EA200971137A1 - Прямое растворение доцетаксела в растворителе в полисорбате 80 - Google Patents

Прямое растворение доцетаксела в растворителе в полисорбате 80

Info

Publication number
EA200971137A1
EA200971137A1 EA200971137A EA200971137A EA200971137A1 EA 200971137 A1 EA200971137 A1 EA 200971137A1 EA 200971137 A EA200971137 A EA 200971137A EA 200971137 A EA200971137 A EA 200971137A EA 200971137 A1 EA200971137 A1 EA 200971137A1
Authority
EA
Eurasian Patent Office
Prior art keywords
solvent
docetaxel
polysorbate
direct dissolution
dissolution
Prior art date
Application number
EA200971137A
Other languages
English (en)
Inventor
Жан-Рене Отелен
Эрик Дидье
Эли Фук
Мостафа Накаш
Original Assignee
Авентис Фарма С.А.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39048780&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA200971137(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Авентис Фарма С.А. filed Critical Авентис Фарма С.А.
Publication of EA200971137A1 publication Critical patent/EA200971137A1/ru

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/337Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D305/00Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems

Abstract

Изобретение относится к растворению доцетаксела в органическом растворителе, его смешиванию с полисорбатом 80 и выпариванию растворителя.
EA200971137A 2007-06-08 2008-06-06 Прямое растворение доцетаксела в растворителе в полисорбате 80 EA200971137A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0704095A FR2917088B1 (fr) 2007-06-08 2007-06-08 Dissolution directe du docetaxel dans un solvant dans le polysorbate 80
PCT/FR2008/000766 WO2009004188A2 (fr) 2007-06-08 2008-06-06 Dissolution directe du docetaxel dans un solvant dans le poly sorbate 80

Publications (1)

Publication Number Publication Date
EA200971137A1 true EA200971137A1 (ru) 2010-04-30

Family

ID=39048780

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200971137A EA200971137A1 (ru) 2007-06-08 2008-06-06 Прямое растворение доцетаксела в растворителе в полисорбате 80

Country Status (32)

Country Link
US (1) US20100197776A1 (ru)
EP (1) EP2155189A2 (ru)
JP (1) JP2010529094A (ru)
KR (1) KR20100022033A (ru)
CN (2) CN101677986A (ru)
AR (1) AR066889A1 (ru)
AU (1) AU2008270141A1 (ru)
BR (1) BRPI0812438A2 (ru)
CA (1) CA2689466A1 (ru)
CL (1) CL2008001650A1 (ru)
CO (1) CO6260063A2 (ru)
CR (1) CR11144A (ru)
DO (1) DOP2009000249A (ru)
EA (1) EA200971137A1 (ru)
EC (1) ECSP099789A (ru)
FR (1) FR2917088B1 (ru)
GT (1) GT200900306A (ru)
HN (1) HN2009003363A (ru)
IL (1) IL202517A0 (ru)
MA (1) MA31671B1 (ru)
MX (1) MX2009013216A (ru)
MY (1) MY151417A (ru)
NI (1) NI200900209A (ru)
NZ (1) NZ581634A (ru)
PA (1) PA8783101A1 (ru)
SV (1) SV2009003428A (ru)
TN (1) TN2009000396A1 (ru)
TW (1) TW200916095A (ru)
UA (1) UA99828C2 (ru)
UY (1) UY31129A1 (ru)
WO (1) WO2009004188A2 (ru)
ZA (1) ZA200908662B (ru)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR101752944B1 (ko) 2010-05-03 2017-07-03 테이코쿠 팔마 유에스에이, 인코포레이티드 비수성의 탁산 프로에멀젼 제제, 및 그의 제조 및 사용 방법
JO3685B1 (ar) * 2012-10-01 2020-08-27 Teikoku Pharma Usa Inc صيغ التشتيت الجسيمي للتاكسين غير المائي وطرق استخدامها

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2678833B1 (fr) * 1991-07-08 1995-04-07 Rhone Poulenc Rorer Sa Nouvelles compositions pharmaceutiques a base de derives de la classe des taxanes.
US6040330A (en) * 1999-01-08 2000-03-21 Bionumerik Pharmaceuticals, Inc. Pharmaceutical formulations of taxanes
GB9920548D0 (en) * 1999-08-31 1999-11-03 Rhone Poulenc Rorer Sa Treatment of hepatocellular carcinoma
US20020041898A1 (en) * 2000-01-05 2002-04-11 Unger Evan C. Novel targeted delivery systems for bioactive agents
US6838569B2 (en) * 2002-12-16 2005-01-04 Dabur India Limited Process for preparation of paclitaxel trihydrate and docetaxel trihydrate
WO2006057429A1 (ja) * 2004-11-24 2006-06-01 Nanocarrier Co., Ltd. ブロックコポリマーのモーフォロジ-の変化方法
BRPI0600194A (pt) * 2006-01-30 2007-10-23 Quiral Quimica Do Brasil S A composições farmacêuticas contendo docetaxel e um inibidor de degradação e processo de obtenção das mesmas

Also Published As

Publication number Publication date
BRPI0812438A2 (pt) 2014-12-02
FR2917088B1 (fr) 2009-09-04
CN101677986A (zh) 2010-03-24
PA8783101A1 (es) 2009-01-23
NZ581634A (en) 2012-05-25
CR11144A (es) 2010-03-23
ECSP099789A (es) 2010-01-29
CO6260063A2 (es) 2011-03-22
CL2008001650A1 (es) 2009-10-23
MY151417A (en) 2014-05-30
MA31671B1 (fr) 2010-09-01
FR2917088A1 (fr) 2008-12-12
US20100197776A1 (en) 2010-08-05
UY31129A1 (es) 2009-01-30
CN102908309A (zh) 2013-02-06
ZA200908662B (en) 2011-04-28
TW200916095A (en) 2009-04-16
TN2009000396A1 (fr) 2010-12-31
MX2009013216A (es) 2010-01-25
KR20100022033A (ko) 2010-02-26
GT200900306A (es) 2011-06-17
EP2155189A2 (fr) 2010-02-24
IL202517A0 (en) 2010-06-30
AR066889A1 (es) 2009-09-16
JP2010529094A (ja) 2010-08-26
UA99828C2 (ru) 2012-10-10
DOP2009000249A (es) 2009-11-30
HN2009003363A (es) 2013-09-18
AU2008270141A1 (en) 2009-01-08
CA2689466A1 (fr) 2009-01-08
WO2009004188A2 (fr) 2009-01-08
SV2009003428A (es) 2010-02-05
NI200900209A (es) 2010-10-04
WO2009004188A3 (fr) 2009-03-26

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