ECSP099537A - METHODS FOR IMPROVED STABILITY OF STEROID DERIVATIVES - Google Patents
METHODS FOR IMPROVED STABILITY OF STEROID DERIVATIVESInfo
- Publication number
- ECSP099537A ECSP099537A EC2009009537A ECSP099537A ECSP099537A EC SP099537 A ECSP099537 A EC SP099537A EC 2009009537 A EC2009009537 A EC 2009009537A EC SP099537 A ECSP099537 A EC SP099537A EC SP099537 A ECSP099537 A EC SP099537A
- Authority
- EC
- Ecuador
- Prior art keywords
- improved stability
- methods
- steroid derivatives
- steroid
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C225/00—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones
- C07C225/22—Compounds containing amino groups and doubly—bound oxygen atoms bound to the same carbon skeleton, at least one of the doubly—bound oxygen atoms not being part of a —CHO group, e.g. amino ketones having amino groups bound to carbon atoms of six-membered aromatic rings of the carbon skeleton
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/136—Amines having aromatic rings, e.g. ketamine, nortriptyline having the amino group directly attached to the aromatic ring, e.g. benzeneamine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/04—Drugs for genital or sexual disorders; Contraceptives for inducing labour or abortion; Uterotonics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/36—Antigestagens
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C221/00—Preparation of compounds containing amino groups and doubly-bound oxygen atoms bound to the same carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
- C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
- C07J41/0077—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom
- C07J41/0083—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 substituted in position 11-beta by a carbon atom, further substituted by a group comprising at least one further carbon atom substituted in position 11-beta by an optionally substituted phenyl group not further condensed with other rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Reproductive Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Gynecology & Obstetrics (AREA)
- Pregnancy & Childbirth (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Se proveen composiciones con estabilidad mejorada que comprenden una sal farmacéuticamente aceptable de un compuesto relacionado con esteroides.Compositions with improved stability are provided comprising a pharmaceutically acceptable salt of a steroid related compound.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US88536307P | 2007-01-17 | 2007-01-17 |
Publications (1)
Publication Number | Publication Date |
---|---|
ECSP099537A true ECSP099537A (en) | 2009-08-28 |
Family
ID=39387140
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EC2009009537A ECSP099537A (en) | 2007-01-17 | 2009-07-23 | METHODS FOR IMPROVED STABILITY OF STEROID DERIVATIVES |
Country Status (16)
Country | Link |
---|---|
EP (1) | EP2125858A2 (en) |
JP (1) | JP2010516686A (en) |
KR (1) | KR20090105944A (en) |
CN (1) | CN101616926A (en) |
AR (1) | AR064947A1 (en) |
AU (1) | AU2008206599A1 (en) |
BR (1) | BRPI0806572A2 (en) |
CA (1) | CA2674440A1 (en) |
CL (1) | CL2008000138A1 (en) |
CR (1) | CR10924A (en) |
EA (1) | EA200970692A1 (en) |
EC (1) | ECSP099537A (en) |
IL (1) | IL199684A0 (en) |
MX (1) | MX2009007313A (en) |
TW (1) | TW200835503A (en) |
WO (1) | WO2008088935A2 (en) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TWI477276B (en) * | 2008-04-28 | 2015-03-21 | Repros Therapeutics Inc | Antiprogestin dosing regimens |
US8512745B2 (en) | 2008-12-08 | 2013-08-20 | Laboratoire Hra Pharma | Ulipristal acetate tablets |
HUP0900171A2 (en) * | 2009-03-20 | 2010-12-28 | Richter Gedeon Nyrt | Novel crystal form of 17-acetoxy-11-[4-(dimethyl-amino)-phenyl]-21-metoxy-19-norpregna-4,9-dien-3,20-dione and process for it's preparation |
HUP0900487A2 (en) * | 2009-08-05 | 2011-03-28 | Richter Gedeon Nyrt | Novel crystal polymorphic form of 17-acetoxy-11 -[4-(dimethylamino)phenyl]-21-methoxy-4,9-diene-3,20-dione and process for it's preparation |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA8231B (en) * | 1981-01-09 | 1982-11-24 | Roussel Uclaf | New 11 -substituted steroid derivatives, their preparation, their use as medicaments, the compositions containing them and the new intermediates thus obtained |
US6020328A (en) * | 1998-03-06 | 2000-02-01 | Research Triangle Institute | 20-keto-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties |
US8044223B2 (en) * | 2003-04-04 | 2011-10-25 | Bridge Organics Co. | Crystalline 19-norsteroids |
-
2008
- 2008-01-03 EP EP08713475A patent/EP2125858A2/en not_active Withdrawn
- 2008-01-03 JP JP2009546454A patent/JP2010516686A/en not_active Withdrawn
- 2008-01-03 BR BRPI0806572-1A patent/BRPI0806572A2/en not_active IP Right Cessation
- 2008-01-03 EA EA200970692A patent/EA200970692A1/en unknown
- 2008-01-03 CA CA002674440A patent/CA2674440A1/en not_active Abandoned
- 2008-01-03 MX MX2009007313A patent/MX2009007313A/en not_active Application Discontinuation
- 2008-01-03 CN CN200880002367A patent/CN101616926A/en active Pending
- 2008-01-03 AU AU2008206599A patent/AU2008206599A1/en not_active Abandoned
- 2008-01-03 WO PCT/US2008/050128 patent/WO2008088935A2/en active Application Filing
- 2008-01-03 KR KR1020097015532A patent/KR20090105944A/en not_active Application Discontinuation
- 2008-01-15 TW TW097101566A patent/TW200835503A/en unknown
- 2008-01-17 CL CL200800138A patent/CL2008000138A1/en unknown
- 2008-01-17 AR ARP080100217A patent/AR064947A1/en unknown
-
2009
- 2009-07-02 IL IL199684A patent/IL199684A0/en unknown
- 2009-07-14 CR CR10924A patent/CR10924A/en not_active Application Discontinuation
- 2009-07-23 EC EC2009009537A patent/ECSP099537A/en unknown
Also Published As
Publication number | Publication date |
---|---|
BRPI0806572A2 (en) | 2014-05-06 |
IL199684A0 (en) | 2010-04-15 |
CA2674440A1 (en) | 2008-07-24 |
CR10924A (en) | 2009-10-30 |
WO2008088935A3 (en) | 2009-03-05 |
EA200970692A1 (en) | 2010-02-26 |
EP2125858A2 (en) | 2009-12-02 |
CL2008000138A1 (en) | 2008-05-16 |
AU2008206599A1 (en) | 2008-07-24 |
JP2010516686A (en) | 2010-05-20 |
MX2009007313A (en) | 2009-07-15 |
KR20090105944A (en) | 2009-10-07 |
WO2008088935A2 (en) | 2008-07-24 |
TW200835503A (en) | 2008-09-01 |
AR064947A1 (en) | 2009-05-06 |
CN101616926A (en) | 2009-12-30 |
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