EP0946556A4 - Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine - Google Patents
Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleineInfo
- Publication number
- EP0946556A4 EP0946556A4 EP97954102A EP97954102A EP0946556A4 EP 0946556 A4 EP0946556 A4 EP 0946556A4 EP 97954102 A EP97954102 A EP 97954102A EP 97954102 A EP97954102 A EP 97954102A EP 0946556 A4 EP0946556 A4 EP 0946556A4
- Authority
- EP
- European Patent Office
- Prior art keywords
- hydrofuroquinoline
- libraries
- preparing
- combinatorial process
- combinatorial
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C40—COMBINATORIAL TECHNOLOGY
- C40B—COMBINATORIAL CHEMISTRY; LIBRARIES, e.g. CHEMICAL LIBRARIES
- C40B40/00—Libraries per se, e.g. arrays, mixtures
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US3366596P | 1996-12-18 | 1996-12-18 | |
US33665P | 1996-12-18 | ||
PCT/US1997/022870 WO1998027093A1 (fr) | 1996-12-18 | 1997-12-15 | Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine |
Publications (2)
Publication Number | Publication Date |
---|---|
EP0946556A1 EP0946556A1 (fr) | 1999-10-06 |
EP0946556A4 true EP0946556A4 (fr) | 2001-07-04 |
Family
ID=21871728
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EP97954102A Withdrawn EP0946556A4 (fr) | 1996-12-18 | 1997-12-15 | Methode combinatoire aux fins de l'elaboration de banques de tetrahydroquinoleine |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0946556A4 (fr) |
JP (1) | JP2001508050A (fr) |
AU (1) | AU5797098A (fr) |
CA (1) | CA2273884A1 (fr) |
WO (1) | WO1998027093A1 (fr) |
Families Citing this family (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US7250423B2 (en) * | 2001-09-24 | 2007-07-31 | Chao-Jun Li | Methods for synthesizing heterocycles and therapeutic use of the heterocycles for cancers |
DE10236910A1 (de) * | 2002-08-12 | 2004-03-11 | Grünenthal GmbH | Substituierte 1,2,3,4-Tetrahydrochinolinderivate |
WO2005016255A2 (fr) * | 2003-07-16 | 2005-02-24 | Ligand Pharmaceuticals Incorporated | Tetrahydroquinolines a substitution, acides phenylacetiques et benzoiques, comme composes modulateurs de recepteur du facteur nucleaire d'hepatocyte 4$g(a) (hnf-4$g(a) ) |
DE102004031656A1 (de) * | 2004-06-30 | 2006-01-19 | Merck Patent Gmbh | Tetrahydrochinoline |
DE102005027170A1 (de) * | 2005-06-13 | 2006-12-14 | Merck Patent Gmbh | Substituierte Tetrahydrochinoline |
EP2647638A1 (fr) * | 2012-04-02 | 2013-10-09 | Almirall, S.A. | Composés tricycliques substitués présentant une activité vis-à-vis des récepteurs ep1 |
Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3632852A (en) * | 1969-03-17 | 1972-01-04 | Parke Davis & Co | Hexahydrobenzofurofuro(3 2-c) quinoline compounds |
WO1994008051A1 (fr) * | 1992-10-01 | 1994-04-14 | The Trustees Of Columbia University In The City Of New York | Banques chimiques combinatoires complexes codees avec des etiquettes |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2650226A (en) * | 1950-05-24 | 1953-08-25 | Schenley Ind Inc | Furo and thieno quinaldines and process for making same |
US2650229A (en) * | 1950-05-27 | 1953-08-25 | Schenley Ind Inc | Derivatives of 2:3-dihydro-4-methyltfuro(3:2-c) quinoline and preparation thereof |
US2650227A (en) * | 1950-05-27 | 1953-08-25 | Schenley Ind Inc | Derivatives of 2:3-dihydro-4-methylfuro (3:2-c) quinoline and preparation thereof |
US3631050A (en) * | 1968-11-13 | 1971-12-28 | Parke Davis & Co | Hexahydro-9b-methylfuro(3 2-c) quinoline compounds |
-
1997
- 1997-12-15 AU AU57970/98A patent/AU5797098A/en not_active Abandoned
- 1997-12-15 JP JP52785698A patent/JP2001508050A/ja active Pending
- 1997-12-15 EP EP97954102A patent/EP0946556A4/fr not_active Withdrawn
- 1997-12-15 WO PCT/US1997/022870 patent/WO1998027093A1/fr not_active Application Discontinuation
- 1997-12-15 CA CA002273884A patent/CA2273884A1/fr not_active Abandoned
Patent Citations (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3632852A (en) * | 1969-03-17 | 1972-01-04 | Parke Davis & Co | Hexahydrobenzofurofuro(3 2-c) quinoline compounds |
WO1994008051A1 (fr) * | 1992-10-01 | 1994-04-14 | The Trustees Of Columbia University In The City Of New York | Banques chimiques combinatoires complexes codees avec des etiquettes |
Non-Patent Citations (8)
Title |
---|
BORRIONE E ET AL: "SYNTHESIS AND CYCLOADDITION REACTIONS OF ETHYL GLYOXYLATE IMINES. SYNTHESIS OF SUBSTITUTED FURO-U3,2-CQUINOLINES AND 7H-INDENO U2,1-CQUINOLINES", JOURNAL OF HETEROCYCLIC CHEMISTRY,US,HETEROCORPORATION. PROVO, vol. 25, 1 November 1988 (1988-11-01), pages 1831 - 1835, XP000670083, ISSN: 0022-152X * |
ELSLAGER E. F., WORTH D. F.: "1,4-Cycloaddition Reactions. I.", J. HETEROCYCL. CHEM, vol. 6, 1969, pages 597 - 598, XP000994873 * |
LUCCHINI V., PRATO M., SCORRANO G., STIVANELLO M., VALLE G.: "Acid-catalysed Addition of N-Aryl Imines to Dihydrofuran.", J. CHEM. SOC. PERKIN TRANS., vol. 2, 1992, pages 259 - 266, XP000994883 * |
MIKHAILOV,B.M. ET AL.: "Reaction of Dihydrosylvan with Schiff Bases", BULL. ACAD. SCI. USSR DIV. CHEM. SCI. (ENGL.TRANSL.), 1964, pages 1597 - 1599, XP000995275 * |
PERRICONE S. C., WORTH F. D., ELSLAGER E. F.: "1,4-Cycloaddition Reactions. III.", J. HETEROCYCL. CHEM., vol. 7, 1970, pages 537 - 542, XP000995005 * |
See also references of WO9827093A1 * |
WORTH F. D., PERRICONE S. C., ELSLAGER E. F.: "1,4-Cycloaddition Reactions. IV.", J. HETEROCYCL. CHEM., vol. 7, 1970, pages 1353 - 1356, XP000995219 * |
WORTH,D.F. ET AL.: "1,4-Cycloaddition Reactions. V.", J. HETEROCYCL. CHEM., vol. 11, 1974, pages 69 - 70, XP000994879 * |
Also Published As
Publication number | Publication date |
---|---|
JP2001508050A (ja) | 2001-06-19 |
EP0946556A1 (fr) | 1999-10-06 |
CA2273884A1 (fr) | 1998-06-25 |
AU5797098A (en) | 1998-07-15 |
WO1998027093A1 (fr) | 1998-06-25 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
PUAI | Public reference made under article 153(3) epc to a published international application that has entered the european phase |
Free format text: ORIGINAL CODE: 0009012 |
|
17P | Request for examination filed |
Effective date: 19990603 |
|
AK | Designated contracting states |
Kind code of ref document: A1 Designated state(s): AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE |
|
RIC1 | Information provided on ipc code assigned before grant |
Free format text: 7C 07D 491/04 A, 7C 07D 491/04 J, 7C 07D 307:00 J, 7C 07D 221:00 J |
|
A4 | Supplementary search report drawn up and despatched |
Effective date: 20010521 |
|
AK | Designated contracting states |
Kind code of ref document: A4 Designated state(s): AT BE CH DE DK ES FI FR GB GR IE IT LI NL PT SE |
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STAA | Information on the status of an ep patent application or granted ep patent |
Free format text: STATUS: THE APPLICATION IS DEEMED TO BE WITHDRAWN |
|
18D | Application deemed to be withdrawn |
Effective date: 20010809 |