ECSP099789A - Disolución directa del docetaxel en un disolvente en polisorbato 80 - Google Patents

Disolución directa del docetaxel en un disolvente en polisorbato 80

Info

Publication number
ECSP099789A
ECSP099789A EC2009009789A ECSP099789A ECSP099789A EC SP099789 A ECSP099789 A EC SP099789A EC 2009009789 A EC2009009789 A EC 2009009789A EC SP099789 A ECSP099789 A EC SP099789A EC SP099789 A ECSP099789 A EC SP099789A
Authority
EC
Ecuador
Prior art keywords
solvent
docetaxel
polisorbate
direct dissolution
dissolution
Prior art date
Application number
EC2009009789A
Other languages
English (en)
Inventor
Eric Didier
Jean Rene Authelin
Elie Fouque
Mostafa Nakach
Original Assignee
Aventis Pharma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39048780&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=ECSP099789(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aventis Pharma Sa filed Critical Aventis Pharma Sa
Publication of ECSP099789A publication Critical patent/ECSP099789A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Epoxy Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
  • Processes Of Treating Macromolecular Substances (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La invención se refiere a la solubilización del docetaxel en un disolvente orgánico, a su mezcla con polisorbato 80 y a la evaporación del disolvente.
EC2009009789A 2007-06-08 2009-12-08 Disolución directa del docetaxel en un disolvente en polisorbato 80 ECSP099789A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0704095A FR2917088B1 (fr) 2007-06-08 2007-06-08 Dissolution directe du docetaxel dans un solvant dans le polysorbate 80
PCT/FR2008/000766 WO2009004188A2 (fr) 2007-06-08 2008-06-06 Dissolution directe du docetaxel dans un solvant dans le poly sorbate 80

Publications (1)

Publication Number Publication Date
ECSP099789A true ECSP099789A (es) 2010-01-29

Family

ID=39048780

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2009009789A ECSP099789A (es) 2007-06-08 2009-12-08 Disolución directa del docetaxel en un disolvente en polisorbato 80

Country Status (32)

Country Link
US (1) US20100197776A1 (es)
EP (1) EP2155189A2 (es)
JP (1) JP2010529094A (es)
KR (1) KR20100022033A (es)
CN (2) CN102908309A (es)
AR (1) AR066889A1 (es)
AU (1) AU2008270141A1 (es)
BR (1) BRPI0812438A2 (es)
CA (1) CA2689466A1 (es)
CL (1) CL2008001650A1 (es)
CO (1) CO6260063A2 (es)
CR (1) CR11144A (es)
DO (1) DOP2009000249A (es)
EA (1) EA200971137A1 (es)
EC (1) ECSP099789A (es)
FR (1) FR2917088B1 (es)
GT (1) GT200900306A (es)
HN (1) HN2009003363A (es)
IL (1) IL202517A0 (es)
MA (1) MA31671B1 (es)
MX (1) MX2009013216A (es)
MY (1) MY151417A (es)
NI (1) NI200900209A (es)
NZ (1) NZ581634A (es)
PA (1) PA8783101A1 (es)
SV (1) SV2009003428A (es)
TN (1) TN2009000396A1 (es)
TW (1) TW200916095A (es)
UA (1) UA99828C2 (es)
UY (1) UY31129A1 (es)
WO (1) WO2009004188A2 (es)
ZA (1) ZA200908662B (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102970990A (zh) 2010-05-03 2013-03-13 帝国制药美国公司 非水性紫杉烷前-乳剂制剂以及制备和使用该制剂的方法
JO3685B1 (ar) 2012-10-01 2020-08-27 Teikoku Pharma Usa Inc صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2678833B1 (fr) * 1991-07-08 1995-04-07 Rhone Poulenc Rorer Sa Nouvelles compositions pharmaceutiques a base de derives de la classe des taxanes.
US6040330A (en) * 1999-01-08 2000-03-21 Bionumerik Pharmaceuticals, Inc. Pharmaceutical formulations of taxanes
GB9920548D0 (en) * 1999-08-31 1999-11-03 Rhone Poulenc Rorer Sa Treatment of hepatocellular carcinoma
US20020041898A1 (en) * 2000-01-05 2002-04-11 Unger Evan C. Novel targeted delivery systems for bioactive agents
US6838569B2 (en) * 2002-12-16 2005-01-04 Dabur India Limited Process for preparation of paclitaxel trihydrate and docetaxel trihydrate
EP1815869A4 (en) * 2004-11-24 2011-04-06 Nanocarrier Co Ltd PROCESS FOR CHANGING THE MORPHOLOGY OF BLOCK COPOLYMERS
BRPI0600194A (pt) * 2006-01-30 2007-10-23 Quiral Quimica Do Brasil S A composições farmacêuticas contendo docetaxel e um inibidor de degradação e processo de obtenção das mesmas

Also Published As

Publication number Publication date
AR066889A1 (es) 2009-09-16
GT200900306A (es) 2011-06-17
NZ581634A (en) 2012-05-25
KR20100022033A (ko) 2010-02-26
EA200971137A1 (ru) 2010-04-30
JP2010529094A (ja) 2010-08-26
UY31129A1 (es) 2009-01-30
UA99828C2 (ru) 2012-10-10
MY151417A (en) 2014-05-30
EP2155189A2 (fr) 2010-02-24
CO6260063A2 (es) 2011-03-22
TW200916095A (en) 2009-04-16
CN102908309A (zh) 2013-02-06
BRPI0812438A2 (pt) 2014-12-02
SV2009003428A (es) 2010-02-05
ZA200908662B (en) 2011-04-28
HN2009003363A (es) 2013-09-18
DOP2009000249A (es) 2009-11-30
AU2008270141A1 (en) 2009-01-08
FR2917088A1 (fr) 2008-12-12
IL202517A0 (en) 2010-06-30
MX2009013216A (es) 2010-01-25
PA8783101A1 (es) 2009-01-23
CA2689466A1 (fr) 2009-01-08
US20100197776A1 (en) 2010-08-05
NI200900209A (es) 2010-10-04
WO2009004188A3 (fr) 2009-03-26
CR11144A (es) 2010-03-23
TN2009000396A1 (fr) 2010-12-31
MA31671B1 (fr) 2010-09-01
CN101677986A (zh) 2010-03-24
WO2009004188A2 (fr) 2009-01-08
CL2008001650A1 (es) 2009-10-23
FR2917088B1 (fr) 2009-09-04

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