ECSP993293A - Inhibidores de proteasas viii - Google Patents
Inhibidores de proteasas viiiInfo
- Publication number
- ECSP993293A ECSP993293A ECSP993293A ECSP993293A EC SP993293 A ECSP993293 A EC SP993293A EC SP993293 A ECSP993293 A EC SP993293A EC SP993293 A ECSP993293 A EC SP993293A
- Authority
- EC
- Ecuador
- Prior art keywords
- excessive
- compounds
- disease
- protease inhibitors
- cartilage
- Prior art date
Links
- 229940042399 direct acting antivirals protease inhibitors Drugs 0.000 title abstract 2
- 239000000137 peptide hydrolase inhibitor Substances 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 4
- 206010065687 Bone loss Diseases 0.000 abstract 2
- 210000000845 cartilage Anatomy 0.000 abstract 2
- 230000015556 catabolic process Effects 0.000 abstract 2
- 238000006731 degradation reaction Methods 0.000 abstract 2
- 239000011159 matrix material Substances 0.000 abstract 2
- QTLLOLTVQMFWDZ-UHFFFAOYSA-N 4-aminoazepan-3-one Chemical compound NC1CCCNCC1=O QTLLOLTVQMFWDZ-UHFFFAOYSA-N 0.000 abstract 1
- 208000037147 Hypercalcaemia Diseases 0.000 abstract 1
- 208000030136 Marchiafava-Bignami Disease Diseases 0.000 abstract 1
- 208000029725 Metabolic bone disease Diseases 0.000 abstract 1
- 208000010191 Osteitis Deformans Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 208000027868 Paget disease Diseases 0.000 abstract 1
- 102000035195 Peptidases Human genes 0.000 abstract 1
- 108091005804 Peptidases Proteins 0.000 abstract 1
- 239000004365 Protease Substances 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- -1 captesin K Substances 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000024693 gingival disease Diseases 0.000 abstract 1
- 208000007565 gingivitis Diseases 0.000 abstract 1
- 150000004677 hydrates Chemical class 0.000 abstract 1
- 230000000148 hypercalcaemia Effects 0.000 abstract 1
- 208000030915 hypercalcemia disease Diseases 0.000 abstract 1
- 230000002401 inhibitory effect Effects 0.000 abstract 1
- 230000003211 malignant effect Effects 0.000 abstract 1
- 208000027202 mammary Paget disease Diseases 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 201000008482 osteoarthritis Diseases 0.000 abstract 1
- 201000001245 periodontitis Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona inhibidores de proteasa de 4-amino-azepan-3-ona y sus sales, hidratos o solvatos de los mismos aceptables farmacéuticamente, que inhiben proteasas, incluyendo la captesina K, composiciones farmacéuticas de tales compuesto, nuevos compuestos intermedios de los compuestos de este tipo, y métodos para tratar enfermedades de pérdida ósea excesiva o degradación excesiva de cartílago o matriz, con inclusión de osteoporosis; enfermedad gingival con inclusión de gingivitis y periodontitis; artritis, más específicamente, osteoartritis y artritis reumatoide; enfermedad de Paget; hipercalcemia de carácetr maligno; y enfermedad metabólica ósea, que comprende inhibir dicha pérdida ósea o degradación excesiva de cartílago o matriz por administración de un compuesto de la presente invención a un paciente que se encuentra en necesidad de ello.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993293 ECSP993293A (es) | 1999-12-23 | 1999-12-23 | Inhibidores de proteasas viii |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP993293 ECSP993293A (es) | 1999-12-23 | 1999-12-23 | Inhibidores de proteasas viii |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP993293A true ECSP993293A (es) | 2000-05-25 |
Family
ID=42044284
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP993293 ECSP993293A (es) | 1999-12-23 | 1999-12-23 | Inhibidores de proteasas viii |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP993293A (es) |
-
1999
- 1999-12-23 EC ECSP993293 patent/ECSP993293A/es unknown
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