ECSP12012352A - Agente terapéutico de liberación sostenida para la hipertensión y la disfunción renal - Google Patents

Agente terapéutico de liberación sostenida para la hipertensión y la disfunción renal

Info

Publication number
ECSP12012352A
ECSP12012352A ECSP12012352A ECSP12012352A EC SP12012352 A ECSP12012352 A EC SP12012352A EC SP12012352 A ECSP12012352 A EC SP12012352A EC SP12012352 A ECSP12012352 A EC SP12012352A
Authority
EC
Ecuador
Prior art keywords
hypertension
renal dysfunction
therapeutic agent
sustained release
release therapeutic
Prior art date
Application number
Other languages
English (en)
Inventor
Takashi Shirakura
Mizuho Tamura
Yoshimasa Takahashi
Ippei Kuwahara
Original Assignee
Teijin Pharma Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45371556&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP12012352(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Teijin Pharma Ltd filed Critical Teijin Pharma Ltd
Publication of ECSP12012352A publication Critical patent/ECSP12012352A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/06Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/06Preparations for care of the skin for countering cellulitis

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La presente invención da a conocer un agente terapéutico o preventivo para la hipertensión o la presión sanguínea alta normal, y para la disfunción renal, que es más eficaz que las drogas existentes.Más específicamente, la presente invención da a conocer una composición farmacéutica de liberación sostenida para el tratamiento o prevención de la hipertensión o la presión sanguínea alta normal, y para la disfunción renal, que comprende, como ingrediente activo, un compuesto de 2-feniltiazol representado por la siguiente fórmula (I)Fórmula química 1 (I)o una sal farmacéuticamente aceptable del mismo.
ECSP12012352 2010-06-25 2012-12-20 Agente terapéutico de liberación sostenida para la hipertensión y la disfunción renal ECSP12012352A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP2010145056 2010-06-25

Publications (1)

Publication Number Publication Date
ECSP12012352A true ECSP12012352A (es) 2013-02-28

Family

ID=45371556

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP12012352 ECSP12012352A (es) 2010-06-25 2012-12-20 Agente terapéutico de liberación sostenida para la hipertensión y la disfunción renal

Country Status (25)

Country Link
US (1) US20130109726A1 (es)
EP (1) EP2586442A4 (es)
JP (1) JPWO2011162390A1 (es)
KR (1) KR20130088755A (es)
CN (1) CN102958521A (es)
AR (1) AR082022A1 (es)
AU (1) AU2011270133B2 (es)
BR (1) BR112012032543A2 (es)
CA (1) CA2803163A1 (es)
CL (1) CL2012003661A1 (es)
CO (1) CO6660504A2 (es)
EC (1) ECSP12012352A (es)
MA (1) MA34328B1 (es)
MX (1) MX2012015040A (es)
MY (1) MY160963A (es)
NZ (1) NZ605516A (es)
PE (1) PE20130241A1 (es)
RU (1) RU2013103366A (es)
SG (1) SG186798A1 (es)
TN (1) TN2012000568A1 (es)
TW (1) TW201215389A (es)
UA (1) UA107716C2 (es)
UY (1) UY33468A (es)
WO (1) WO2011162390A1 (es)
ZA (1) ZA201209388B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA112632C2 (uk) 2010-06-16 2016-10-10 Такеда Фармасьютикалз Ю.Ес.Ей., Інк. Дозована форма з модифікованим вивільненням фебуксостату (варіанти)
KR101797936B1 (ko) 2010-09-10 2017-11-15 다케다 파마슈티칼스 유에스에이, 인코포레이티드 테오필린과 페북소스타트의 병용 치료 방법
MX2014008484A (es) * 2012-01-27 2014-10-14 Teijin Pharma Ltd Agente terapeutico para la diabetes mellitus.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1992009279A1 (en) 1990-11-30 1992-06-11 Teijin Limited 2-arylthiazole derivative and pharmaceutical composition containing the same
WO2003013543A1 (en) * 2001-08-08 2003-02-20 Genomed, Llc Treatment or prevention of acute renal failure
CA2617248C (en) * 2005-08-03 2015-09-29 Tap Pharmaceutical Products, Inc. Methods for treating hypertension
US9028867B2 (en) * 2005-08-18 2015-05-12 Teijin Pharma Limited Formulation having accurate dose-dividing function
BRPI0718611A2 (pt) * 2006-11-13 2014-02-25 Takeda Pharmaceuticals North America Inc Métodos para preservar a função renal utilizando inibidores da xantina oxidoredutase.
CN101658505A (zh) * 2009-09-29 2010-03-03 北京华禧联合科技发展有限公司 非布索坦的缓释制剂及其制备方法
UA112632C2 (uk) * 2010-06-16 2016-10-10 Такеда Фармасьютикалз Ю.Ес.Ей., Інк. Дозована форма з модифікованим вивільненням фебуксостату (варіанти)

Also Published As

Publication number Publication date
ZA201209388B (en) 2013-08-28
CO6660504A2 (es) 2013-04-30
MY160963A (en) 2017-03-31
US20130109726A1 (en) 2013-05-02
AR082022A1 (es) 2012-11-07
PE20130241A1 (es) 2013-03-04
KR20130088755A (ko) 2013-08-08
CA2803163A1 (en) 2011-12-29
AU2011270133A1 (en) 2013-01-10
EP2586442A4 (en) 2014-01-01
JPWO2011162390A1 (ja) 2013-08-22
AU2011270133B2 (en) 2014-03-20
SG186798A1 (en) 2013-02-28
RU2013103366A (ru) 2014-07-27
BR112012032543A2 (pt) 2016-11-22
MX2012015040A (es) 2013-02-07
CN102958521A (zh) 2013-03-06
NZ605516A (en) 2015-02-27
CL2012003661A1 (es) 2013-04-01
MA34328B1 (fr) 2013-06-01
TN2012000568A1 (en) 2014-04-01
UY33468A (es) 2012-01-31
EP2586442A1 (en) 2013-05-01
TW201215389A (en) 2012-04-16
WO2011162390A1 (ja) 2011-12-29
UA107716C2 (ru) 2015-02-10

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