EP1140961A1 - Process for the preparation of ganglioside gm3 by acid hydrolysis of ganglioside inner esters and its use in the pharmaceutical field - Google Patents

Process for the preparation of ganglioside gm3 by acid hydrolysis of ganglioside inner esters and its use in the pharmaceutical field

Info

Publication number
EP1140961A1
EP1140961A1 EP99963541A EP99963541A EP1140961A1 EP 1140961 A1 EP1140961 A1 EP 1140961A1 EP 99963541 A EP99963541 A EP 99963541A EP 99963541 A EP99963541 A EP 99963541A EP 1140961 A1 EP1140961 A1 EP 1140961A1
Authority
EP
European Patent Office
Prior art keywords
ganglioside
derivatives
preparation
process according
gml
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
EP99963541A
Other languages
German (de)
English (en)
French (fr)
Inventor
Günter Kirschner
Sandro Sonnino
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fidia Farmaceutici SpA
Original Assignee
Fidia SpA
Fidia Farmaceutici SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fidia SpA, Fidia Farmaceutici SpA filed Critical Fidia SpA
Publication of EP1140961A1 publication Critical patent/EP1140961A1/en
Withdrawn legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/02—Acyclic radicals, not substituted by cyclic structures
    • C07H15/04—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical
    • C07H15/10—Acyclic radicals, not substituted by cyclic structures attached to an oxygen atom of the saccharide radical containing unsaturated carbon-to-carbon bonds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Biotechnology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Saccharide Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
EP99963541A 1998-12-16 1999-12-15 Process for the preparation of ganglioside gm3 by acid hydrolysis of ganglioside inner esters and its use in the pharmaceutical field Withdrawn EP1140961A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ITPD980293 1998-12-16
IT000293 IT1302530B1 (it) 1998-12-16 1998-12-16 Processo di preparazione del ganglioside gm3 e dei suoi lisoderivati apartire dal ganglioside gm1.
PCT/EP1999/009958 WO2000035932A1 (en) 1998-12-16 1999-12-15 Process for the preparation of ganglioside gm3 by acid hydrolysis of ganglioside inner esters and its use in the pharmaceutical field

Publications (1)

Publication Number Publication Date
EP1140961A1 true EP1140961A1 (en) 2001-10-10

Family

ID=11392394

Family Applications (1)

Application Number Title Priority Date Filing Date
EP99963541A Withdrawn EP1140961A1 (en) 1998-12-16 1999-12-15 Process for the preparation of ganglioside gm3 by acid hydrolysis of ganglioside inner esters and its use in the pharmaceutical field

Country Status (5)

Country Link
EP (1) EP1140961A1 (it)
AU (1) AU1979800A (it)
CA (1) CA2355106A1 (it)
IT (1) IT1302530B1 (it)
WO (1) WO2000035932A1 (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT201800007093A1 (it) * 2018-07-11 2020-01-11 Oligosaccaridi per l’uso nel trattamento della malattia di Parkinson
CN110507663A (zh) * 2019-08-07 2019-11-29 南昌大学 神经节苷脂gm3在制备治疗动脉粥样硬化药物中的应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4476119A (en) * 1981-08-04 1984-10-09 Fidia S.P.A. Method for preparing ganglioside derivatives and use thereof in pharmaceutical compositions
IT1199116B (it) * 1984-07-03 1988-12-30 Fidia Farmaceutici Derivati di gangliosidi
JP3845121B2 (ja) * 1994-09-30 2006-11-15 雪印乳業株式会社 ガングリオシドの製造法
US5977329A (en) * 1996-02-16 1999-11-02 Ludwig Institute For Cancer Research Methods of synthesizing GM3

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
See references of WO0035932A1 *

Also Published As

Publication number Publication date
WO2000035932A1 (en) 2000-06-22
IT1302530B1 (it) 2000-09-05
ITPD980293A1 (it) 2000-06-16
CA2355106A1 (en) 2000-06-22
AU1979800A (en) 2000-07-03

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