ECSP034692A - Antagonistas de receptores de histamina - Google Patents
Antagonistas de receptores de histaminaInfo
- Publication number
- ECSP034692A ECSP034692A EC2003004692A ECSP034692A ECSP034692A EC SP034692 A ECSP034692 A EC SP034692A EC 2003004692 A EC2003004692 A EC 2003004692A EC SP034692 A ECSP034692 A EC SP034692A EC SP034692 A ECSP034692 A EC SP034692A
- Authority
- EC
- Ecuador
- Prior art keywords
- histamine
- receptor
- receiver antagonists
- histamine receiver
- antagonists
- Prior art date
Links
- 239000005557 antagonist Substances 0.000 title abstract 2
- NTYJJOPFIAHURM-UHFFFAOYSA-N Histamine Chemical compound NCCC1=CN=CN1 NTYJJOPFIAHURM-UHFFFAOYSA-N 0.000 title 2
- 229960001340 histamine Drugs 0.000 title 1
- 102000004187 Histamine H4 receptors Human genes 0.000 abstract 2
- 108090000796 Histamine H4 receptors Proteins 0.000 abstract 2
- 229940124056 Histamine H1 receptor antagonist Drugs 0.000 abstract 1
- 102000004384 Histamine H3 receptors Human genes 0.000 abstract 1
- 108090000981 Histamine H3 receptors Proteins 0.000 abstract 1
- 102000000543 Histamine Receptors Human genes 0.000 abstract 1
- 108010002059 Histamine Receptors Proteins 0.000 abstract 1
- 239000000938 histamine H1 antagonist Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Otolaryngology (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona una combinación de (a) un antagonista de receptor H1 de histamina y (b) un antagonista que es al menos 10 veces más selectivo para el receptor H4 de histamina en comparación con el receptor H3 de histamina que es al menos 10 veces más selectivo para el receptor H4 de histamina en comparación con el receptor 3 de histamina; y sus composiciones y usos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0101223.6A GB0101223D0 (en) | 2001-01-17 | 2001-01-17 | Histamine receptor antagonists |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034692A true ECSP034692A (es) | 2003-08-29 |
Family
ID=9906993
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2003004692A ECSP034692A (es) | 2001-01-17 | 2003-07-17 | Antagonistas de receptores de histamina |
Country Status (31)
| Country | Link |
|---|---|
| EP (1) | EP1353657A1 (es) |
| JP (1) | JP2004517883A (es) |
| KR (1) | KR20030069216A (es) |
| CN (1) | CN1486178A (es) |
| AP (1) | AP2002002401A0 (es) |
| AR (1) | AR032101A1 (es) |
| BG (1) | BG107834A (es) |
| BR (1) | BR0206502A (es) |
| CA (1) | CA2435121A1 (es) |
| CR (1) | CR6983A (es) |
| CZ (1) | CZ20031853A3 (es) |
| DO (1) | DOP2002000325A (es) |
| EA (1) | EA200300537A1 (es) |
| EC (1) | ECSP034692A (es) |
| EE (1) | EE200300335A (es) |
| GB (1) | GB0101223D0 (es) |
| GT (1) | GT200200003A (es) |
| HU (1) | HUP0302767A2 (es) |
| IL (1) | IL156087A0 (es) |
| IS (1) | IS6818A (es) |
| MA (1) | MA26980A1 (es) |
| MX (1) | MXPA03006408A (es) |
| NO (1) | NO20033223D0 (es) |
| OA (1) | OA12440A (es) |
| PA (1) | PA8537101A1 (es) |
| PL (1) | PL362793A1 (es) |
| SK (1) | SK8572003A3 (es) |
| SV (1) | SV2003000849A (es) |
| TN (1) | TNSN02003A1 (es) |
| WO (1) | WO2002056871A2 (es) |
| ZA (1) | ZA200304180B (es) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20030133931A1 (en) * | 2001-12-21 | 2003-07-17 | Robin Thurmond | Use of histamine H4 receptor antagonist for the treatment of inflammatory responses |
| JP2006510590A (ja) * | 2002-09-06 | 2006-03-30 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | アレルギー及び喘息の処置のためのヒスタミンｈ４受容体モジュレーターの使用 |
| US20050090527A1 (en) * | 2003-01-28 | 2005-04-28 | Schering Corporation | Combination of H1, H3 and H4 receptor antagonists for treatment of allergic and non-allergic pulmonary inflammation, congestion and allergic rhinitis |
| US8236786B2 (en) | 2008-08-07 | 2012-08-07 | Pulmagen Therapeutics (Inflammation) Limited | Respiratory disease treatment |
| WO2013151982A1 (en) | 2012-04-03 | 2013-10-10 | Arena Pharmaceuticals, Inc. | Methods and compounds useful in treating pruritus, and methods for identifying such compounds |
| DK2858647T3 (en) | 2012-06-08 | 2018-08-20 | Sensorion | H4 RECEPTOR INHIBITORS FOR TINNITUS TREATMENT |
| CN119823227B (zh) * | 2025-01-14 | 2025-07-04 | 广州迪卡德营养科技有限公司 | 一种益生菌的制备方法及其在治疗过敏性鼻炎中的用途 |
-
2001
- 2001-01-17 GB GBGB0101223.6A patent/GB0101223D0/en not_active Ceased
-
2002
- 2002-01-10 SK SK857-2003A patent/SK8572003A3/sk unknown
- 2002-01-10 KR KR10-2003-7009493A patent/KR20030069216A/ko not_active Ceased
- 2002-01-10 CA CA002435121A patent/CA2435121A1/en not_active Abandoned
- 2002-01-10 CN CNA028036840A patent/CN1486178A/zh active Pending
- 2002-01-10 IL IL15608702A patent/IL156087A0/xx unknown
- 2002-01-10 PL PL02362793A patent/PL362793A1/xx not_active Application Discontinuation
- 2002-01-10 EE EEP200300335A patent/EE200300335A/xx unknown
- 2002-01-10 MX MXPA03006408A patent/MXPA03006408A/es unknown
- 2002-01-10 JP JP2002557379A patent/JP2004517883A/ja not_active Withdrawn
- 2002-01-10 CZ CZ20031853A patent/CZ20031853A3/cs unknown
- 2002-01-10 EA EA200300537A patent/EA200300537A1/ru unknown
- 2002-01-10 BR BR0206502-9A patent/BR0206502A/pt not_active IP Right Cessation
- 2002-01-10 WO PCT/IB2002/000042 patent/WO2002056871A2/en not_active Ceased
- 2002-01-10 EP EP02732099A patent/EP1353657A1/en not_active Withdrawn
- 2002-01-10 HU HU0302767A patent/HUP0302767A2/hu unknown
- 2002-01-10 OA OA1200300174A patent/OA12440A/en unknown
- 2002-01-11 DO DO2002000325A patent/DOP2002000325A/es unknown
- 2002-01-14 PA PA20028537101A patent/PA8537101A1/es unknown
- 2002-01-16 AR ARP020100145A patent/AR032101A1/es not_active Application Discontinuation
- 2002-01-16 TN TNTNSN02003A patent/TNSN02003A1/fr unknown
- 2002-01-16 GT GT200200003A patent/GT200200003A/es unknown
- 2002-01-16 SV SV2002000849A patent/SV2003000849A/es not_active Application Discontinuation
- 2002-01-17 AP APAP/P/2002/002401A patent/AP2002002401A0/en unknown
-
2003
- 2003-05-15 IS IS6818A patent/IS6818A/is unknown
- 2003-05-21 BG BG107834A patent/BG107834A/bg unknown
- 2003-05-22 CR CR6983A patent/CR6983A/es not_active Application Discontinuation
- 2003-05-29 ZA ZA200304180A patent/ZA200304180B/en unknown
- 2003-07-11 MA MA27233A patent/MA26980A1/fr unknown
- 2003-07-16 NO NO20033223A patent/NO20033223D0/no not_active Application Discontinuation
- 2003-07-17 EC EC2003004692A patent/ECSP034692A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IS6818A (is) | 2003-05-15 |
| IL156087A0 (en) | 2003-12-23 |
| NO20033223L (no) | 2003-07-16 |
| HUP0302767A2 (hu) | 2003-11-28 |
| AP2002002401A0 (en) | 2002-03-31 |
| PL362793A1 (en) | 2004-11-02 |
| CZ20031853A3 (cs) | 2004-07-14 |
| EP1353657A1 (en) | 2003-10-22 |
| CR6983A (es) | 2003-11-25 |
| OA12440A (en) | 2006-05-22 |
| GB0101223D0 (en) | 2001-02-28 |
| BR0206502A (pt) | 2003-10-21 |
| GT200200003A (es) | 2002-08-19 |
| AR032101A1 (es) | 2003-10-22 |
| BG107834A (bg) | 2004-01-30 |
| EE200300335A (et) | 2003-12-15 |
| EA200300537A1 (ru) | 2004-02-26 |
| MXPA03006408A (es) | 2003-10-15 |
| CN1486178A (zh) | 2004-03-31 |
| SV2003000849A (es) | 2003-01-13 |
| NO20033223D0 (no) | 2003-07-16 |
| SK8572003A3 (en) | 2004-07-07 |
| CA2435121A1 (en) | 2002-07-25 |
| WO2002056871A2 (en) | 2002-07-25 |
| TNSN02003A1 (fr) | 2005-12-23 |
| JP2004517883A (ja) | 2004-06-17 |
| PA8537101A1 (es) | 2002-08-29 |
| KR20030069216A (ko) | 2003-08-25 |
| ZA200304180B (en) | 2004-06-15 |
| MA26980A1 (fr) | 2004-12-20 |
| DOP2002000325A (es) | 2003-01-31 |
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