07-29 1999-01-12 Abbott Laboratories Crystal form I of clarithromycin
US5780604A (en) * 1997-09-26 1998-07-14 Abbott Laboratories 11,12-cyclic phosphite or phosphate derivatives of erythromycin and related macrolides
WO2000054811A1 (fr) * 1999-03-17 2000-09-21 Daiichi Pharmaceutical Co., Ltd. Compositions medicamenteuses
WO2000069415A2 (en) * 1999-05-19 2000-11-23 LEK, tovarna farmacevtskih in kemičnih izdelkov, d.d. Melt granulation

Also Published As

Publication number Publication date
AU2002239232A1 (en) 2002-05-21
JP2004528272A (ja) 2004-09-16
WO2002038577A3 (en) 2002-09-19
EP1333807A2 (en) 2003-08-13
CA2425688A1 (en) 2002-05-16
WO2002038577A2 (en) 2002-05-16
MXPA03003146A (es) 2004-12-06

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Legal Events

Date Code Title Description
PUAI Public reference made under article 153(3) epc to a published international application that has entered the european phase

Free format text: ORIGINAL CODE: 0009012

17P Request for examination filed

Effective date: 20030509

AK Designated contracting states

Designated state(s): AT BE CH CY DE DK ES FI FR GB GR IE IT LI LU MC NL PT SE TR

AX Request for extension of the european patent

Extension state: AL LT LV MK RO SI

RIN1 Information on inventor provided before grant (corrected)

Inventor name: RUDNIC, EDWARD, M.

Inventor name: TREACY, DONALD, J., JR.

Inventor name: WASSINK, SANDRA, E.

A4 Supplementary search report drawn up and despatched

Effective date: 20050518

RIC1 Information provided on ipc code assigned before grant

Ipc: 7A 61K 31/7048 B

Ipc: 7A 61K 47/14 B

Ipc: 7A 61K 47/10 B

Ipc: 7A 61K 47/02 B

Ipc: 7A 61K 9/22 B

Ipc: 7A 61K 9/20 A

STAA Information on the status of an ep patent application or granted ep patent

Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN

18D Application deemed to be withdrawn

Effective date: 20050803