ECSP19015143A - Compuestos de tiazolo-piridina sustituida como inhibidores de malt1 - Google Patents

Compuestos de tiazolo-piridina sustituida como inhibidores de malt1

Info

Publication number
ECSP19015143A
ECSP19015143A ECSENADI201915143A ECDI201915143A ECSP19015143A EC SP19015143 A ECSP19015143 A EC SP19015143A EC SENADI201915143 A ECSENADI201915143 A EC SENADI201915143A EC DI201915143 A ECDI201915143 A EC DI201915143A EC SP19015143 A ECSP19015143 A EC SP19015143A
Authority
EC
Ecuador
Prior art keywords
thiazolo
pyridine compounds
compounds substituted
malt1 inhibitors
malt1
Prior art date
Application number
ECSENADI201915143A
Other languages
English (en)
Inventor
Venkata Palle
Vinod Vyavahare
Neelima Sinha
Gokul Deshmukh
Arun Jagdale
Nageswara Irlapati
Kiran Kulkarni
Gagan Kukreja
Rajender Kamboj
Original Assignee
Lupin Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lupin Ltd filed Critical Lupin Ltd
Publication of ECSP19015143A publication Critical patent/ECSP19015143A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders

Abstract

Por favor, ver archivo adjunto.
ECSENADI201915143A 2016-07-29 2019-02-28 Compuestos de tiazolo-piridina sustituida como inhibidores de malt1 ECSP19015143A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN201621026107 2016-07-29
IN201621043859 2016-12-22
IN201721009450 2017-03-17

Publications (1)

Publication Number Publication Date
ECSP19015143A true ECSP19015143A (es) 2019-05-31

Family

ID=65656144

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSENADI201915143A ECSP19015143A (es) 2016-07-29 2019-02-28 Compuestos de tiazolo-piridina sustituida como inhibidores de malt1

Country Status (9)

Country Link
US (1) US20210052556A1 (es)
EP (2) EP3736277A1 (es)
BR (1) BR112019001824A2 (es)
CO (1) CO2019001967A2 (es)
CR (1) CR20190110A (es)
EC (1) ECSP19015143A (es)
IL (1) IL264465B (es)
MA (2) MA45787A (es)
RU (1) RU2021113671A (es)

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4235871A (en) 1978-02-24 1980-11-25 Papahadjopoulos Demetrios P Method of encapsulating biologically active materials in lipid vesicles
US4501728A (en) 1983-01-06 1985-02-26 Technology Unlimited, Inc. Masking of liposomes from RES recognition
US5019369A (en) 1984-10-22 1991-05-28 Vestar, Inc. Method of targeting tumors in humans
US4837028A (en) 1986-12-24 1989-06-06 Liposome Technology, Inc. Liposomes with enhanced circulation time
WO2008146259A2 (en) 2007-06-01 2008-12-04 University Of Lausanne Malt1 specific cleavage in assay and screening method
US8309523B2 (en) 2007-11-21 2012-11-13 Vib Vzw Inhibitors of MALT1 proteolytic activity and uses thereof
US9504692B2 (en) 2011-08-02 2016-11-29 Helmholtz Zentrum Munchen, Deutsches Forschungszentrum Fur Gesundheit Und Umwelt (Gmbh) Selective inhibition of MALT1 protease by phenothiazine derivatives
WO2013053765A1 (en) 2011-10-11 2013-04-18 Proyecto De Biomedicina Cima, S.L. A non-human animal model of mucosa-associated lymphoid tissue (malt) lymphoma
MX2015005744A (es) 2012-11-09 2016-02-10 Univ Cornell Inhibidores de malti de molecula pequeña.
WO2014086478A1 (en) 2012-12-03 2014-06-12 Helmholtz Zentrum München - Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) Inhibitors of malt1 protease
US9718811B2 (en) 2013-06-26 2017-08-01 Helmholtz Zentrum München—Deutsches Forschungszentrum für Gesundheit und Umwelt (GmbH) (S)-enantiomer of mepazine
EP3097124B1 (en) 2014-01-21 2018-12-19 Helmholtz Zentrum München Means and methods for detecting activated malt1
CU24393B1 (es) 2014-05-28 2019-04-04 Novartis Ag Nuevos derivados de pirazolo pirimidina y su uso como inhibidores de malt1
DE102015210224A1 (de) 2015-06-02 2016-12-08 Universitätsklinikum Hamburg-Eppendorf Neuer wirkstoff zur behandlung von krebs
WO2017040304A1 (en) 2015-08-28 2017-03-09 Cornell University Malt1 inhibitors and uses thereof
WO2017057695A1 (ja) 2015-09-30 2017-04-06 東レ株式会社 ジフェニルピラゾール誘導体及びその医薬用途
BR112018009511A2 (pt) 2015-11-13 2018-11-06 Novartis Ag derivados de pirazolo pirimidina
WO2018165385A1 (en) * 2017-03-08 2018-09-13 Cornell University Inhibitors of malt1 and uses thereof

Also Published As

Publication number Publication date
BR112019001824A2 (pt) 2019-05-07
RU2021113671A (ru) 2021-07-08
CO2019001967A2 (es) 2019-05-31
EP3490995A1 (en) 2019-06-05
CR20190110A (es) 2019-08-27
EP3736277A1 (en) 2020-11-11
US20210052556A1 (en) 2021-02-25
IL264465B (en) 2022-02-01
IL264465A (en) 2019-02-28
MA53299A (fr) 2022-02-23
MA45787A (fr) 2019-06-05

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